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CSF-1R

CSF-1R

Os inibidores de CSF-1R são compostos que visam e inibem o receptor do Fator Estimulante de Colônias 1 (CSF-1R), uma tirosina quinase receptora envolvida na regulação de macrófagos e outras células imunológicas. A inibição de CSF-1R tem potencial terapêutico em doenças caracterizadas por atividade excessiva de macrófagos, como câncer, inflamação e distúrbios autoimunes. Na CymitQuimica, oferecemos inibidores de CSF-1R para apoiar sua pesquisa em imunologia, oncologia e inflamação.

Foram encontrados 42 produtos de "CSF-1R"

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  • Anti-CSF1R Antibody (5C535)


    <p>Anti-CSF1R Antibody (5C535) is a Rabbit antibody targeting CSF1R. Anti-CSF1R Antibody (5C535) can be used in ELISA.</p>
    Cor e Forma:Odour Liquid
  • Anti-CSF1R Antibody (1R707)


    <p>Anti-CSF1R Antibody (1R707) is a Rabbit antibody targeting CSF1R. Anti-CSF1R Antibody (1R707) can be used in ELISA.</p>
    Cor e Forma:Odour Liquid
  • Anti-CSF1R Antibody (2I506)


    <p>Anti-CSF1R Antibody (2I506) is a Mouse antibody targeting CSF1R. Anti-CSF1R Antibody (2I506) can be used in ELISA.</p>
    Cor e Forma:Odour Liquid
  • Anti-CSF1R Antibody-FITC (4Y587)


    <p>Anti-CSF1R Antibody-FITC (4Y587) is a FITC-conjugated Mouse antibody targeting CSF1R. Anti-CSF1R Antibody-FITC (4Y587) can be used in FCM.</p>
    Cor e Forma:Odour Liquid
  • Anti-CSF1R Antibody (7V18)


    <p>Anti-CSF1R Antibody (7V18) is a Rabbit antibody targeting CSF1R. Anti-CSF1R Antibody (7V18) can be used in ELISA.</p>
    Cor e Forma:Odour Liquid
  • Anti-CSF1R Antibody (5B661)


    <p>Anti-CSF1R Antibody (5B661) is a Mouse antibody targeting CSF1R. Anti-CSF1R Antibody (5B661) can be used in ELISA,ELISA(Cap).</p>
    Cor e Forma:Odour Liquid
  • PLX5622

    CAS:
    <p>PLX5622 is a selective, orally active and blood-brain barrier permeable CSF1R inhibitor. PLX5622 induces elimination of microglia. Cost effective and quality assured.</p>
    Fórmula:C21H19F2N5O
    Pureza:98% - 99.92%
    Cor e Forma:Solid
    Peso molecular:395.41
  • Sotuletinib

    CAS:
    <p>Sotuletinib (BLZ945) is an orally active, effective and specific CSF-1R inhibitor, &gt;1000-fold selective against its closest receptor tyrosine kinase homologs.</p>
    Fórmula:C20H22N4O3S
    Pureza:97.43% - 99.82%
    Cor e Forma:Solid
    Peso molecular:398.48
  • Ki20227

    CAS:
    <p>Ki-20227 is a specific c-Fms tyrosine kinase(CSF1R) inhibitor (IC50: 2 nM).</p>
    Fórmula:C24H24N4O5S
    Pureza:98.97% - 99.88%
    Cor e Forma:Solid
    Peso molecular:480.54
  • cFMS Receptor Inhibitor II

    CAS:
    <p>cFMS Receptor Inhibitor II is a CSF1R kinase inhibitor</p>
    Fórmula:C23H20N4O
    Pureza:99.8%
    Cor e Forma:Solid
    Peso molecular:368.43
  • AZD7507

    CAS:
    <p>AZD7507 is a CSF-1R inhibitor with an IC50 of 32 nM. AZD7507 has antitumor activity.</p>
    Fórmula:C23H27FN6O3
    Pureza:99.55% - 99.78%
    Cor e Forma:Solid
    Peso molecular:454.5
  • PF 477736

    CAS:
    <p>PF 477736 (PF-736,PF-00477736) is a specifc, effective and ATP-competitive Chk1 inhibitor (Ki: 0.49 nM ) and also inhibits FGFR3, Aurora-A, VEGFR2, Flt3, Fms (</p>
    Fórmula:C22H25N7O2
    Pureza:97.58% - 99.94%
    Cor e Forma:Solid
    Peso molecular:419.48
  • GW2580

    CAS:
    <p>GW2580 (SC-203877) is a specific, oral-bioavailable CSF-1R inhibitor for c-FMS.</p>
    Fórmula:C20H22N4O3
    Pureza:99.48% - >99.99%
    Cor e Forma:Solid
    Peso molecular:366.41
  • OSI-930

    CAS:
    <p>OSI-930 is an oral c-Kit/VEGFR-2 inhibitor targeting tumor growth and angiogenesis.</p>
    Fórmula:C22H16F3N3O2S
    Pureza:99.67%
    Cor e Forma:Solid
    Peso molecular:443.44
  • Dovitinib

    CAS:
    <p>Dovitinib is an orally active, multi-targeted tyrosine kinase (RTK) inhibitor with anti-tumor effects.Cost-effective and quality-assured.</p>
    Fórmula:C21H21FN6O
    Pureza:99.35% - 99.92%
    Cor e Forma:Solid
    Peso molecular:392.43
  • Linifanib

    CAS:
    <p>Linifanib (AL-39324) (ABT-869) is a novel, potent ATP-competitive VEGFR/PDGFR inhibitor for KDR (IC50: 4 nM), CSF-1R (IC50: 3 nM), Flt-1/3 (IC50: 3/4 nM) and</p>
    Fórmula:C21H18FN5O
    Pureza:98% - 98.24%
    Cor e Forma:Solid
    Peso molecular:375.4
  • Pexidartinib

    CAS:
    <p>Pexidartinib (PLX-3397) is a capsule formulation containing a small-molecule receptor tyrosine kinase (RTK) inhibitor of KIT, CSF1R and FLT3 with potential</p>
    Fórmula:C20H15ClF3N5
    Pureza:98.34% - 99.45%
    Cor e Forma:Solid
    Peso molecular:417.81
  • PRN1371

    CAS:
    <p>PRN1371 is a specific and potent FGFR1-4 and CSF1R inhibitor (IC50s: 0.6/1.3/4.1/19.3/8.1 nM for FGFR1/2/3/4 and CSF1R).</p>
    Fórmula:C26H30Cl2N6O4
    Pureza:98.65%
    Cor e Forma:Solid
    Peso molecular:561.46
  • Vimseltinib

    CAS:
    <p>Vimseltinib (DCC-3014) is a c-FMS (CSF-IR) and c-Kit dual inhibitor (IC50s: &lt;0.01 μM and 0.1-1 μM).</p>
    Fórmula:C23H25N7O2
    Pureza:99.05% - 99.57%
    Cor e Forma:Solid
    Peso molecular:431.49
  • GW786034B

    CAS:
    <p>Pazopanib HCl (Votrient) inhibits VEGFR1-3, PDGFR, FGFR, c-Kit, c-Fms with IC50 range 10-146 nM in cell-free assays.</p>
    Fórmula:C21H23N7O2S·HCl
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:473.98