Receptor de Histamina
Os receptores de histamina são GPCRs que mediam os efeitos da histamina, uma amina biogênica envolvida em respostas imunológicas, secreção de ácido gástrico e neurotransmissão. Existem quatro subtipos de receptores de histamina (H1, H2, H3 e H4), cada um desempenhando papéis distintos em reações alérgicas, função gástrica e atividade do sistema nervoso central. Antagonistas dos receptores de histamina são amplamente utilizados no tratamento de alergias, úlceras pépticas e enjoo de movimento. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores de histamina de alta qualidade para apoiar sua pesquisa em imunologia, gastroenterologia e neurofarmacologia.
Foram encontrados 358 produtos de "Receptor de Histamina"
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Dimenhydrinate
CAS:<p>Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.</p>Fórmula:C24H28ClN5O3Pureza:99.57% - 99.77%Cor e Forma:Crystals Physical Description Crystalline White Powder (Ntp 1992)Peso molecular:469.96Pimethixene
CAS:<p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>Fórmula:C19H19NSPureza:97.50%Cor e Forma:SolidPeso molecular:293.43Histamine
CAS:<p>Histamine (Ergamine) is an amine derived by the enzymatic decarboxylation of histamine. Histamine is a potent stimulant of gastric secretion of central action. High-Quality, Low-Cost!</p>Fórmula:C5H9N3Pureza:96.63% - >99.99%Cor e Forma:Needles From Chloroform SolidPeso molecular:111.15Levodropropizine
CAS:<p>Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.</p>Fórmula:C13H20N2O2Pureza:99.87% - 99.93%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:236.31Astemizole
CAS:<p>Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.</p>Fórmula:C28H31FN4OPureza:98.24% - 99.67%Cor e Forma:White Crystals SolidPeso molecular:458.57Chloropyramine hydrochloride
CAS:<p>Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.</p>Fórmula:C16H20ClN3·HClPureza:99.45% - 99.8%Cor e Forma:SolidPeso molecular:326.26Azacyclonol
CAS:<p>Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.</p>Fórmula:C18H21NOPureza:99.46%Cor e Forma:Solid PowderPeso molecular:267.37Lafutidine
CAS:<p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>Fórmula:C22H29N3O4SPureza:98.55%Cor e Forma:Yellowish White Crystalline PowderPeso molecular:431.55Amodiaquine dihydrochloride dihydrate
CAS:<p>Amodiaquine dihydrochloride dihydrate (Amodiaquin hydrochloride) is an orally active 4-aminoquinoline derivative with antimalarial and anti-inflammatory effects</p>Fórmula:C20H28Cl3N3O3Pureza:99.97%Cor e Forma:SolidPeso molecular:464.82Antazoline hydrochloride
CAS:<p>Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous</p>Fórmula:C17H19N3·HClPureza:98% - 99.53%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:301.82Brompheniramine maleate
CAS:<p>Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.</p>Fórmula:C16H19BrN2·C4H4O4Pureza:99.80%Cor e Forma:Crystal PowderPeso molecular:435.31Fexofenadine hydrochloride
CAS:<p>Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with</p>Fórmula:C32H40ClNO4Pureza:>99.99%Cor e Forma:White Crystalline PowderPeso molecular:538.12Perphenazine
CAS:<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Fórmula:C21H26ClN3OSPureza:99.3% - 99.99%Cor e Forma:SolidPeso molecular:403.97Fenspiride hydrochloride
CAS:<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Fórmula:C15H20N2O2·HClPureza:99.64% - 99.92%Cor e Forma:SolidPeso molecular:296.79Tripelennamine hydrochloride
CAS:<p>Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.</p>Fórmula:C16H21N3·HClPureza:99.54% - 99.81%Cor e Forma:White SolidPeso molecular:291.82Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Fórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Cor e Forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53Famotidine
CAS:<p>Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.</p>Fórmula:C8H15N7O2S3Pureza:98.93% - 99.91%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:337.45Rupatadine Fumarate
CAS:<p>Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM.</p>Fórmula:C26H26ClN3·C4H4O4Pureza:99.86%Cor e Forma:White Or Almost-White PowderPeso molecular:532.03Ketotifen fumarate
CAS:<p>Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.</p>Fórmula:C23H23NO5SPureza:99.25% - 99.73%Cor e Forma:SolidPeso molecular:425.50Chlorprothixene hydrochloride
CAS:<p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>Fórmula:C18H18ClNS·HClPureza:99.76%Cor e Forma:White PowderPeso molecular:352.32Diphenylpyraline hydrochloride
CAS:<p>Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.</p>Fórmula:C19H23NO·HClPureza:98.72%Cor e Forma:SolidPeso molecular:317.85Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine（IC50=6.5 nM） and cholinergic（IC50=10 nM）.</p>Fórmula:C28H30N2O8Pureza:99.7% - >99.99%Cor e Forma:PowderPeso molecular:522.55Mepyramine maleate
CAS:<p>Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.</p>Fórmula:C21H27N3O5Pureza:99.51% - 99.7%Cor e Forma:White Crystalline PowderPeso molecular:401.47Dexchlorpheniramine Maleate
CAS:<p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>Fórmula:C20H23ClN2O4Pureza:99.58%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:390.86Cyproheptadine hydrochloride sesquihydrate
CAS:<p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>Fórmula:C21H24ClNOPureza:99.77% - >99.99%Cor e Forma:White To Slightly Yellowish Crystalline SolidPeso molecular:341.88Cimetidine
CAS:<p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>Fórmula:C10H16N6SPureza:99.82%Cor e Forma:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Peso molecular:252.34Mifentidine
CAS:<p>Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.</p>Fórmula:C13H16N4Pureza:98.34% - 99.73%Cor e Forma:SolidPeso molecular:228.29Promethazine hydrochloride
CAS:<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Fórmula:C17H20N2S·HClPureza:99.85%Cor e Forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecular:320.88Doxylamine succinate
CAS:<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Fórmula:C21H28N2O5Pureza:99.61%Cor e Forma:5 1 (Ntp 1992)Peso molecular:388.46Mebhydrolin napadisylate
CAS:<p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>Fórmula:C19H20N2C10H8O6S2Pureza:99.35% - 99.96%Cor e Forma:White Or Almost White CrystallinePeso molecular:420.52Mizolastine
CAS:<p>Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever and hives.</p>Fórmula:C24H25FN6OPureza:98% - 99.75%Cor e Forma:SolidPeso molecular:432.49Terfenadine
CAS:<p>Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.</p>Fórmula:C32H41NO2Pureza:98.76% - 99.75%Cor e Forma:SolidPeso molecular:471.67Doxepin hydrochloride
CAS:<p>Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.</p>Fórmula:C19H22ClNOPureza:99.65% - 99.91%Cor e Forma:White To Off-White PowderPeso molecular:315.84Triprolidine hydrochloride monohydrate
CAS:<p>Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.</p>Fórmula:C19H25ClN2OPureza:99.68% - 99.81%Cor e Forma:White Crystalline PowderPeso molecular:332.87Talastine
CAS:<p>Talastine is an antihistamine compound that can induce an allergic rash.</p>Fórmula:C19H21N3OPureza:98.50% - 99.44%Cor e Forma:SolidPeso molecular:307.39Pheniramine maleate
CAS:<p>Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.</p>Fórmula:C16H20N2·C4H4O4Pureza:99.85%Cor e Forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CPeso molecular:356.42Cetirizine dihydrochloride
CAS:<p>Cetirizine dihydrochloride is a potent non-drowsy antihistamine for allergies and asthma.</p>Fórmula:C21H27Cl3N2O3Pureza:99.4% - 99.97%Cor e Forma:SolidPeso molecular:461.81Hydroxyzine Pamoate
CAS:<p>Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.</p>Fórmula:C44H43ClN2O8Pureza:99.49%Cor e Forma:SolidPeso molecular:763.27Ranitidine Hydrochloride
CAS:<p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>Fórmula:C13H23ClN4O3SPureza:99.30% - 99.49%Cor e Forma:SolidPeso molecular:350.86Carbinoxamine Maleate Salt
CAS:<p>Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.</p>Fórmula:C20H23ClN2O5Pureza:99.97%Cor e Forma:Off-White SolidPeso molecular:406.86Cinnarizine
CAS:<p>Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.</p>Fórmula:C26H28N2Pureza:99.94%Cor e Forma:SolidPeso molecular:368.51Meclizine dihydrochloride
CAS:<p>Meclizine dihydrochloride (NSC28728) is a histamine H1 antagonist used in the treatment of motion sickness, vertigo, and nausea during pregnancy and radiation</p>Fórmula:C25H27ClN2·2HClPureza:98.05% - 99.79%Cor e Forma:White Slightly Yellowish Crystalline PowderPeso molecular:463.87Levocetirizine
CAS:<p>Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.</p>Fórmula:C21H25ClN2O3Pureza:98% - 99.9%Cor e Forma:White PowderPeso molecular:388.89JNJ-39758979
CAS:<p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>Fórmula:C11H19N5Pureza:98.33% - 99.62%Cor e Forma:SolidPeso molecular:221.3Orphenadrine hydrochloride
CAS:<p>Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.</p>Fórmula:C18H23NO·HClPureza:99.88%Cor e Forma:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Peso molecular:305.85MK-0249 FA
<p>MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.</p>Fórmula:C24H26F3N3O4Pureza:99.98%Cor e Forma:SolidPeso molecular:477.48Pemirolast potassium
CAS:<p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>Fórmula:C10H7KN6OPureza:98.91% - 99.63%Cor e Forma:Crystals From Dimethylformamide Crystalline SolidPeso molecular:266.31Clemastine fumarate
CAS:<p>Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.</p>Fórmula:C25H30ClNO5Pureza:99.52% - >99.99%Cor e Forma:Colorless To Faintly Yellow Crystalline Powder Appearance White Or Almost White Crystalline PowderPeso molecular:459.97Roxatidine Acetate hydrochloride
CAS:<p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>Fórmula:C19H29ClN2O4Pureza:99.49%Cor e Forma:SolidPeso molecular:384.9Loratadine
CAS:<p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>Fórmula:C22H23ClN2O2Pureza:99.71% - 99.98%Cor e Forma:White PowderPeso molecular:382.88
