Receptor de Histamina
Os receptores de histamina são GPCRs que mediam os efeitos da histamina, uma amina biogênica envolvida em respostas imunológicas, secreção de ácido gástrico e neurotransmissão. Existem quatro subtipos de receptores de histamina (H1, H2, H3 e H4), cada um desempenhando papéis distintos em reações alérgicas, função gástrica e atividade do sistema nervoso central. Antagonistas dos receptores de histamina são amplamente utilizados no tratamento de alergias, úlceras pépticas e enjoo de movimento. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores de histamina de alta qualidade para apoiar sua pesquisa em imunologia, gastroenterologia e neurofarmacologia.
Foram encontrados 385 produtos de "Receptor de Histamina"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Betahistine
CAS:<p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>Fórmula:C8H12N2Pureza:99.87% - 99.87%Cor e Forma:Yellowish Liquid Liquid LiquidPeso molecular:136.19Buclizine dihydrochloride
CAS:Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic andFórmula:C28H33ClN2·2HClPureza:98.05%Cor e Forma:Off-White PowderPeso molecular:505.95S 38093
CAS:S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).Fórmula:C17H24N2O2Pureza:99.95%Cor e Forma:SolidPeso molecular:288.38Dioxopromethazine
CAS:Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.Fórmula:C17H20N2O2SPureza:98%Cor e Forma:SolidPeso molecular:316.42Carcinine ditrifluoroacetate Acetate
Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.Fórmula:C14H20F6N4O7Pureza:98.18%Cor e Forma:SolidPeso molecular:470.32Decloxizine dihydrochloride
CAS:<p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>Fórmula:C21H28N2O2·2ClHPureza:99.73%Cor e Forma:SolidPeso molecular:413.39Histamine Phosphate
CAS:Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.Fórmula:C5H9N·2H3O4PPureza:>99.99%Cor e Forma:White Crystal PowderPeso molecular:307.14Alginic acid
CAS:Alginic acid, a polysaccharide from brown seaweed, has anti-anaphylactic and anti-inflammatory properties and is used in food industry.Fórmula:C14H22O13Pureza:≥98%Cor e Forma:SolidPeso molecular:398.317Betahistine dihydrochloride
CAS:Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.Fórmula:C8H14Cl2N2Pureza:99.22% - 99.88%Cor e Forma:White To Light Yellow Crystalline PowderPeso molecular:209.12Thonzylamine
CAS:Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.Fórmula:C16H22N4OPureza:99.45%Cor e Forma:SolidPeso molecular:286.37Alimemazine hemitartrate
CAS:Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Fórmula:C18H22N2SC4H6O6Pureza:98.16% - 99.69%Cor e Forma:SolidPeso molecular:448.53JNJ-5207852
CAS:JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.Fórmula:C20H32N2OPureza:97.19%Cor e Forma:SolidPeso molecular:316.48LML134
CAS:LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).Fórmula:C19H29N5O3Pureza:99.36%Cor e Forma:SolidPeso molecular:375.47S 38093 HCl
CAS:S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.Fórmula:C17H25ClN2O2Pureza:97.91%Cor e Forma:SolidPeso molecular:324.85Hydroxyzine dihydrochloride
CAS:<p>Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.</p>Fórmula:C21H27ClN2O2·2HClPureza:99.46% - 99.79%Cor e Forma:Oil PowderPeso molecular:447.83OXOMEMAZINE
CAS:Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Fórmula:C18H22N2O2SPureza:99.58%Cor e Forma:SolidPeso molecular:330.44Ranitidine
CAS:Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).Fórmula:C13H22N4O3SPureza:99.52%Cor e Forma:Solid SolidPeso molecular:314.40Bepotastine
CAS:Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.Fórmula:C21H25ClN2O3Pureza:99.75%Cor e Forma:SolidPeso molecular:388.89Latrepirdine dihydrochloride
CAS:Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Fórmula:C21H25N3·2HClPureza:98.45%Cor e Forma:SolidPeso molecular:392.37Levocetirizine Dihydrochloride
CAS:<p>Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.</p>Fórmula:C21H27Cl3N2O3Pureza:99.89%Cor e Forma:White Or Off-White Crystalline PowderPeso molecular:461.81
