Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 297 produtos de "Receptor opioide"
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Allyphenyline oxalate
CAS:<p>The pKi values of Allyphenyline oxalate (compound 9) for the α2-adrenergic receptor subtypes α2A, α2B, and α2C are 7.24, 6.47, and 7.07, respectively.</p>Fórmula:C16H20N2O5Cor e Forma:SolidPeso molecular:320.34rel-SB-612111 hydrochloride
CAS:<p>NOP receptor antagonist</p>Fórmula:C24H30Cl3NOPureza:98%Cor e Forma:SolidPeso molecular:454.86Naldemedine tosylate
CAS:<p>Naldemedine (S-297995) tosylate, a PAMORA, targets μ-, δ-, κ-opioid receptors, aiding OIC research, may bind to SARS-CoV2's 3CL pro.</p>Fórmula:C39H42N4O9SCor e Forma:SolidPeso molecular:742.84(S)-MCOPPB
CAS:<p>(S)-MCOPPB is the S-enantiomer of MCOPPB, an orally active selective agonist for the Nociceptin/Orphanin FQ-Receptor. It inhibits signal transduction in mouse brain NOP receptors and is utilized in anxiety disorder research.</p>Fórmula:C26H40N4Cor e Forma:SolidPeso molecular:408.623Opioid receptor antagonist 1
CAS:<p>Opioid receptor antagonist 1 (Compound 10) is an Orvinol-based antagonist of opioid receptors. It exhibits activity as an antagonist against the analgesic properties of morphine.</p>Fórmula:C24H29ClF3NO4Cor e Forma:SolidPeso molecular:487.94Naltrindole 5′-isothiocyanate
CAS:<p>Naltrindole 5′-isothiocyanate (5'-NTII) is an irreversible delta opioid receptor antagonist that counters the analgesic effects induced by DSLET without altering the effects caused by DPDPE.</p>Fórmula:C27H25N3O3SCor e Forma:SolidPeso molecular:471.571Bromadoline
CAS:<p>Bromadoline is an opioid compound that exhibits anti-nociceptive properties in rodents.</p>Fórmula:C15H21BrN2OCor e Forma:SolidPeso molecular:325.244KNT-127
CAS:<p>KNT-127 is an agonist of δ-Opioid receptor.</p>Fórmula:C24H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:372.46(±)-J 113397
CAS:<p>(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM).</p>Fórmula:C24H37N3O2Cor e Forma:SolidPeso molecular:399.575′-Guanidinonaltrindole
CAS:<p>5′-Guanidinonaltrindole (GNTI) is a selective antagonist of the kappa opioid receptor.</p>Fórmula:C27H29N5O3Cor e Forma:SolidPeso molecular:471.551GNTI dihydrochloride
CAS:<p>κ opioid receptor antagonist</p>Fórmula:C27H30ClN5O3Pureza:98%Cor e Forma:SolidPeso molecular:508.01Sunobinop
CAS:<p>Sunobinop (S 117957) is an opioid receptor-like orphan receptor (ORL1) modulator.</p>Fórmula:C26H33N3O3Cor e Forma:SolidPeso molecular:435.56σ1 Receptor/μ Opioid receptor modulator 2
CAS:<p>Compound 4x, also known as σ1 Receptor/μOpioid receptormodulator 2, acts as a μOR agonist and a σ1R antagonist, exhibiting a potent μOR EC50 of 0.6 nM and strong σ1R inhibitory activity (Ki: 363.7 nM). It demonstrates significant analgesic effects in various pain models.</p>Fórmula:C23H31N3OPeso molecular:365.51Norbinaltorphimine dihydrochloride
CAS:<p>Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.</p>Fórmula:C40H45Cl2N3O6Pureza:98.17% - 99.88%Cor e Forma:SolidPeso molecular:734.71BU72
CAS:<p>BU72 is a potent, long-lasting agonist for μ and κ opioid receptors, with partial agonistic activity at the δ opioid receptor (EC50 values of 0.054, 0.033, and 0.58 nM, respectively). It provides strong, enduring analgesic effects primarily mediated through μ opioid receptors. BU72 also exhibits a prolonged duration of activity and can partially reverse morphine-induced analgesia. It is applicable in studies of opioid dependence.</p>Fórmula:C28H32N2O2Cor e Forma:SolidPeso molecular:428.57Riminkefon
CAS:<p>Riminkefon is a kappa opioid receptor agonist .</p>Fórmula:C38H57N7O6Cor e Forma:SolidPeso molecular:707.9JDTic Dihydrochloride
CAS:JDTic Dihydrochloride is a high-affinity and selective κ-opioid receptor (KOR) antagonist that blocks dynorphin-KOR signalling,antidepressant.Fórmula:C28H41Cl2N3O3Pureza:98%Cor e Forma:SolidPeso molecular:538.55Mu opioid receptor antagonist 8
CAS:<p>Muopioid Receptor Antagonist 8 (368) serves as an antagonist to the μ-opioid receptor, significantly inhibiting the activation of Gi induced by met-enkephalin at the µOR.</p>Fórmula:C36H35N3O4SCor e Forma:SolidPeso molecular:605.756β-Naltrexol
CAS:<p>6β-Naltrexol is a peripherally selective opioid antagonist that reduces constipation from opioids while minimizing central nervous system effects.</p>Fórmula:C20H25NO4Pureza:99.933%Cor e Forma:SolidPeso molecular:343.42DS34942424
<p>DS34942424 is an orally potent analgesic which did not exhibit mu opioid receptor agonist activity.</p>Fórmula:C15H17FN2OCor e Forma:SolidPeso molecular:260.31
