Receptor opioide
Os receptores opioides são um grupo de receptores acoplados à proteína G que mediam os efeitos dos opioides endógenos e exógenos. Estes receptores desempenham um papel central na modulação da dor, regulação do humor e comportamentos aditivos. Agonistas e antagonistas dos receptores opioides são amplamente utilizados no manejo da dor e tratamento de dependências, bem como em pesquisas sobre distúrbios neurológicos e psiquiátricos. Na CymitQuimica, oferecemos uma seleção abrangente de moduladores de receptores opioides de alta qualidade para apoiar sua pesquisa em neurobiologia, manejo da dor e terapia de dependência.
Foram encontrados 297 produtos de "Receptor opioide"
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Mu opioid receptor antagonist 5
<p>Compound NAP: MOR antagonist, crosses blood-brain barrier, EC50: 1.14 nM, Ki: 0.37 nM, useful for OUD research.</p>Fórmula:C26H29N3O4Cor e Forma:SolidPeso molecular:447.53BW 443C
CAS:<p>BW 443C is a selective agonist of mu-opioid receptor.</p>Fórmula:C33H46N10O10Cor e Forma:SolidPeso molecular:742.791Mu opioid receptor antagonist 2
<p>Compound 25: potent, selective MOR antagonist, crosses blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM), for OUD research.</p>Fórmula:C25H28N2O4SCor e Forma:SolidPeso molecular:452.57SB-612111
CAS:<p>SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.</p>Fórmula:C24H29Cl2NOCor e Forma:SolidPeso molecular:418.40Isotodesnitazene
CAS:<p>Isotodesnitazene is an opioid compound that primarily targets the μ-opioid receptor (MOR). It exhibits EC50 values of 34.8 nM and 142 nM for MOR-βarr2 and MOR-mini-Gi, respectively. Isotodesnitazene can be utilized for research in opioid drugs.</p>Fórmula:C23H31N3OCor e Forma:SolidPeso molecular:365.51Anilopam
CAS:<p>Anilopam is an opioid analgesic belonging to the benzazepine class and acts as an agonist at opioid receptors.</p>Fórmula:C20H26N2OCor e Forma:SolidPeso molecular:310.4322-Thiocyanatosalvinorin A
CAS:<p>22-Thiocyanatosalvinorin A (RB-64) is a potent selective agonist for the kappa-opioid receptor, exhibiting an EC50 value of 0.077 nM.</p>Fórmula:C24H27NO8SCor e Forma:SolidPeso molecular:489.54CCG258747
CAS:<p>CCG258747 is a novel, selective inhibitor of the GRK2 subfamily.</p>Fórmula:C28H27FN4O4Cor e Forma:SolidPeso molecular:502.54BNTX maleate
CAS:<p>δ1 opioid receptor antagonist</p>Fórmula:C31H31NO8Pureza:98%Cor e Forma:SolidPeso molecular:545.58Daeatal
CAS:<p>Dynorphin A ethylamide (1-9), the opioid activities were examined in the bioassays.</p>Fórmula:C56H93N19O10Pureza:98%Cor e Forma:SolidPeso molecular:1192.46Nalmefene
CAS:<p>Nalmefene (ORF 11676) is a μ-opioid antagonist and partial κ agonist used in the study of opioid overdose and alcohol dependence.</p>Fórmula:C21H25NO3Pureza:99.86%Cor e Forma:SolidPeso molecular:339.43Propiram fumarate HCl
CAS:<p>Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.</p>Fórmula:C16H25N3O·xClHPureza:99.25%Cor e Forma:SoildSR17018
CAS:<p>SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.</p>Fórmula:C19H18Cl3N3OPureza:99.89%Cor e Forma:SolidPeso molecular:410.72Cebranopadol
CAS:<p>Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP)</p>Fórmula:C24H27FN2OPureza:98.32% - 99.78%Cor e Forma:SolidPeso molecular:378.48Bromadoline maleate
CAS:<p>Bromadoline is an opioid analgesic selective for the μ-opioid receptor.</p>Fórmula:C19H25BrN2O5Pureza:98%Cor e Forma:SolidPeso molecular:441.322SR14150
CAS:<p>SR14150 is a partial agonist of high-affinity NOP receptor.</p>Fórmula:C21H30N2OPureza:98%Cor e Forma:SolidPeso molecular:326.48MOR agonist-1
CAS:<p>MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associated</p>Fórmula:C22H26ClFN2O2Pureza:98%Cor e Forma:SolidPeso molecular:404.91
