
Receptor Glucagon
Os receptores de glucagon são GPCRs que mediam os efeitos do glucagon, um hormônio envolvido na regulação da homeostase da glicose, promovendo a quebra de glicogênio e a liberação de glicose pelo fígado. Esses receptores são críticos na gestão dos níveis de açúcar no sangue e são de particular interesse no estudo do diabetes e distúrbios metabólicos. Antagonistas dos receptores de glucagon estão sendo explorados como potenciais tratamentos para hiperglicemia no diabetes tipo 2. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores de glucagon de alta qualidade para apoiar sua pesquisa em endocrinologia, diabetes e regulação metabólica.
Foram encontrados 164 produtos de "Receptor Glucagon"
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Anti-GCGR Antibody (7J909)
<p>Anti-GCGR Antibody (7J909) is an antibody targeting GCGR. Anti-GCGR Antibody (7J909) can be used in ELISA.</p>Cor e Forma:Odour LiquidSCO-267
CAS:<p>SCO-267 is a full agonist of GPR40/FFAR1, stimulating insulin secretion and GLP-1 release in diabetic rats, improving glucose tolerance,type 2 diabetes.</p>Fórmula:C36H46N4O5Pureza:99.89%Cor e Forma:SolidPeso molecular:614.77GLP-1R modulator C5
CAS:<p>GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.</p>Fórmula:C24H21NO3Pureza:99.59%Cor e Forma:SolidPeso molecular:371.43Liraglutide
CAS:<p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>Fórmula:C172H265N43O51Pureza:97.65% - 99.04%Cor e Forma:SolidPeso molecular:3751.25PF-06882961 Tris
CAS:<p>PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>Fórmula:C35H41FN6O7Pureza:98.74% - 99.79%Cor e Forma:SolidPeso molecular:676.7GRA Ex-25
CAS:<p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>Fórmula:C29H36F3N3O5Pureza:98.2% - 98.88%Cor e Forma:SolidPeso molecular:563.61Shanzhiside methyl ester
CAS:<p>Shanzhiside methylester soothes neuropathic pain by triggering spinal GLP-1 receptors, boosting microglial β-endorphin through p38 MAPK.</p>Fórmula:C17H26O11Pureza:98.998% - 99.32%Cor e Forma:SolidPeso molecular:406.38Lixisenatide acetate (320367-13-3 free base)
CAS:<p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>Fórmula:C215H347N61O65S·6C2H4O2Pureza:98% - 99.9%Cor e Forma:SolidPeso molecular:5218.88BETP
CAS:<p>BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).</p>Fórmula:C20H17F3N2O2SPureza:98.51%Cor e Forma:SolidPeso molecular:406.42HAEGTFTSDVSSYLE
<p>HAEGTFTSDVSSYLE is a peptide. GLP-I analog contains the sequence.</p>Fórmula:C71H103N17O28Pureza:>99.99%Cor e Forma:SolidPeso molecular:1642.71GLP-1(7-36), amide
CAS:<p>GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.</p>Fórmula:C149H226N40O45Pureza:99.85%Cor e Forma:White PowderPeso molecular:3297.63Exendin-4
CAS:<p>Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.</p>Fórmula:C184H282N50O60SPureza:97.71% - 99.78%Cor e Forma:SolidPeso molecular:4186.57Semaglutide
CAS:<p>Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).</p>Fórmula:C187H291N45O59Pureza:96.92% - 99.78%Cor e Forma:SolidPeso molecular:4114Exendin-4 acetate
CAS:<p>Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).</p>Fórmula:C186H286N50O62SPureza:98.48% - 99.78%Cor e Forma:SolidPeso molecular:4247Oxyntomodulin acetate
<p>Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].</p>Pureza:99.24%Cor e Forma:LiquidPeso molecular:N/ABay 55-9837 acetate
<p>Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.</p>Pureza:98.27%Cor e Forma:LiquidPeso molecular:N/ASecretin (33-59), rat
CAS:<p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>Fórmula:C129H216N42O42Pureza:98.12%Cor e Forma:SolidPeso molecular:3027.35Glucagon (19-29), human acetate
<p>Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.</p>Fórmula:C63H93N15O20SPureza:98.11%Cor e Forma:SolidPeso molecular:1412.57HAEGTFT acetate(926018-95-3 free base)
<p>HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.</p>Fórmula:C35H51N9O14Pureza:>99.99%Cor e Forma:SolidPeso molecular:821.84Tirzepatide Acetate(2023788-19-2 free base)
<p>Tirzepatide (LY3298176) Acetate (2023788-19-2 free base) is a new molecule that can control blood glucose levels.Cost-effective and quality-assured.</p>Fórmula:C227H352N48O70Pureza:97.3% - 98.05%Cor e Forma:SolidPeso molecular:4873.5

