Receptor de Bradicinina
Os receptores de bradicinina são GPCRs que mediam os efeitos da bradicinina, um peptídeo envolvido em respostas inflamatórias, sensação de dor e regulação da pressão arterial. Existem dois principais tipos de receptores de bradicinina, B1 e B2, cada um desempenhando papéis distintos em processos fisiopatológicos. Antagonistas dos receptores de bradicinina são usados no tratamento de condições como angioedema hereditário, dor crônica e hipertensão. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores de bradicinina de alta qualidade para apoiar sua pesquisa em inflamação, manejo da dor e biologia cardiovascular.
Foram encontrados 63 produtos para "Receptor de Bradicinina".
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Methionyl-Lysyl-Bradykinin
CAS:Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .Fórmula:C61H94N18O13SCor e Forma:SolidPeso molecular:1319.58Lys-[Des-Arg9]Bradykinin TFA
CAS:Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.Fórmula:C54H75F6N13O15Cor e Forma:SolidPeso molecular:1260.24JMV-1645
CAS:JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.Fórmula:C49H69N13O12SPureza:98%Cor e Forma:SolidPeso molecular:1064.23L 366811
CAS:L 366811 is a potent oxytocin antagonist.Fórmula:C43H56N8O6Cor e Forma:SolidPeso molecular:780.95FR190997
CAS:FR190997 is an agonist of bradykinin B2 receptor.Fórmula:C37H33Cl2N5O5Cor e Forma:SolidPeso molecular:698.59Thrombostatin cont-1
CAS:Thrombostatin cont-1, an analogue of the bradykinin metabolite thrombostatin, has been shown to reduce platelet activation in the canine carotid arteryFórmula:C87H142N34O29S2Peso molecular:2192.4NPC 567 acetate
NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease.Fórmula:C62H91N19O15Pureza:99.81%Cor e Forma:SolidPeso molecular:1342.5Bombinakinin M acetate
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and isFórmula:C102H163N31O26Pureza:99.80%Cor e Forma:White SolidPeso molecular:2239.58Des-Arg9-[Leu8]-Bradykinin acetate
CAS:Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].Fórmula:C43H67N11O12Pureza:98%Cor e Forma:SolidPeso molecular:930.06(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.Fórmula:C52H77N15O14Pureza:97.74%Cor e Forma:SolidPeso molecular:1136.26Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].Fórmula:C47H75N13O11Pureza:98%Cor e Forma:SolidPeso molecular:998.18RPP-(Gly-113C2,15N)-FSPFR TFA
RPP-(Gly-113C2,15N)-FSPFR TFA is a 13C- and 15N-labeled form of bradykinin. Bradykinin is a potent endothelium-dependent vasodilator that can lower blood pressure. It also induces contraction of non-vascular smooth muscles in the bronchi and intestines, increases vascular permeability, and plays a role in pain mechanisms.Breceptin
CAS:Breceptin (B 9870) serves as an antagonist and partial agonist for bradykinin B1/B2 receptors (B1/B2R). In rabbit jugular vein contraction assays, it functions as an irreversible B2R antagonist, inhibiting bradykinin-induced vasoconstriction. B-9870 exhibits partial agonist characteristics in HEK 293 cells with high rabbit B2R expression, activating ERK1/2 phosphorylation, calcium mobilization, arachidonic acid release, and receptor internalization. Breceptin is applicable in research on breast cancer and non-small cell lung cancer inhibition.Fórmula:C136H200N38O28Peso molecular:2815.33Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.Fórmula:C47H66N12O11Pureza:98%Cor e Forma:SolidPeso molecular:975.11Labradimil
CAS:Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Fórmula:C49H75N15O12SPureza:98%Cor e Forma:SolidPeso molecular:1098.29[Des-Arg10]-HOE I40 TFA
[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.Fórmula:C53H77N15O12S·xC2HF3O2Cor e Forma:SolidFasitibant chloride hydrochloride
CAS:Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.Fórmula:C36H50Cl4N6O6SCor e Forma:SolidPeso molecular:836.7Lys-Bradykinin
CAS:Endogenous bradykinin receptor agonistFórmula:C56H85N17O12Pureza:98%Cor e Forma:SolidPeso molecular:1188.38Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Fórmula:C58H89N17O14Pureza:99.98%Cor e Forma:SolidPeso molecular:1248.43Bradykinin (acetate)
CAS:Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Fórmula:C52H77N15O13Pureza:99.68% - >99.99%Cor e Forma:White ViscousPeso molecular:1120.26
![Lys-[Des-Arg9]Bradykinin TFA](https://static.cymitquimica.com/products/TM/thumb-webp/T73646.webp)
![Des-Arg9-[Leu8]-Bradykinin acetate](https://static.cymitquimica.com/products/TM/thumb-webp/T80072.webp)
![Sar-[D-Phe8]-des-Arg9-Bradykinin](https://static.cymitquimica.com/products/TM/thumb-webp/TP1917.webp)
