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Receptor de Bradicinina

Receptor de Bradicinina

Os receptores de bradicinina são GPCRs que mediam os efeitos da bradicinina, um peptídeo envolvido em respostas inflamatórias, sensação de dor e regulação da pressão arterial. Existem dois principais tipos de receptores de bradicinina, B1 e B2, cada um desempenhando papéis distintos em processos fisiopatológicos. Antagonistas dos receptores de bradicinina são usados no tratamento de condições como angioedema hereditário, dor crônica e hipertensão. Na CymitQuimica, oferecemos uma variedade de moduladores de receptores de bradicinina de alta qualidade para apoiar sua pesquisa em inflamação, manejo da dor e biologia cardiovascular.

Foram encontrados 61 produtos de "Receptor de Bradicinina"

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produtos por página.
  • Emorfazone

    CAS:
    Emorfazone (PH011085) has an anti-nociceptive effect.
    Fórmula:C11H17N3O3
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:239.27

    Ref: TM-T9132

    1mg
    84,00€
    1mL*10mM (DMSO)
    152,00€
    5mg
    168,00€
    10mg
    245,00€
    25mg
    404,00€
    50mg
    567,00€
    100mg
    767,00€
    200mg
    1.018,00€
  • ELN-441958

    CAS:
    ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.
    Fórmula:C29H29ClN4O2
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:501.02

    Ref: TM-T2086

    1mg
    58,00€
    5mg
    128,00€
    1mL*10mM (DMSO)
    141,00€
    10mg
    200,00€
    25mg
    339,00€
    50mg
    485,00€
    100mg
    658,00€
    200mg
    889,00€
  • SSR240612

    CAS:
    SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,
    Fórmula:C42H53ClN4O7S
    Pureza:98.59% - 99.16%
    Cor e Forma:Solid
    Peso molecular:793.41

    Ref: TM-T5048

    1mg
    222,00€
    5mg
    512,00€
    1mL*10mM (DMSO)
    612,00€
    10mg
    700,00€
    25mg
    982,00€
    50mg
    1.333,00€
    100mg
    1.783,00€
  • Bradykinin (acetate)

    CAS:
    Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.
    Fórmula:C52H77N15O13
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1120.26

    Ref: TM-T21610

    1mg
    34,00€
    5mg
    58,00€
    10mg
    87,00€
    25mg
    138,00€
    50mg
    207,00€
    100mg
    286,00€
  • Lys-[Des-Arg9]Bradykinin,TFA


    Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2
    Fórmula:C54H75F6N13O15
    Pureza:97.35%
    Cor e Forma:Solid
    Peso molecular:1260.24

    Ref: TM-TP1918L

    1mg
    49,00€
    5mg
    100,00€
    10mg
    149,00€
    25mg
    260,00€
    50mg
    371,00€
    100mg
    530,00€
  • [Des-Arg9]-Bradykinin TFA

    CAS:
    [Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.
    Fórmula:C46H62F3N11O12
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1018.05

    Ref: TM-T8809

    2mg
    34,00€
    5mg
    37,00€
    10mg
    50,00€
    25mg
    94,00€
    50mg
    126,00€
    100mg
    182,00€
    200mg
    264,00€
  • Bradykinin (2-9)

    CAS:
    Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.
    Fórmula:C44H61N11O10
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:904.02

    Ref: TM-TP1181

    1mg
    39,00€
    5mg
    88,00€
    10mg
    130,00€
    1mL*10mM (DMSO)
    144,00€
    25mg
    210,00€
    50mg
    313,00€
    100mg
    464,00€
    200mg
    660,00€
  • R715 TFA(185052-09-9 free base)


    R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).
    Fórmula:C59H82F3N13O14
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1254.36

    Ref: TM-TP1933

    1mg
    141,00€
    5mg
    294,00€
    10mg
    442,00€
    25mg
    705,00€
    50mg
    982,00€
    100mg
    1.333,00€
  • Lys-Bradykinin acetate(342-10-9 free base)

    CAS:
    Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.
    Fórmula:C58H89N17O14
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:1248.43

    Ref: TM-TP2268L

    1mg
    62,00€
    5mg
    124,00€
    10mg
    180,00€
    25mg
    304,00€
    50mg
    427,00€
    100mg
    605,00€
  • Lys-[Des-Arg9]Bradykinin acetate


    Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and
    Fórmula:C52H77N13O13
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:1092.27

    Ref: TM-TP1918L1

    1mg
    84,00€
    5mg
    170,00€
    10mg
    248,00€
    25mg
    452,00€
    50mg
    655,00€
    100mg
    928,00€
  • B 4148

    CAS:
    B 4148 is a bradykinin inhibitor.
    Fórmula:C62H95N19O14S2
    Cor e Forma:Solid
    Peso molecular:1394.67

    Ref: TM-T71571

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • NPC 17731

    CAS:
    NPC 17731 is a bradykinin receptor antagonist.
    Fórmula:C59H95N19O14
    Cor e Forma:Solid
    Peso molecular:1294.5

    Ref: TM-T70576

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • BKM-570

    CAS:
    BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.
    Fórmula:C34H34Cl2F5N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:698.55

    Ref: TM-T26833

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Anatibant

    CAS:
    Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.
    Fórmula:C34H36Cl2N6O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:711.66

    Ref: TM-T26627

    500mg
    A consultar
    25mg
    1.504,00€
    50mg
    1.963,00€
    100mg
    2.520,00€
  • Fulimetibant

    CAS:
    Fulimetibant is a bradykinin receptor antagonist.
    Fórmula:C25H21F4N3O3
    Cor e Forma:Solid
    Peso molecular:487.45

    Ref: TM-T63241

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • MK-0686

    CAS:
    MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.
    Fórmula:C22H19ClF4N2O4
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:486.84

    Ref: TM-T33421

    1mg
    107,00€
    5mg
    254,00€
    10mg
    371,00€
    25mg
    583,00€
    50mg
    830,00€
    100mg
    1.134,00€
    200mg
    1.521,00€
  • Safotibant

    CAS:
    Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edema
    Fórmula:C25H34N4O5S
    Pureza:99.62% - 99.67%
    Cor e Forma:Solid
    Peso molecular:502.63

    Ref: TM-T34485

    1mg
    92,00€
    5mg
    190,00€
    10mg
    286,00€
    25mg
    464,00€
    50mg
    637,00€
    100mg
    858,00€
    200mg
    1.153,00€
  • NVP-SAA164

    CAS:
    NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.
    Fórmula:C36H45N5O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:659.84

    Ref: TM-T25895

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • FK-3657

    CAS:
    FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.
    Fórmula:C30H27Cl2N5O4
    Cor e Forma:Solid
    Peso molecular:592.47

    Ref: TM-T24065

    25mg
    2.015,00€
    50mg
    2.642,00€
    100mg
    3.515,00€
  • BI-113823

    CAS:
    BI-113823 is an orally active and selective bradykinin B1 receptor antagonist. It alleviates mechanical hyperalgesia induced by complete Freund's adjuvant in rats. BI-113823 is applicable for research on chronic inflammatory pain.
    Fórmula:C26H44N4O5S
    Cor e Forma:Solid
    Peso molecular:524.716

    Ref: TM-T205108

    10mg
    A consultar
    50mg
    A consultar