
Receptor de Dopamina
Os receptores de dopamina são um grupo de GPCRs que respondem ao neurotransmissor dopamina, desempenhando um papel fundamental na regulação do movimento, motivação, recompensa e várias funções cognitivas. Esses receptores são divididos em famílias semelhantes a D1 e D2, cada uma com funções e perfis farmacológicos distintos. Moduladores de receptores de dopamina são amplamente estudados por suas aplicações no tratamento da doença de Parkinson, esquizofrenia, dependência e outros transtornos neuropsiquiátricos. Na CymitQuimica, oferecemos uma ampla gama de moduladores de receptores de dopamina de alta qualidade para apoiar sua pesquisa em neurociência, saúde mental e sinalização GPCR.
Foram encontrados 407 produtos de "Receptor de Dopamina"
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carfenazine
CAS:<p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>Fórmula:C24H31N3O2SPureza:98.06%Cor e Forma:SolidPeso molecular:425.59Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Fórmula:C18H18ClNOSPureza:99.78%Cor e Forma:SolidPeso molecular:331.86Tiapride
CAS:<p>Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.</p>Fórmula:C15H24N2O4SCor e Forma:SolidPeso molecular:328.43Pergolide mesylate
CAS:<p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>Fórmula:C20H30N2O3S2Pureza:99.70%Cor e Forma:White To Off-White SolidPeso molecular:410.59Metoclopramide
CAS:<p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>Fórmula:C14H22ClN3O2Pureza:99.75%Cor e Forma:SolidPeso molecular:299.80Rotigotine-
CAS:<p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>Fórmula:C19H25NOSPureza:98.08% - 99.59%Cor e Forma:SolidPeso molecular:315.47J-147
CAS:<p>J-147, a curcumin derivative, is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging.</p>Fórmula:C18H17F3N2O2Pureza:99.61% - >99.99%Cor e Forma:SolidPeso molecular:350.33Pergolide
CAS:<p>Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's disease</p>Fórmula:C19H26N2SPureza:99.95%Cor e Forma:SolidPeso molecular:314.49Tavapadon
CAS:<p>Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.</p>Fórmula:C19H16F3N3O3Pureza:99.33% - 99.8%Cor e Forma:SolidPeso molecular:391.34Piribedil
CAS:<p>Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.</p>Fórmula:C16H18N4O2Pureza:99.79% - 99.82%Cor e Forma:SolidPeso molecular:298.34FAUC 346
CAS:<p>FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.</p>Fórmula:C24H29N3O2SPureza:99.46%Cor e Forma:SolidPeso molecular:423.57Vanoxerine dihydrochloride
CAS:<p>Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)</p>Fórmula:C28H34Cl2F2N2OPureza:98.16% - 98.35%Cor e Forma:White SolidPeso molecular:523.49Azaperone
CAS:<p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>Fórmula:C19H22FN3OPureza:98.73%Cor e Forma:White Or Off-White CrystallinePeso molecular:327.4SKF38393 hydrobromide
CAS:<p>SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;</p>Fórmula:C16H18BrNO2Pureza:98.99%Cor e Forma:SolidPeso molecular:336.22Pramipexole dihydrochloride hydrate
CAS:<p>Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.</p>Fórmula:C10H17N3S·2HCl·H2OPureza:99.68%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:302.26Dasotraline
CAS:<p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>Fórmula:C16H15Cl2NCor e Forma:SolidPeso molecular:292.2PD 168568
CAS:<p>PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.</p>Fórmula:C22H27N3OCor e Forma:SolidPeso molecular:349.47Alizapride
CAS:<p>Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].</p>Fórmula:C16H21N5O2Cor e Forma:SolidPeso molecular:315.37FAUC 213
CAS:<p>FAUC 213 is a selective full antagonist of the dopamine D4 receptor.</p>Fórmula:C18H19ClN4Pureza:99.84%Cor e Forma:SolidPeso molecular:326.82BP 897
CAS:<p>BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.</p>Fórmula:C26H31N3O2Pureza:99.44%Cor e Forma:SolidPeso molecular:417.54Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Fórmula:C25H27N3O2SPureza:99.06% - 99.96%Cor e Forma:SolidPeso molecular:433.57JNJ-37822681
CAS:<p>JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.</p>Fórmula:C17H17F5N4Pureza:99.84%Cor e Forma:SolidPeso molecular:372.34Rotigotine Hydrochloride
CAS:<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Fórmula:C19H26ClNOSPureza:99.53% - 99.56%Cor e Forma:Almost White To White Crystalline PowderPeso molecular:351.93Haloperidol hydrochloride
CAS:<p>Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.</p>Fórmula:C21H24Cl2FNO2Cor e Forma:SolidPeso molecular:412.33Diclofensine hydrochloride
CAS:<p>Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。</p>Fórmula:C17H18Cl3NOPureza:98.86% - 99.93%Cor e Forma:SolidPeso molecular:358.69Sultopride hydrochloride
CAS:<p>Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.</p>Fórmula:C17H27ClN2O4SPureza:≥95%Cor e Forma:White Or Yellowish PowderPeso molecular:390.93Ritanserin
CAS:<p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>Fórmula:C27H25F2N3OSPureza:99.77% - 99.89%Cor e Forma:SolidPeso molecular:477.57L-745870 trihydrochloride
CAS:<p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>Fórmula:C18H22Cl4N4Pureza:97.52%Cor e Forma:SolidPeso molecular:436.21Raclopride
CAS:<p>Raclopride is a selective antagonist of dopamine D2/D3 receptor.</p>Fórmula:C15H20Cl2N2O3Pureza:99.17%Cor e Forma:SolidPeso molecular:347.24Nuciferine
CAS:<p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>Fórmula:C19H21NO2Pureza:98.76% - 99.79%Cor e Forma:SolidPeso molecular:295.38Rotundine
CAS:<p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>Fórmula:C21H25NO4Pureza:99.8% - 99.91%Cor e Forma:Off-White SolidPeso molecular:355.43Lurasidone
CAS:<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Fórmula:C28H36N4O2SPureza:99.78% - 99.91%Cor e Forma:SolidPeso molecular:492.68L-DOPA methyl ester (hydrochloride)
CAS:<p>L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.</p>Fórmula:C10H14ClNO4Pureza:98.69% - 99.81%Cor e Forma:White SolidPeso molecular:247.675Zuclopenthixol dihydrochloride
CAS:<p>Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.</p>Fórmula:C22H27Cl3N2OSPureza:98%Cor e Forma:SolidPeso molecular:473.89AHN 1-055 hydrochloride
CAS:<p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>Fórmula:C21H24ClF2NOPureza:99.89%Cor e Forma:SolidPeso molecular:379.87L-745870 hydrochloride
CAS:<p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>Fórmula:C18H20Cl2N4Pureza:97.36%Cor e Forma:SolidPeso molecular:363.28FAUC-365
CAS:<p>FAUC-365 is a D3 dopamine receptor agonist.</p>Fórmula:C23H25Cl2N3OSPureza:99.62%Cor e Forma:SolidPeso molecular:462.44Tetrahydropalmatine hydrochloride
CAS:<p>Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.</p>Fórmula:C21H26ClNO4Pureza:98% - 99.59%Cor e Forma:SolidPeso molecular:391.888Mesdopetam hemitartrate
CAS:<p>Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.</p>Fórmula:C28H42F2N2O12S2Pureza:99.98%Cor e Forma:SolidPeso molecular:700.77(+)-PD 128907 hydrochloride
CAS:<p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>Fórmula:C14H20ClNO3Pureza:97.76%Cor e Forma:SolidPeso molecular:285.77Metergoline
CAS:<p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>Fórmula:C25H29N3O2Pureza:99.83% - 99.97%Cor e Forma:SolidPeso molecular:403.52WAY-100635 Monomaleate
CAS:<p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>Fórmula:C25H34N4O2·C4H4O4Pureza:98.44% - 99.46%Cor e Forma:SolidPeso molecular:538.64Sertindole
CAS:<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Fórmula:C24H26ClFN4OPureza:99.87% - 99.92%Cor e Forma:Off-White To Pale Yellow SolidPeso molecular:440.94Fenoldopam mesylate
CAS:<p>Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.</p>Fórmula:C16H16ClNO3·CH4O3SPureza:99.19%Cor e Forma:SolidPeso molecular:401.86Clebopride malate
CAS:<p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>Fórmula:C24H30ClN3O7Pureza:99.52%Cor e Forma:SolidPeso molecular:507.96Flupentixol dihydrochloride
CAS:<p>Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.</p>Fórmula:C23H27Cl2F3N2OSPureza:98.76% - >99.99%Cor e Forma:White Or Off-White SolidPeso molecular:507.43Decynium 22
CAS:<p>Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor</p>Fórmula:C23H23IN2Pureza:99.92%Cor e Forma:Dark Red CrystalsPeso molecular:454.35Domperidone monomaleate
CAS:<p>Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.</p>Fórmula:C26H28ClN5O6Cor e Forma:SolidPeso molecular:541.98GBR 12935 dihydrochloride
CAS:<p>GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.</p>Fórmula:C28H36Cl2N2OPureza:99.09% - ≥95%Cor e Forma:SolidPeso molecular:487.5Thozalinone
CAS:<p>Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.</p>Fórmula:C11H12N2O2Pureza:99.68%Cor e Forma:SolidPeso molecular:204.23
