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Receptor de adenosina

Receptor de adenosina

Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.

Foram encontrados 249 produtos de "Receptor de adenosina"

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  • Apadenoson

    CAS:
    Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.
    Fórmula:C23H30N6O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:486.52

    Ref: TM-T26641

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • Lu AA 47070

    CAS:
    adenosine A2A receptor antagonist
    Fórmula:C17H20F2N3O6PS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:463.39

    Ref: TM-T22934

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • A1AR antagonist 2

    CAS:
    Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.
    Fórmula:C17H12N4O
    Cor e Forma:Solid
    Peso molecular:288.3

    Ref: TM-T60580

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • A1/A3 AR antagonist 2

    CAS:
    The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.
    Fórmula:C22H16N2O3S
    Cor e Forma:Solid
    Peso molecular:388.44

    Ref: TM-T61744

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • AB-MECA

    CAS:
    AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.
    Fórmula:C18H21N7O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:399.4

    Ref: TM-T14082

    1mg
    239,00€
    5mg
    1.018,00€
    10mg
    1.783,00€
  • A2AAR/HDAC-IN-1

    CAS:
    A2AAR/HDAC-IN-1 (compound 14c) is an orally active, balanced A2AAR/HDAC dual inhibitor of A2AAR (Ki: 163.5 nM), HDAC1 (IC50: 145.3 nM). effect.
    Fórmula:C24H21N7O2
    Cor e Forma:Solid
    Peso molecular:439.47

    Ref: TM-T62521

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • LASSBio-1359

    CAS:
    LASSBio-1359 is an adenosine receptor agonist. It acts by inducing relaxation of the corpus cavernosum. It also acts as a novel selective phosphodiesterase.
    Fórmula:C17H18N2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:298.34

    Ref: TM-T24388

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • PSB 11 hydrochloride

    CAS:
    PSB 11 hydrochloride is a human adenosine A3 receptor antagonist.
    Fórmula:C16H18ClN5O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:331.8

    Ref: TM-T23199

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Adenosine receptor antagonist 3

    CAS:
    Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1].
    Fórmula:C16H14N6S
    Cor e Forma:Solid
    Peso molecular:322.39

    Ref: TM-T60872

    25mg
    858,00€
    50mg
    1.116,00€
    100mg
    1.791,00€
  • Adentri

    CAS:
    Adentri is a novel antagonist of adenosine A1 receptor with unique diuretic activity.
    Fórmula:C18H24N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:344.41

    Ref: TM-T26565

    25mg
    1.369,00€
  • A2A receptor antagonist 3

    CAS:
    A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).
    Fórmula:C26H26N6O2
    Cor e Forma:Solid
    Peso molecular:454.52

    Ref: TM-T62797

    25mg
    1.927,00€
    50mg
    2.507,00€
    100mg
    3.168,00€
  • MRS1186

    CAS:
    MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).
    Fórmula:C16H12ClN5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:341.75

    Ref: TM-T16138

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Adenosine receptor A1 antagonist 5

    CAS:
    1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.
    Fórmula:C17H20N4O2
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:312.37

    Ref: TM-T22466

    1mg
    46,00€
    5mg
    94,00€
    10mg
    137,00€
    25mg
    226,00€
    50mg
    324,00€
    100mg
    447,00€
    200mg
    600,00€
  • MRS1177

    CAS:
    MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).
    Fórmula:C20H12ClN5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:389.79

    Ref: TM-T16137

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • XU1

    CAS:
    XU1(Benzo[c][1,8]naphthyridin-6(5h)-One) is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation or
    Fórmula:C12H8N2O
    Pureza:97.81% - 99.59%
    Cor e Forma:Solid
    Peso molecular:196.2

    Ref: TM-T29170

    1mg
    295,00€
    5mg
    705,00€
    10mg
    982,00€
    25mg
    1.485,00€
    50mg
    2.008,00€
    100mg
    2.655,00€
  • HEMADO

    CAS:
    HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).
    Fórmula:C17H23N5O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:361.4

    Ref: TM-T15468

    1mg
    112,00€
    5mg
    388,00€
  • A1AR antagonist 6

    CAS:
    A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].
    Fórmula:C17H15N3O2
    Cor e Forma:Solid
    Peso molecular:293.32

    Ref: TM-T60615

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Lu AA41063

    CAS:
    Lu AA41063 is a potent and selective antagonist of the hA2A receptor.
    Fórmula:C16H17F2N3O2S
    Cor e Forma:Solid
    Peso molecular:353.39

    Ref: TM-T24418

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Neladenoson dalanate HCl

    CAS:
    Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).
    Fórmula:C35H35Cl2N7O4S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:752.73

    Ref: TM-T24526

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • A3AR antagonist 1

    CAS:
    A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.
    Fórmula:C32H24N4O4S
    Cor e Forma:Solid
    Peso molecular:560.62

    Ref: TM-T63960

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€