
Receptor de adenosina
Os receptores de adenosina são uma classe de GPCRs que respondem ao nucleosídeo endógeno adenosina. Esses receptores estão envolvidos na regulação de vários processos fisiológicos, incluindo função cardiovascular, ciclos de sono-vigília e respostas imunes. Moduladores de receptores de adenosina têm potencial terapêutico no tratamento de condições como arritmias cardíacas, inflamação e doenças neurodegenerativas. Na CymitQuimica, oferecemos uma seleção de moduladores de receptores de adenosina de alta qualidade para apoiar sua pesquisa em biologia cardiovascular, neurociência e imunologia.
Foram encontrados 249 produtos de "Receptor de adenosina"
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A2AAR/HDAC-IN-2
CAS:A2AAR/HDAC-IN-2: potent dual A2AAR/HDAC inhib., Ki 10.3 nM, IC50 18.5 nM, anti-tumor potential.Fórmula:C23H26N6O4Cor e Forma:SolidPeso molecular:450.49Theophylline sodium glycinate
CAS:Theophylline sodium glycinate inhibits PDE3, treats asthma/COPD, blocks adenosine receptors, activates HDAC, reduces inflammation and induces apoptosis.Fórmula:C9H12N5NaO4Cor e Forma:SolidPeso molecular:277.216hA2AAR antagonist 1
CAS:Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.Fórmula:C15H15N5OCor e Forma:SolidPeso molecular:281.31LUF5831
CAS:LUF5831 is an agonist of adenosine A1 receptor.Fórmula:C15H12N4O2SCor e Forma:SolidPeso molecular:312.35Draflazine
CAS:Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.Fórmula:C30H33Cl2F2N5O2Pureza:98%Cor e Forma:SolidPeso molecular:604.52LUF5981
CAS:LUF5981 is a selective agonist of human adenosine A1 receptor.Fórmula:C24H23N3Cor e Forma:SolidPeso molecular:353.46Cirazoline hydrochloride
CAS:Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.Fórmula:C13H17ClN2OPureza:99.863%Cor e Forma:SolidPeso molecular:252.74Bamifylline Hydrochloride
CAS:Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.Fórmula:C20H28ClN5O3Cor e Forma:SolidPeso molecular:421.92MRS1067
CAS:MRS1067 is an antagonist of A3 adenosine receptor.Fórmula:C19H16Cl2O3Cor e Forma:SolidPeso molecular:363.23VUF8504
CAS:VUF8504 is a novel ligand of adenosine A3 receptor.Fórmula:C22H17N3O2Cor e Forma:SolidPeso molecular:355.39WRC-0571
CAS:WRC-0571 is a highly potent, selective antagonist of A1 adenosine receptors.Fórmula:C17H26N6OPureza:98%Cor e Forma:SolidPeso molecular:330.43Naxifylline
CAS:Naxifylline is an A1 adenosine receptor blocker that increases urine and protects kidneys during edema treatment in heart failure.Fórmula:C18H24N4O3Cor e Forma:SolidPeso molecular:344.41CP 66713
CAS:CP-66713 is an adenosine A2 receptor antagonist.Fórmula:C15H10ClN5Cor e Forma:SolidPeso molecular:295.73A2AAR antagonist 1
CAS:Compound 21a, A2AAR antagonist with 20 nM Ki, useful in neurodegenerative disease study.Fórmula:C12H8BrN3OCor e Forma:SolidPeso molecular:290.12MRE3008F20
CAS:MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.Fórmula:C21H20N8O3Pureza:97.29%Cor e Forma:SolidPeso molecular:432.44A2AR-antagonist-1
CAS:Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.Fórmula:C27H25N5O2Pureza:98%Cor e Forma:SolidPeso molecular:451.52VUF 5574
CAS:VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.Fórmula:C21H17N5O2Pureza:99.53%Cor e Forma:SolidPeso molecular:371.39ST3932
CAS:ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).Fórmula:C12H16N8OPureza:98%Cor e Forma:SolidPeso molecular:288.31N6-Cyclopentyladenosine
CAS:N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's ofFórmula:C15H21N5O4Pureza:99.95%Cor e Forma:SolidPeso molecular:335.36N-[(4-Aminophenyl)methyl]adenosine
CAS:N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).Fórmula:C17H20N6O4Pureza:98.75%Cor e Forma:SolidPeso molecular:372.38Ref: TM-T16166
1mg52,00€5mg111,00€10mg166,00€25mg318,00€50mg504,00€100mg803,00€1mL*10mM (DMSO)141,00€
