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Sinalização Citoesquelética

Sinalização Citoesquelética

Os inibidores de sinalização do citoesqueleto são compostos que interrompem as vias de sinalização que regulam o citoesqueleto, crucial para a forma celular, motilidade, divisão e transporte intracelular. Esses inibidores são usados para estudar a dinâmica das proteínas do citoesqueleto, como actina e tubulina, e seu papel em processos como migração celular, adesão e metástase do câncer. Os inibidores de sinalização do citoesqueleto são valiosos na pesquisa em biologia celular, câncer e neurobiologia. Na CymitQuimica, oferecemos uma ampla gama de inibidores de sinalização do citoesqueleto de alta qualidade para apoiar sua pesquisa nessas áreas.

Foram encontrados 1381 produtos de "Sinalização Citoesquelética"

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produtos por página.
  • XL228

    CAS:
    <p>XL228 is an inhibitor of multi-targeted tyrosine kinase (IC50s: 5, 3.1, 1.6, 6.1, 2 nM for Bcr-Abl, Aurora A, IGF-1R, Src, and Lyn, respectively).</p>
    Fórmula:C22H31N9O
    Pureza:99.07%
    Cor e Forma:Solid
    Peso molecular:437.54
  • Imatinib

    CAS:
    <p>Imatinib (STI571) is a multi-targeted receptor tyrosine kinase inhibitor that selectively inhibits the kinase activities of BCR/ABL, v-Abl, PDGFR, and c-kit</p>
    Fórmula:C29H31N7O
    Pureza:99.42% - 99.94%
    Cor e Forma:Off White Powder
    Peso molecular:493.6
  • OSU-T315

    CAS:
    <p>OSU-T315 (OSU-T315 (1,5-regioisomer)) (1,5-regioisomer) is a ILK inhibitor.</p>
    Fórmula:C30H30F3N5O
    Pureza:98.69%
    Cor e Forma:Solid
    Peso molecular:533.59
  • TPPB

    CAS:
    <p>TPPB is a kinase C activator of cell-permeable benzolactam-derived protein (Ki: 11.9 nM).</p>
    Fórmula:C27H30F3N3O3
    Pureza:97.71% - 98.00%
    Cor e Forma:Solid
    Peso molecular:501.54
  • Ro 31-8220 Mesylate

    CAS:
    <p>Ro 31-8220 Mesylate (Bisindolylmaleimide IX mesylate) is a pan-PKC inhibitor, and also shows potent inhibition against MSK1, MAPKAP-K1b, S6K1, and GSK3β.</p>
    Fórmula:C25H23N5O2S·CH4O3S
    Pureza:98.79% - 99.02%
    Cor e Forma:Solid
    Peso molecular:553.65
  • Flumatinib mesylate

    CAS:
    <p>Flumatinib mesylate (HHGV678 mesylate) is a selective inhibitor of c-Abl, PDGFRβ and c-Kit, effectively overcomes drug resistance of certain KIT mutants.</p>
    Fórmula:C30H33F3N8O4S
    Pureza:99.82%
    Cor e Forma:Solid
    Peso molecular:658.69
  • D-64131

    CAS:
    <p>D-64131 is a tubulin polymerization inhibitor with an IC50 value of 0.53 μM.</p>
    Fórmula:C16H13NO2
    Pureza:99.48% - 99.67%
    Cor e Forma:Solid
    Peso molecular:251.28
  • Tirbanibulin

    CAS:
    <p>Tirbanibulin (KX2-391) is a highly selective Src kinase inhibitor that has demonstrated efficacy in pre-Clinicalal animal models of a variety of cancers.</p>
    Fórmula:C26H29N3O3
    Pureza:99.43% - 99.67%
    Cor e Forma:Solid
    Peso molecular:431.53
  • Procyanidin A1

    CAS:
    <p>Procyanidin A1 (Proanthocyanidin A1) has antiallergic effects, it inhibits degranulation downstream of protein kinase C activation or Ca2+.</p>
    Fórmula:C30H24O12
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:576.5
  • Borussertib

    CAS:
    <p>Borussertib is a covalent-allosteric and first-in-class inhibitor of protein kinase Akt(IC50 of 0.8 nM and a Ki of 2.2 nM for Aktwt)</p>
    Fórmula:C36H32N6O3
    Pureza:99.00%
    Cor e Forma:Solid
    Peso molecular:596.68
  • Ingenol

    CAS:
    <p>Ingenol mebutate treats actinic keratosis, has anticancer properties, and may reactivate latent HIV.</p>
    Fórmula:C20H28O5
    Pureza:99.78% - 99.87%
    Cor e Forma:Solid
    Peso molecular:348.43
  • BX517

    CAS:
    <p>BX517 (PDK1 inhibitor 2) is a potent and selective inhibitor of PDK1.</p>
    Fórmula:C15H14N4O2
    Pureza:99.26%
    Cor e Forma:Solid
    Peso molecular:282.3
  • Monastrol

    CAS:
    <p>Monastrol ((±)-Monastrol) is a potent and cell-permeable inhibitor of the mitotic kinesin Eg5.</p>
    Fórmula:C14H16N2O3S
    Pureza:98.02% - 98.59%
    Cor e Forma:Solid
    Peso molecular:292.35
  • Sotrastaurin

    CAS:
    <p>Sotrastaurin (AEB071) is a potent pan-PKC inhibitor (Kis: 0.95/0.64/2.1/3.2/1.8/0.22 nM for PKCα/βI/δ/ε/η/θ).</p>
    Fórmula:C25H22N6O2
    Pureza:98% - 99.70%
    Cor e Forma:Solid
    Peso molecular:438.48
  • Valrubicin

    CAS:
    <p>Valrubicin (AD-32) (AD 32) inhibits TPA- and PDBu-induced PKC activation (IC50s: 0.85 and 1.25 μM) and has antitumor and anti-inflammatory activity.</p>
    Fórmula:C34H36F3NO13
    Pureza:98.63%
    Cor e Forma:Solid
    Peso molecular:723.64
  • Pep2m, myristoylated acetate


    <p>Pep2m, a myristoylated acetate, inhibits GluA2-NSF interaction, reducing AMPA receptor function and expression in neurons.</p>
    Fórmula:C65H122N18O16S
    Pureza:99.62%
    Cor e Forma:Solid
    Peso molecular:1443.96
  • PF-431396

    CAS:
    <p>PF-431396 is a dual PYK2/FAK inhibitor (IC50: 11/2 nM).</p>
    Fórmula:C22H21F3N6O3S
    Pureza:98.83% - 99.82%
    Cor e Forma:Solid
    Peso molecular:506.5
  • Vodobatinib

    CAS:
    <p>Vodobatinib (K-0706) is a novel 3rd generation (3G) TKI effective against wild-type and mutated BCR-ABL1 with limited off-target activity.</p>
    Fórmula:C27H20ClN3O2
    Pureza:99.06% - 99.55%
    Cor e Forma:Solid
    Peso molecular:453.92
  • Decursin

    CAS:
    <p>Decursin: potential antiepileptic, hepatoprotective, anti-cancer, anti-amnesic; affects NOX activation, PKCα/MAPK/NF-κB pathways, AChE.</p>
    Fórmula:C19H20O5
    Pureza:97.22% - 99.84%
    Cor e Forma:Solid
    Peso molecular:328.36
  • Pimitespib

    CAS:
    <p>Pimitespib (TAS-116) is an ATP-competitive and highly specific HSP90α/HSP90β inhibitor (Kis: 34.7 nM and 21.3 nM, respectively).</p>
    Fórmula:C25H26N8O
    Pureza:99.22% - 99.49%
    Cor e Forma:Solid
    Peso molecular:454.53
  • Ζ-Stat

    CAS:
    <p>ζ-Stat (NSC37044), a specific and atypical inhibitor of PKC-ζ with an IC50 of 5 μM, demonstrates the ability to inhibit proliferation and induce apoptosis in</p>
    Fórmula:C10H8O10S3
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:384.36
  • Dimethylenastron

    CAS:
    <p>Dimethylenastron, an Eg5 inhibitor, arrests cells with monopolar spindles to which all chromosomes attach in a syntelic manner.</p>
    Fórmula:C16H18N2O2S
    Pureza:98.07%
    Cor e Forma:Solid
    Peso molecular:302.39
  • GLPG0187

    CAS:
    <p>GLPG0187, a broad spectrum integrin receptor antagonist, inhibits αvβ1-integrin (IC50: 1.3 nM).</p>
    Fórmula:C29H37N7O5S
    Pureza:99.4% - 99.70%
    Cor e Forma:Solid
    Peso molecular:595.71
  • Chelerythrine chloride

    CAS:
    <p>Chelerythrine Chloride is a cell-permeable inhibitor of protein kinase C, competitive with respect to the phosphate acceptor and non-competitive with respect to</p>
    Fórmula:C21H18ClNO4
    Pureza:95% - 99.19%
    Cor e Forma:Yellow To Orange Solid
    Peso molecular:383.83
  • T807

    CAS:
    <p>T807 (AV-1451) is a novel tracer of tau positron emission tomography (PET).</p>
    Fórmula:C16H10FN3
    Pureza:99.72%
    Cor e Forma:Solid
    Peso molecular:263.27
  • LP-261

    CAS:
    <p>LP-261 is a novel tubulin targeting anticancer agent that binds at the colchicine site on tubulin, inducing G2/M arrest.</p>
    Fórmula:C22H19N3O4S
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:421.47
  • VER-82576

    CAS:
    <p>VER-82576 (NVP-BEP800), a synthetic HSP90β inhibitor (IC50: 58 nM), exhibits &gt;70-fold selectivity against Hsp90 family members Trap-1 and Grp94.</p>
    Fórmula:C21H23Cl2N5O2S
    Pureza:97.31% - 99.85%
    Cor e Forma:Solid
    Peso molecular:480.41
  • PND-1186

    CAS:
    <p>PND-1186 (VS-4718) is a reversible and specific FAK inhibitor (IC50: 1.5 nM).</p>
    Fórmula:C25H26F3N5O3
    Pureza:99.14% - 99.75%
    Cor e Forma:Solid
    Peso molecular:501.5
  • PF-562271 hydrochloride

    CAS:
    <p>PF-562271 hydrochloride (PF-562271 HCl) is a potent, ATP-competitive, reversible inhibitor of FAK with IC50 of 1.5 nM, ~10-fold less potent for Pyk2 than FAK.</p>
    Fórmula:C21H20F3N7O3SHCl
    Pureza:97.08%
    Cor e Forma:Solid
    Peso molecular:543.95
  • R59949

    CAS:
    <p>R59949 is used as a Diacylglycerol kinase (DGK) inhibitor.</p>
    Fórmula:C28H25F2N3OS
    Pureza:97.04%
    Cor e Forma:Solid
    Peso molecular:489.58
  • Natalizumab

    CAS:
    <p>Natalizumab used for the treatment of relapsing remitting multiple sclerosis and Crohn's disease.</p>
    Pureza:98.00%
    Cor e Forma:Liquid
    Peso molecular:N/A
  • Empesertib

    CAS:
    <p>Empesertib (BAY 1161909) is an orally bioavailable and selective inhibitor Mps1(IC50 &lt; 1 nM), with potential antineoplastic activity.</p>
    Fórmula:C29H26FN5O4S
    Pureza:97.45% - 99.4%
    Cor e Forma:Solid
    Peso molecular:559.61
  • MAP4343

    CAS:
    <p>Map4343, a 3-methyl ether pregnenolone derivative, binds MAP2, boosts tubulin polymerization, spurs neurite growth, and guards neurons.</p>
    Fórmula:C22H34O2
    Pureza:97.024%
    Cor e Forma:Solid
    Peso molecular:330.5
  • HSF1A

    CAS:
    <p>HSF1A is a cell-permeable activator of HSF1 that protects mammalian cells against stress-induced apoptosis.</p>
    Fórmula:C21H19N3O2S2
    Pureza:98.89%
    Cor e Forma:Solid
    Peso molecular:409.52
  • Curvulin

    CAS:
    <p>Curvulin is the active metabolite isolated from Paraphoma sp. VIZR 1.46. Curvularin inhibits iNOS expression and microtubule assembly.</p>
    Fórmula:C12H14O5
    Pureza:98.65%
    Cor e Forma:Solid
    Peso molecular:238.24
  • TASP0415914

    CAS:
    <p>TASP0415914 is an orally potent inhibitor of phosphoinositide 3-kinase γ (PI3Kγ). T</p>
    Fórmula:C13H17N5O3S
    Pureza:98.14%
    Cor e Forma:Solid
    Peso molecular:323.37
  • Mavacamten

    CAS:
    <p>Mavacamten (MYK-461) is an orally bioavailable inhibitor of cardiac myosin ATPase,( IC50s of 490, 711 nM for bovine cardiac and human cardiac, respectively)</p>
    Fórmula:C15H19N3O2
    Pureza:99.53% - 99.98%
    Cor e Forma:Solid
    Peso molecular:273.33
  • Hydroxy-Dynasore

    CAS:
    <p>Hydroxy-Dynasore (Dyngo-4a) , a effective dynamin inhibitor, inhibits withDynI (brain), DynI (rec), and DynII (rec) of IC50 of 0.38 μM, 1.1 μM, and 2.3 μM,</p>
    Fórmula:C18H14N2O5
    Pureza:97.60% - >99.99%
    Cor e Forma:Solid
    Peso molecular:338.31
  • PKCβ inhibitor 1

    CAS:
    <p>PKCβ inhibitor 1 (KUN79359)(KUN79359) is a potent, selective and ATP-competitive inhibitor of PKC isozymes(IC50s of 21 and 5 nM for human PKCβ1 and PKCβ2,</p>
    Fórmula:C24H21N5O2
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:411.46
  • ARQ 621

    CAS:
    <p>ARQ 621 is an allosteric, and selective Eg5 mitotic motor protein inhibitor. Phase 1.</p>
    Fórmula:C28H24Cl2FN5O2
    Pureza:97.01% - 98.38%
    Cor e Forma:Solid
    Peso molecular:552.43
  • HM03

    CAS:
    <p>HM03 is a potent and selective inhibitor of HSPA5, and has anticancer activity.</p>
    Fórmula:C26H27ClN4O2
    Pureza:97.15%
    Cor e Forma:Solid
    Peso molecular:462.97
  • CZC-8004

    CAS:
    <p>CZC-8004 (CZC-00008004) is a pan-kinase(ABL kinase) inhibitor and binds a range of tyrosine kinases.</p>
    Fórmula:C17H16FN5
    Pureza:99.29%
    Cor e Forma:Solid
    Peso molecular:309.34
  • Taurolithocholic acid sodium salt

    CAS:
    <p>Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but</p>
    Fórmula:C26H44NNaO5S
    Pureza:99.79% - 99.93%
    Cor e Forma:Solid
    Peso molecular:505.69
  • Teduglutide acetate


    <p>Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy.</p>
    Fórmula:C166H256N44O56S
    Pureza:97.39%
    Cor e Forma:Soild
    Peso molecular:3812.13
  • BAY1125976

    CAS:
    <p>BAY1125976 is an allosteric inhibitor of Akt1 and Akt2 (IC50s of 5.2 and 18 nM, respectively, in a time-resolved FRET assay)</p>
    Fórmula:C23H21N5O
    Pureza:99.28% - ≥98%
    Cor e Forma:Solid
    Peso molecular:383.45
  • Desmethylglycitein

    CAS:
    <p>Desmethylglycitein (6,7,4'-Trihydroxyisoflavone) , is a novel inhibitor of PKCα in suppressing solar UV-induced matrix metalloproteinase 1, which has</p>
    Fórmula:C15H10O5
    Pureza:97.93%
    Cor e Forma:Solid
    Peso molecular:270.24
  • Hexapeptide-10 Acetate


    <p>Hexapeptide-10 Acetate (Hexapeptide-10 Acetate) is a synthetic peptide.</p>
    Fórmula:C30H57N7O10
    Pureza:98.84%
    Cor e Forma:Solid
    Peso molecular:675.81
  • KW-2478

    CAS:
    <p>KW-2478 is a non-ansamycin HSP90 inhibitor with IC50 of 3.8 nM.</p>
    Fórmula:C30H42N2O9
    Pureza:98.68% - 99.52%
    Cor e Forma:Solid
    Peso molecular:574.66
  • LXW7

    CAS:
    <p>LXW7 is an octamer disulfide cyclic peptide and αvβ3 integrin ligand, acts as a potent and specific endothelial progenitor cells (EPCs) and endothelial cells (</p>
    Fórmula:C29H48N12O12S2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:820.89
  • Multi-kinase inhibitor 1

    CAS:
    <p>Multi-kinase inhibitor 1 (Multi-kinase inhibitor I) is a Multi-kinase inhibitor.</p>
    Fórmula:C20H17F3N4O3
    Pureza:99.34%
    Cor e Forma:Solid
    Peso molecular:418.37
  • MMAF

    CAS:
    <p>MMAF (MonoMethyl auristatin F), an antimitotic agent, inhibits cell division by blocking the polymerization of tubulin.</p>
    Fórmula:C39H65N5O8
    Pureza:97.00% - 99.88%
    Cor e Forma:Solid
    Peso molecular:731.96
  • Ispinesib

    CAS:
    <p>Ispinesib (SB-715992), a selective, effectvie and reversible inhibitor of kinesin spindle protein (KSP), is derived from quinazolinone, with antineoplastic</p>
    Fórmula:C30H33ClN4O2
    Pureza:98% - 99.09%
    Cor e Forma:Solid
    Peso molecular:517.06
  • Gap 26

    CAS:
    <p>Gap 26 is a mimetic peptide corresponding to the residues 63-75 of connexin 43, which is a gap junction blocker.</p>
    Fórmula:C70H107N19O19S
    Pureza:98.26%
    Cor e Forma:Solid
    Peso molecular:1550.78
  • Dasatinib N-oxide

    CAS:
    <p>Dasatinib N-oxide is a key metabolite and potential impurity of the kinase inhibitor dasatinib.</p>
    Fórmula:C22H26ClN7O3S
    Pureza:98.54% - 99.94%
    Cor e Forma:Solid
    Peso molecular:504
  • PF04929113

    CAS:
    <p>PF04929113 (SNX-5422), a synthetic small molecule Hsp90 inhibitor, offers potent efficacy orally for various cancers.</p>
    Fórmula:C25H30F3N5O4
    Pureza:99.04%
    Cor e Forma:Solid
    Peso molecular:521.53
  • XL888

    CAS:
    <p>XL888 is an orally bioavailable Hsp90 inhibitor, blocking cell proliferation and inducing tumor regression with an IC50 of 24 nM.</p>
    Fórmula:C29H37N5O3
    Pureza:99.18%
    Cor e Forma:Solid
    Peso molecular:503.64
  • H-Gly-Arg-Gly-Asp-Asn-Pro-OH

    CAS:
    <p>RGD peptide (GRGDNP) (RGD peptide GRGDNP(2TFA)) is a integrin-ligand interactions inhibitor.</p>
    Fórmula:C23H38N10O10
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:614.61
  • PKC ζ pseudosubstrate acetate


    <p>PKC ζ pseudosubstrate acetate is an inhibitor of protein kinase C (PKC) ζ; attached to cell permeabilisation Antennapedia domain vector peptide.</p>
    Fórmula:C78H132N30O18
    Pureza:98.78%
    Cor e Forma:Solid
    Peso molecular:1778.10
  • ILK-IN-2

    CAS:
    <p>ILK-IN-2 (OSU-T315) is a novel potent, orally active ILK (integrin-linked kinase) inhibitor with IC50 of 0.6 μM.</p>
    Fórmula:C30H30F3N5O
    Pureza:99.30%
    Cor e Forma:Solid
    Peso molecular:533.59
  • Fingolimod hydrochloride

    CAS:
    <p>Fingolimod hydrochloride (FTY720) , a novel immune modulator, is a sphingosine 1-phosphate (S1P) antagonist (IC50: 0.033 nM in K562 and NK cells).</p>
    Fórmula:C19H34ClNO2
    Pureza:99.26% - 99.83%
    Cor e Forma:White Solid
    Peso molecular:343.93
  • HA-100

    CAS:
    <p>HA-100 is an inhibitor of protein kinase</p>
    Fórmula:C13H15N3O2S
    Pureza:99.44%
    Cor e Forma:Pale Yellow Crystalline Solid
    Peso molecular:277.34
  • TAT-Gap19 acetate


    <p>TAT-Gap19 acetate, a Cx43 HC inhibitor, crosses blood-brain barrier, reduces liver fibrosis in mice, and spares Cx43 GJCs.</p>
    Fórmula:C119H212N46O26
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:2703.25
  • Plinabulin

    CAS:
    <p>Plinabulin (NPI-2358) (NPI-2358) is a vascular disrupting agent (VDA) against tubulin-depolymerizing tumor cells ( IC50: 9.8-18 nM).</p>
    Fórmula:C19H20N4O2
    Pureza:98.69% - >99.99%
    Cor e Forma:Solid
    Peso molecular:336.39
  • Hypocrellin A

    CAS:
    <p>Hypocrellin A is a natural PKC inhibitor with light-induced antitumor, antifungal and antiviral activities.Cost-effective and quality-assured.</p>
    Fórmula:C30H26O10
    Pureza:98% - 99.81%
    Cor e Forma:Solid
    Peso molecular:546.52
  • Nilotinib monohydrochloride monohydrate

    CAS:
    <p>Nilotinib monohydrochloride monohydrate (Nilotinib (monohydrochloride monohydrate)) is significantly potent BCR-ABL against, is a second generation tyrosine</p>
    Fórmula:C28H22F3N7O·HCl·H2O
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:583.99
  • Soblidotin

    CAS:
    <p>Soblidotin (TZT-1027) (Auristatin PE) is an inhibitor of tubulin polymerization. It is also a novel synthetic Dolastatin 10 derivative.</p>
    Fórmula:C39H67N5O6
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:701.98
  • Adaphostin

    CAS:
    <p>Adaphostin (NSC-680410) is a p210Bcr/Abl tyrosine kinase inhibitor with IC50 of 14 μM.</p>
    Fórmula:C24H27NO4
    Pureza:98.29%
    Cor e Forma:Solid
    Peso molecular:393.48
  • Protein Kinase C 19-31 acetate


    <p>PKC 19-31 acetate, a serine-altered PKCa-derived PKC inhibitor, tests PKC activity.</p>
    Fórmula:C69H122N26O18
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1603.9
  • Hypericin

    CAS:
    <p>Hypericin (Cyclosan) is a natural anthraquinone compound. Hypericin exhibits antimicrobial, antiviral, antitumor, and antidepressant effects. Cost-effective and quality-assured.</p>
    Fórmula:C30H16O8
    Pureza:99.05% - ≥98%
    Cor e Forma:Red-Coloured Anthraquinone-Derivative
    Peso molecular:504.44
  • Gly-Arg-Gly-Asp-Ser acetate(96426-21-0 free base)


    <p>Gly-Arg-Gly-Asp-Ser (GRGDS) acetate is a cell binding protein domain derived from the cell-binding region of fibronectin.</p>
    Fórmula:C19H34N8O11
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:550.52
  • Lifitegrast

    CAS:
    <p>Lifitegrast (SAR 1118) is a lymphocyte, function-associated antigen-1 antagonist.</p>
    Fórmula:C29H24Cl2N2O7S
    Pureza:99.39% - 99.66%
    Cor e Forma:Solid
    Peso molecular:615.48
  • PF-562271

    CAS:
    <p>PF-562271 is an effective ATP-competitive, reversible inhibitor of FAK(IC50=1.5 nM) and Pyk2 kinase(IC50=13 nM).</p>
    Fórmula:C21H20F3N7O3S
    Pureza:97.17% - >99.99%
    Cor e Forma:Solid
    Peso molecular:507.49
  • Bisindolylmaleimide V

    CAS:
    <p>Bisindolylmaleimide V, a bisindolylmaleimide derivative, is an inactive of a kinase inhibitor.</p>
    Fórmula:C21H15N3O2
    Pureza:90%
    Cor e Forma:Red Solid
    Peso molecular:341.36
  • Defactinib

    CAS:
    <p>Defactinib (VS-6063) is a second-generation inhibitor of FAK. Defactinib has potential antitumor activity. Cost-effective and quality-assured.</p>
    Fórmula:C20H21F3N8O3S
    Pureza:98% - 99.71%
    Cor e Forma:Solid
    Peso molecular:510.49
  • PF-AKT400

    CAS:
    <p>PF-AKT400 (AKT protein kinase inhibitor) is a broadly selective and ATP-competitive inhibitor of Akt.</p>
    Fórmula:C20H22F2N6O
    Pureza:98.21%
    Cor e Forma:Solid
    Peso molecular:400.43
  • Estramustine

    CAS:
    <p>Estramustine (LEO-275), a nitrogen mustard-estradiol compound, treats prostate cancer and protects against radiation.</p>
    Fórmula:C23H31Cl2NO3
    Pureza:98.09%
    Cor e Forma:Solid
    Peso molecular:440.4
  • ML346

    CAS:
    <p>ML346 is a novel activator of Hsp70.</p>
    Fórmula:C14H12N2O4
    Pureza:97.32% - 99.36%
    Cor e Forma:Solid
    Peso molecular:272.26
  • PD173955

    CAS:
    <p>PD173955 is src family-selective tyrosine kinase inhibitor with IC50 of ~22 nM for Src, Yes and Abl kinase; less potent for FGFRα and no activity on InsR and</p>
    Fórmula:C21H16Cl2N4OS
    Pureza:98.52% - 98.99%
    Cor e Forma:Solid
    Peso molecular:443.35
  • ILK-IN-3

    CAS:
    ILK-IN-3 is an inhibitor of integrin linked kinase, and with antitumor activity.
    Fórmula:C10H12N6O
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:232.24
  • Ansamitocin P 3'

    CAS:
    <p>Ansamitocin P 3' (Maytansinol butyrate) is an antibody-drug conjugate cytotoxin with antitumor activity.</p>
    Fórmula:C32H43ClN2O9
    Pureza:98.16% - 99.16%
    Cor e Forma:Solid
    Peso molecular:635.14
  • AST 487

    CAS:
    <p>AST 487 (NVP-AST 487) is a RET kinase inhibitor, inhibiting RET autophosphorylation and activation of downstream effectors. It also can inhibit Flt-3.</p>
    Fórmula:C26H30F3N7O2
    Pureza:98.17% - 99.56%
    Cor e Forma:Solid
    Peso molecular:529.56
  • Pamidronate disodium pentahydrate

    CAS:
    <p>Pamidronate disodium pentahydrate strengthens bones and prevents osteoporosis.</p>
    Fórmula:C3H21NNa2O12P2
    Pureza:99.84%
    Cor e Forma:White To Off-White Crystalline Powder
    Peso molecular:371.13
  • roxifiban

    CAS:
    <p>Roxifiban, a prodrug of XV459, is an antiplatelet agent with high affinity and specificity for platelet glycoprotein IIb/IIIa complex(GPIIb/IIIa) receptors.</p>
    Fórmula:C21H29N5O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:447.48
  • IM-12

    CAS:
    <p>IM-12, an effective GSK-3β inhibitor(IC50=53 nM), regulates Wnt signalling.</p>
    Fórmula:C22H20FN3O2
    Pureza:99.42% - >99.99%
    Cor e Forma:Solid
    Peso molecular:377.41
  • Dynamin inhibitory peptide, myristoylated acetate


    <p>Myristoylated acetate peptide inhibits DynaMin, blocking amphiphysin binding; myristoylated TFA variant hinders endocytosis.</p>
    Fórmula:C63H111N19O16
    Pureza:99.42%
    Cor e Forma:Solid
    Peso molecular:1390.67
  • Olverembatinib

    CAS:
    <p>Olverembatinib (GZD 824) is an orally bioavailable Bcr-Abl inhibitor for Bcr-Abl(WT, IC50: 0.34 nM) and Bcr-Abl(T315I, IC50: 0.68 nM).</p>
    Fórmula:C29H27F3N6O
    Pureza:98.53% - >99.99%
    Cor e Forma:Solid
    Peso molecular:532.56
  • [Ala107]-MBP (104-118) acetate


    <p>[Ala107]-MBP (104-118) acetate ([Ala107]-MBP ) is synthetic peptide analog of bovine myelin basic protein (MBP).</p>
    Fórmula:C59H108N20O21
    Pureza:99.23%
    Cor e Forma:Solid
    Peso molecular:1553.72
  • VER49009

    CAS:
    <p>VER49009 (CCT0129397) is an effective HSP90 inhibitor(IC50 =25 nM, Kd=78 nM).</p>
    Fórmula:C19H18ClN3O4
    Pureza:98.95% - >99.99%
    Cor e Forma:Solid
    Peso molecular:387.82
  • Cyclo(RADfK)

    CAS:
    <p>Cyclo(RADfK) is a selective α(v)β(3) integrin ligand used in neoangiogenesis research, therapy, and diagnostics; it's a control for RGD peptides.</p>
    Fórmula:C28H43N9O7
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:617.7
  • Trimethyloctadecylammonium bromide

    CAS:
    <p>Trimethyloctadecylammonium bromide is an inhibitor of Dynamin I(IC50 : 1.9 μM) and also inhibits Dynamin Ⅱ.</p>
    Fórmula:C21H46N·Br
    Pureza:99.09%
    Cor e Forma:Solid Solid
    Peso molecular:392.5
  • E7820

    CAS:
    <p>E7820 (ER68203-00) is an angiogenesis inhibitor by suppressing integrin a2 (a cell adhesion molecule expressed on endothelial cells).</p>
    Fórmula:C17H12N4O2S
    Pureza:98.31% - 99.11%
    Cor e Forma:Solid
    Peso molecular:336.37
  • CK-636

    CAS:
    <p>CK-636 (CK-0944636), an Arp2/3 complex inhibitor, can inhibit actin polymerization induced by the human, fission yeast and bovine Arp2/3 complex.</p>
    Fórmula:C16H16N2OS
    Pureza:98.1% - 98.88%
    Cor e Forma:Solid
    Peso molecular:284.38
  • N-Phenylbenzylamine

    CAS:
    <p>A series of N-Phenylbenzylamine (Benzenemethanamine) as potential cytotoxic and antimitotic agents acting by inhibition of tubulin polymerization</p>
    Fórmula:C13H13N
    Pureza:98.75%
    Cor e Forma:Colorless To Pale Yellow Crystalline Powder
    Peso molecular:183.25
  • Y15

    CAS:
    <p>Y15 (1,2,4,5-Benzenetetramine tetrahydrochlor) is a potent and specificsmall-molecule FAK scaffolding inhibitor that inhibits its autophosphorylation activity,</p>
    Fórmula:C6H14Cl4N4
    Pureza:98% - 99.32%
    Cor e Forma:Dark Brown Crystals
    Peso molecular:284.01
  • Tianeptine sodium salt

    CAS:
    <p>Tianeptine sodium salt 是一种选择性5-HT 摄取促进剂,具有抗抑郁、抗焦虑和神经保护作用,可用于缓解疼痛的研究。</p>
    Fórmula:C21H24ClN2NaO4S
    Pureza:99.82%
    Cor e Forma:Solid
    Peso molecular:458.93
  • Eptifibatide acetate (148031-34-9 free base)

    CAS:
    <p>Eptifibatide acetate (148031-34-9), a cyclic heptapeptide GP IIb/IIIa inhibitor antiplatelet drug.</p>
    Fórmula:C35H49N11O9S2·xC2H4O2
    Pureza:99.7% - 99.87%
    Cor e Forma:Solid
    Peso molecular:831.96 (free base)
  • KNK437

    CAS:
    <p>KNK437 (Heat Shock Protein Inhibitor I), a pan-HSP inhibitor, suppresses the synthesis of inducible HSPs(HSP105, HSP72, and HSP40).</p>
    Fórmula:C13H11NO4
    Pureza:98.90%
    Cor e Forma:Solid
    Peso molecular:245.23
  • TAS-301

    CAS:
    <p>TAS-301, an inhibitor of smooth muscle cell migration and proliferation, inhibits intimal thickening after balloon injury to rat carotid arteries.</p>
    Fórmula:C23H19NO3
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:357.4
  • GNF-7

    CAS:
    <p>GNF-7 is Bcr-Abl WT and Bcr-Abl T315I inhibitor with IC50 of 133 nM and 61 nM, respectively.</p>
    Fórmula:C28H24F3N7O2
    Pureza:97.05% - 99.7%
    Cor e Forma:Solid
    Peso molecular:547.53
  • Verbascoside

    CAS:
    <p>Verbascoside (Kusaginin) is a protein kinase C inhibitor with antimicrobial, anti-inflammatory activities.</p>
    Fórmula:C29H36O15
    Pureza:97.46% - 99.55%
    Cor e Forma:Solid
    Peso molecular:624.59