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Inibidores

Inibidores

Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.

Subcategorias de "Inibidores"

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Foram encontrados 66641 produtos de "Inibidores"

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  • S63845

    CAS:
    <p>S63845 is a selective myeloid leukemia 1(MCL1) inhibitor that binds to human MCL1 with a Kd of 0.19 nM.Cost-effective and quality-assured.</p>
    Fórmula:C39H37ClF4N6O6S
    Pureza:97.7% - ≥98%
    Cor e Forma:Solid
    Peso molecular:829.26
  • Nigakinone

    CAS:
    <p>Nigakinone, isolated from Kumu, is an alkaloid with the pharmacological activity.</p>
    Fórmula:C15H10N2O3
    Pureza:98.66%
    Cor e Forma:Solid
    Peso molecular:266.25
  • Homogentisic acid

    CAS:
    <p>Homogentisic acid: antioxidant with anti-radical effects, protects against thermal cholesterol damage, melanin precursor, and Pfnek-1 inhibitor.</p>
    Fórmula:C8H8O4
    Pureza:98.35% - 99.62%
    Cor e Forma:Solid
    Peso molecular:168.15
  • AN2718

    CAS:
    <p>AN2718, a benzoxaborole, halts fungi protein synthesis by inhibiting LeuRS in molds/yeasts; IC50: 2 μM (A. fumigatus), 4.2 μM (C. albicans).</p>
    Fórmula:C7H6BClO2
    Pureza:98.89% - >99.99%
    Cor e Forma:Solid
    Peso molecular:168.39
  • PD 168568

    CAS:
    <p>PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.</p>
    Fórmula:C22H27N3O
    Cor e Forma:Solid
    Peso molecular:349.47
  • WNK-IN-11

    CAS:
    <p>WNK-IN-11 (Allosteric WNK Kinase Inhibitor) is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)</p>
    Fórmula:C21H21Cl2N5OS
    Pureza:98.32%
    Cor e Forma:Solid
    Peso molecular:462.4
  • 2,5-Dihydroxyacetophenone

    CAS:
    <p>2,5-Dihydroxyacetophenone has anti-anxiety, neuroprotective, anti-inflammatory properties, and modulates cell signaling and melanogenesis.</p>
    Fórmula:C8H8O3
    Pureza:99.75%
    Cor e Forma:Yellow Powder
    Peso molecular:152.15
  • Butylphthalide

    CAS:
    <p>Butylphthalide (3-Butylphthalide) is an anti-cerebral-ischemia drug; first isolated from the seeds of Apium graveolens Linn.</p>
    Fórmula:C12H14O2
    Pureza:98.34%
    Cor e Forma:Solid
    Peso molecular:190.24
  • N-Acetyl-DL-methionine

    CAS:
    <p>N-acetyl-L-methionine equals L-methionine in diet &amp; metabolism, essential for growth and methyl group transfers.</p>
    Fórmula:C7H13NO3S
    Pureza:98.94%
    Cor e Forma:White Crystalline Powder
    Peso molecular:191.25
  • Pargyline

    CAS:
    <p>Pargyline (Pargylamine) is a monoamine oxidase inhibitor with antihypertensive properties.</p>
    Fórmula:C11H13N
    Pureza:95.64% - 97.21%
    Cor e Forma:Solid
    Peso molecular:159.23
  • Sinapine thiocyanate

    CAS:
    <p>Sinapine Thiocyanate, is a derivative of Sinapine (S486605), an alkaloidal amine found in black mustard seeds.</p>
    Fórmula:C16H24NO5·CNS
    Pureza:99.79% - ≥95%
    Cor e Forma:Solid
    Peso molecular:368.45
  • Glabridin

    CAS:
    <p>Glabridin aids in diabetes by reducing inflammation and glucose levels and may prevent liver cancer spread.</p>
    Fórmula:C20H20O4
    Pureza:99.78% - 99.99%
    Cor e Forma:Light Yellow Powder Insoluble In Water
    Peso molecular:324.37
  • Dasotraline

    CAS:
    <p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>
    Fórmula:C16H15Cl2N
    Cor e Forma:Solid
    Peso molecular:292.2
  • PD153035

    CAS:
    <p>PD153035 (NSC-669364) hydrochloride is an effective and selective inhibitor of EGFR (Ki/IC50: 5.2/29 pM, in cell-free assays); little inhibitory against FGFR,</p>
    Fórmula:C16H14BrN3O2
    Pureza:98.47% - 99.29%
    Cor e Forma:Solid
    Peso molecular:360.21
  • Decursin

    CAS:
    <p>Decursin: potential antiepileptic, hepatoprotective, anti-cancer, anti-amnesic; affects NOX activation, PKCα/MAPK/NF-κB pathways, AChE.</p>
    Fórmula:C19H20O5
    Pureza:97.22% - 99.84%
    Cor e Forma:Solid
    Peso molecular:328.36
  • 2,2-Dihydroxy-1-phenylethan-1-one

    CAS:
    <p>2,2-Dihydroxy-1-phenylethan-1-one (Phenylglyoxal hydrate) has antioxidant activity.</p>
    Fórmula:C8H8O3
    Pureza:97.10%
    Cor e Forma:Solid
    Peso molecular:152.15
  • Almotriptan

    CAS:
    <p>Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.</p>
    Fórmula:C17H25N3O2S
    Pureza:99.85%
    Cor e Forma:Light Yellow Or White Power
    Peso molecular:335.46
  • α-Lipoic Acid sodium

    CAS:
    <p>α-Lipoic Acid (Thioctic acid) sodium, an essential cofactor for mitochondrial enzyme complexes, serves as an antioxidant.</p>
    Fórmula:C8H13NaO2S2
    Cor e Forma:Solid
    Peso molecular:228.31
  • Ursocholic acid

    CAS:
    <p>Ursocholic acid, a bile acid found predominantly in bile of mammals.</p>
    Fórmula:C24H40O5
    Pureza:98.89% - 99.62%
    Cor e Forma:Solid
    Peso molecular:408.57
  • Velsecorat

    CAS:
    <p>Velsecorat (AZD7594) is an effective and selective nonsteroidal glucocorticoid receptor modulator (IC50: 0.9 nM).</p>
    Fórmula:C32H32F2N4O6
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:606.62
  • Endoxifen (Z-isomer)

    CAS:
    <p>Endoxifen Z-isomer (EDX) is a key active metabolite of tamoxifen with higher affinity and specificity to estrogen receptors that inhibits aromatase activity.</p>
    Fórmula:C25H27NO2
    Pureza:99.19% - 99.81%
    Cor e Forma:Solid
    Peso molecular:373.49
  • Hydroxy-PEG10-acid

    CAS:
    <p>Hydroxy-PEG10-acid (HO-PEG10-CH2CH2COOH) is a PEG-based PROTAC linker that can be used to synthesize PROTACs[1].</p>
    Fórmula:C23H46O13
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:530.6
  • Gefitinib-based PROTAC 3

    CAS:
    <p>Gefitinib-PROTAC 3 degrades EGFR in cancer cells; DC50s: 11.7 nM (HCC827) and 22.3 nM (H3255).</p>
    Fórmula:C47H57ClFN7O8S
    Pureza:97.29% - 98.25%
    Cor e Forma:Solid
    Peso molecular:934.51
  • Hirsuteine

    CAS:
    <p>Hirsuteine: natural product; blocks nicotine effects on dopamine by hindering ion flow in receptor channels.</p>
    Fórmula:C22H26N2O3
    Pureza:99.36% - 99.83%
    Cor e Forma:Solid
    Peso molecular:366.45
  • Prunin

    CAS:
    <p>Prunin (Naringenin 7-0-glucoside) possesses anti-diabetic, and anti-abacterial properties, it can inhibit protein tyrosine phosphatase 1B (PTP1B) and stimulate</p>
    Fórmula:C21H22O10
    Pureza:99.52% - 99.62%
    Cor e Forma:Solid
    Peso molecular:434.39
  • Glyphosate

    CAS:
    <p>Glyphosate (Atila) is an herbicide. It also is a possible carcinogen to humans.</p>
    Fórmula:C3H8NO5P
    Pureza:99.12% - 99.91%
    Cor e Forma:White Crystals (Darkens) Ph (1% Solution In Water) 2 5 (Ntp 1992)
    Peso molecular:169.07
  • Selonsertib HCl

    CAS:
    <p>Selonsertib (GS-4997) is an oral ASK1 inhibitor with potential anti-inflammatory, antineoplastic, and anti-fibrotic effects.</p>
    Fórmula:C24H25ClFN7O
    Cor e Forma:Solid
    Peso molecular:481.96
  • Pentagastrin

    CAS:
    <p>Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis of</p>
    Fórmula:C37H49N7O9S
    Pureza:96.98% - 99.49%
    Cor e Forma:Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water Solid
    Peso molecular:767.89
  • Ipsapirone hydrochloride

    CAS:
    <p>Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.</p>
    Fórmula:C19H24ClN5O3S
    Cor e Forma:Solid
    Peso molecular:437.94
  • Pencycuron

    CAS:
    <p>Pencycuron (Monceren) is a phenylurea fungicide.</p>
    Fórmula:C19H21ClN2O
    Pureza:99.45%
    Cor e Forma:Red Liquid With A Slight Characteristic Odor
    Peso molecular:328.84
  • KF38789

    CAS:
    <p>KF38789 is a selective inhibitor of P-selectin-mediated cell adhesion and P-selectin immunoglobulin G chimeric protein.</p>
    Fórmula:C19H21NO5S
    Pureza:97.29% - 98.15%
    Cor e Forma:Solid
    Peso molecular:375.44
  • kaempferide

    CAS:
    <p>kaempferide (4'-Methylkaempferol) is an O-methylated flavonol present in Kaempferia kaempferi with antiviral activity.</p>
    Fórmula:C16H12O6
    Pureza:98.31% - 99.66%
    Cor e Forma:Solid
    Peso molecular:300.26
  • 4,4'-Dimethoxychalcone

    CAS:
    <p>4,4'-Dimethoxychalcone (4,4-Dimethoxychalcone) is a natural product.</p>
    Fórmula:C17H16O3
    Pureza:99.57%
    Cor e Forma:Solid
    Peso molecular:268.31
  • Clindamycin hydrochloride

    CAS:
    <p>Clindamycin hydrochloride (Clinimycin HCl) inhibits protein synthesis by acting on the 50S ribosomal. Clindamycin is a chlorinated broad-spectrum antibiotic.</p>
    Fórmula:C18H33ClN2O5S·HCl
    Pureza:99.80%
    Cor e Forma:White Crystalline Powder
    Peso molecular:461.44
  • Ceftaroline fosamil

    CAS:
    <p>Ceftaroline fosamil (TAK-599) is a cephalosporin, with activity against Gram-positive pathogens.</p>
    Fórmula:C24H25N8O10PS4
    Pureza:97.09% - ≥98%
    Cor e Forma:Solid
    Peso molecular:744.74
  • Punicalagin

    CAS:
    <p>Punicalagin, an ellagitannin in pomegranates, has antioxidant, anti-inflammatory, anticancer properties, and combats heart issues from high-fat diets.</p>
    Fórmula:C48H28O30
    Pureza:98% - 99.7%
    Cor e Forma:White Crystalline Powder
    Peso molecular:1084.72
  • Nystose

    CAS:
    <p>Nystose (1,1-Kestotetraose) is a tetrasaccharide composed of two fructose molecules linked via beta (1→2) bonds to the fructosyl moiety of sucrose.</p>
    Fórmula:C24H42O21
    Pureza:98% - 99.93%
    Cor e Forma:Solid
    Peso molecular:666.58
  • 6-O-Methyl Guanosine

    CAS:
    <p>6-O-Methyl Guanosine inhibit colony-forming ability in a malignant xeroderma pigmentosum cell line.</p>
    Fórmula:C11H15N5O5
    Pureza:97.5%
    Cor e Forma:Solid
    Peso molecular:297.27
  • Remibrutinib

    CAS:
    <p>Remibrutinib inhibits BTK activity with an IC50 value of 0.023 μM in blood.</p>
    Fórmula:C27H27F2N5O3
    Pureza:99.5% - 99.81%
    Cor e Forma:Solid
    Peso molecular:507.53
  • Liensinine diperchlorate

    CAS:
    <p>Liensinine Diperchlorate is an isoquinoline alkaloid extracted from the embryonic seeds of the sacred lotus.</p>
    Fórmula:C37H44Cl2N2O14
    Pureza:99.8% - ≥95%
    Cor e Forma:Solid
    Peso molecular:811.67
  • Atractylodin

    CAS:
    <p>Atractylodin inhibits lipase (IC50: 39.12 µM) and repels T. castaneum adults (LD50: 1.83 µg/cm, &gt;90% repellency at 0.63 µg/cm).</p>
    Fórmula:C13H10O
    Pureza:99.35% - 99.74%
    Cor e Forma:Solid
    Peso molecular:182.22
  • Diclofensine hydrochloride

    CAS:
    <p>Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂,在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。</p>
    Fórmula:C17H18Cl3NO
    Pureza:98.86% - 99.93%
    Cor e Forma:Solid
    Peso molecular:358.69
  • LOXO-195

    CAS:
    <p>(6RS)-LOXO-195 (BAY 2731954) is a potent and selective Trk tyrosine kinase inhibitor.</p>
    Fórmula:C20H21FN6O
    Pureza:99.54%
    Cor e Forma:Solid
    Peso molecular:380.42
  • S 38093

    CAS:
    <p>S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).</p>
    Fórmula:C17H24N2O2
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:288.38
  • Camelliaside B

    CAS:
    <p>Camelliaside B possesses deglycosylation activity.</p>
    Fórmula:C32H38O19
    Pureza:95.92% - 99.92%
    Cor e Forma:Solid
    Peso molecular:726.63
  • Bafetinib

    CAS:
    <p>Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.</p>
    Fórmula:C30H31F3N8O
    Pureza:94.16% - 99.68%
    Cor e Forma:Solid
    Peso molecular:576.62
  • 3,4-Dimethoxycinnamic acid

    CAS:
    <p>3,4-Dimethoxycinnamic acid, a monomer in Securidaca inappendiculata, prevents cell death in L-02 cells via ROS pathways.</p>
    Fórmula:C11H12O4
    Pureza:99.51%
    Cor e Forma:Yellow To Beige Crystals
    Peso molecular:208.21
  • RX-3117

    CAS:
    <p>RX-3117 (fluorocyclopentenylcytosine) is a novel a cytidine analog.</p>
    Fórmula:C10H12FN3O4
    Pureza:97.46%
    Cor e Forma:Solid
    Peso molecular:257.22
  • Trovirdine

    CAS:
    <p>Trovirdine (LY300046) is a thiourea non-nucleoside reverse transcriptase inhibitor.</p>
    Fórmula:C13H13BrN4S
    Pureza:98.12% - 98.50%
    Cor e Forma:Solid
    Peso molecular:337.24
  • ORY1001

    CAS:
    <p>ORY1001: Oral LSD1/KDM1A inhibitor, highly selective, IC50 &lt;20 nM.</p>
    Fórmula:C15H22N2·2HCl
    Pureza:99.85% - 99.96%
    Cor e Forma:Solid
    Peso molecular:303.27
  • 3,4-Dihydroxyflavone

    CAS:
    <p>3,4-Dihydroxyflavone Acts as an Antioxidant and Antiapoptotic Agent .</p>
    Fórmula:C15H10O4
    Pureza:97.18%
    Cor e Forma:Solid
    Peso molecular:254.24
  • Angiotensin (1-7)

    CAS:
    <p>Angiotensin (1-7) (ASP-ARG-VAL-TYR-ILE-HIS-PRO) is a synthetic heptapeptide, inhibits canine ACE activity with vasodilator and antiproliferative activities.</p>
    Fórmula:C41H62N12O11
    Pureza:>99.99%
    Cor e Forma:White Lyophilised Solid
    Peso molecular:899
  • N-terminally acetylated Leu-enkephalin


    <p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>
    Fórmula:C30H39N5O8
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:597.66
  • Theaflavin 3,3′-digallate

    CAS:
    <p>Theaflavin 3,3'-digallate, a major polyphenol found in black tea, is an inducer of oxidative stress which has anti-inflammatory and cancer</p>
    Fórmula:C43H32O20
    Pureza:98.71% - 99.86%
    Cor e Forma:Solid
    Peso molecular:868.7
  • CPFX4158

    CAS:
    <p>CPFX4158 is a mannose deriviative and an antibacterial agent that is potentially useful in transgenic humanized- CEACAM6 mouse.</p>
    Fórmula:C51H55NO19
    Pureza:98.37%
    Cor e Forma:Solid
    Peso molecular:985.98
  • GW786034B

    CAS:
    <p>Pazopanib HCl (Votrient) inhibits VEGFR1-3, PDGFR, FGFR, c-Kit, c-Fms with IC50 range 10-146 nM in cell-free assays.</p>
    Fórmula:C21H23N7O2S·HCl
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:473.98
  • Ruxolitinib

    CAS:
    <p>Ruxolitinib (INCB018424) is a JAK1/2 inhibitor (IC50=3.3/2.8 nM) that is potent and selective.</p>
    Fórmula:C17H18N6
    Pureza:99.4% - >99.99%
    Cor e Forma:Solid
    Peso molecular:306.36
  • β-Glycerophosphate disodium salt hydrate

    CAS:
    <p>β-Glycerophosphate is a classical serine-threonine phosphatase inhibitor used in kinase reaction buffers.</p>
    Fórmula:C3H7O6PNa2·xH2O
    Pureza:99.83% - ≥98%
    Cor e Forma:Solid
    Peso molecular:234.05
  • EHop-016

    CAS:
    <p>EHop-016 is a specific Rac GTPase inhibitor with IC50 of 1.1 μM for Rac1 in MDA-MB-231 and MDA-MB-435 cells, equally effective inhibition for Rac3.</p>
    Fórmula:C25H30N6O
    Pureza:98.99% - >99.99%
    Cor e Forma:Solid
    Peso molecular:430.55
  • BAY-545

    CAS:
    <p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>
    Fórmula:C18H22F3N3O4S
    Pureza:98.05%
    Cor e Forma:Solid
    Peso molecular:433.45
  • Dovitinib

    CAS:
    <p>Dovitinib is an orally active, multi-targeted tyrosine kinase (RTK) inhibitor with anti-tumor effects.Cost-effective and quality-assured.</p>
    Fórmula:C21H21FN6O
    Pureza:99.35% - 99.92%
    Cor e Forma:Solid
    Peso molecular:392.43
  • BI-69A11

    CAS:
    <p>BI-69A11 is a dual AKT/NFkB inhibitor, increasing colon cancer cell sensitivity to mda-7/IL-24.</p>
    Fórmula:C25H16ClN3O2
    Pureza:96.97%
    Cor e Forma:Solid
    Peso molecular:425.87
  • PROPYL DISULFIDE

    CAS:
    <p>PROPYL DISULFIDE is a natural product.</p>
    Fórmula:C6H14S2
    Pureza:97.67%
    Cor e Forma:Liquid
    Peso molecular:150.31
  • Azomycin

    CAS:
    <p>Azomycin (Ro 05-9129) is an antimicrobial antibiotic produced by a strain of Nocardia mesenterica.</p>
    Fórmula:C3H3N3O2
    Pureza:≥95%
    Cor e Forma:Yellow Orange Powder
    Peso molecular:113.07
  • Presatovir

    CAS:
    <p>Presatovir (GS-5806) (GS-5806) is a novel, orally bioavailable RSV fusion inhibitor (mean EC50: 0.43 nM).</p>
    Fórmula:C24H30ClN7O3S
    Pureza:99.14% - 99.92%
    Cor e Forma:Solid
    Peso molecular:532.06
  • Mirogabalin

    CAS:
    <p>Mirogabalin (DS5565) is a calcium channel blocker with analgesic effects.</p>
    Fórmula:C12H19NO2
    Pureza:98.57%
    Cor e Forma:Solid
    Peso molecular:209.28
  • Tazarotenic acid

    CAS:
    <p>Tazarotenic acid (AGN-190299) is a retinoid prodrug which is converted to its active form</p>
    Fórmula:C19H17NO2S
    Pureza:97.83%
    Cor e Forma:Solid
    Peso molecular:323.41
  • Ginsenoside Rb2

    CAS:
    <p>Ginsenoside Rb2 (Ginsenoside C) found in species of Panax, upregulating GPR120 gene expression.</p>
    Fórmula:C53H90O22
    Pureza:99.01% - 99.93%
    Cor e Forma:White Powder
    Peso molecular:1079.27
  • Vorapaxar sulfate

    CAS:
    <p>Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.</p>
    Fórmula:C29H35FN2O8S
    Pureza:99.9% - >99.99%
    Cor e Forma:Solid
    Peso molecular:590.66
  • Grazoprevir

    CAS:
    <p>Grazoprevir (MK-5172) is a protease inhibitor targeting hepatitis C virus NS3/4A used for treating chronic HCV genotypes 1 or 4 infections. Cost-effective and quality-assured.</p>
    Fórmula:C38H50N6O9S
    Pureza:99.36% - >99.99%
    Cor e Forma:Solid
    Peso molecular:766.9
  • B7/CD28 interaction inhibitor 1

    CAS:
    <p>B7/CD28 interaction inhibitor 1 (CTLA-4 inhibitor) is a potent CTLA-4 inhibitor.</p>
    Fórmula:C21H13F4N5O
    Pureza:99.5% - 99.63%
    Cor e Forma:Solid
    Peso molecular:427.35
  • AZD9496

    CAS:
    <p>AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.</p>
    Fórmula:C25H25F3N2O2
    Pureza:97.28% - 98.47%
    Cor e Forma:Solid
    Peso molecular:442.47
  • SHR0302

    CAS:
    <p>SHR0302 (ARQ252) is a JAK inhibitor that binds JAK1 with stronger affinity than others (Selectivity for JAK1 is more than 10 times for JAK2, 77 times for JAK3,</p>
    Fórmula:C18H22N8O2S
    Pureza:99.11%
    Cor e Forma:Solid
    Peso molecular:414.48
  • Oxysanguinarine

    CAS:
    <p>Oxysanguinarine (Hydroxysanguinarine) possesses antiplatelet aggregation activity, it has potential inhibitory properties against the dengue virus.</p>
    Fórmula:C20H13NO5
    Pureza:99.57%
    Cor e Forma:Solid
    Peso molecular:347.32
  • RG13022

    CAS:
    <p>RG13022 (Tyrphostin RG13022) is a tyrosine kinase inhibitor; inhibits the autophosphorylation reaction of the EGF receptor (IC50: 4 μM).</p>
    Fórmula:C16H14N2O2
    Pureza:98.38%
    Cor e Forma:Solid
    Peso molecular:266.29
  • D-JNKI-1 acetate


    <p>D-JNKI-1 acetate (AM-111 acetate) is a highly potent and cell-permeable peptide inhibitor of JNK.</p>
    Fórmula:C166H290N66O42
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:3882.5
  • Ethyl cinnamate

    CAS:
    <p>Ethyl cinnamate has antifungal, and vasorelaxant effects.</p>
    Fórmula:C11H12O2
    Pureza:99.53%
    Cor e Forma:Liquid
    Peso molecular:176.21
  • Neurokinin A

    CAS:
    <p>Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.</p>
    Fórmula:C50H80N14O14S
    Pureza:>99.99%
    Cor e Forma:White To Off-White Lyophilized Solid
    Peso molecular:1133.32
  • GSK591

    CAS:
    <p>GSK591 (GSK3203591), Alternative Names are EPZ015866, GSK3203591, is a potent selective inhibitor of the arginine methyltransferase PRMT5 (IC50=11 nM).</p>
    Fórmula:C22H28N4O2
    Pureza:99.35% - 99.45%
    Cor e Forma:Solid
    Peso molecular:380.48
  • Methyl 2-(1H-indol-3-yl)acetate

    CAS:
    <p>Methyl indole-3-acetate, in apples, is isolated from seeds of peas, Vicia, soybeans, and beans.</p>
    Fórmula:C11H11NO2
    Pureza:98.13%
    Cor e Forma:White To Yellow Powder
    Peso molecular:189.21
  • Cadazolid

    CAS:
    <p>Cadazolid (ACT-179811) is an oxazolidinone-type antibiotic, with activity against gram-positive bacteria, including Clostridium difficile.</p>
    Fórmula:C29H29F2N3O8
    Pureza:98.1% - 99.9%
    Cor e Forma:Solid
    Peso molecular:585.55
  • Dymanthine

    CAS:
    <p>Dymanthine (ADMA 18) is an agent of veterinary anthelmintic.</p>
    Fórmula:C20H43N
    Pureza:99.85%
    Cor e Forma:Colorless To White Solid Or Semi-Solid Or Liquid
    Peso molecular:297.56
  • Vonoprazan fumarate

    CAS:
    <p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>
    Fórmula:C17H16FN3O2S·C4H4O4
    Pureza:99.16% - 99.98%
    Cor e Forma:Solid
    Peso molecular:461.46
  • UNC926 hydrochloride

    CAS:
    <p>UNC926 hydrochloride is a methyl-lysine (Kme) reader domain inhibitor.</p>
    Fórmula:C16H22BrClN2O
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:373.72
  • 5-Fluoroorotic acid

    CAS:
    <p>5-Fluoroorotic acid is an inhibitor of thymidylate synthase.</p>
    Fórmula:C5H3FN2O4
    Pureza:99.7% - >99.99%
    Cor e Forma:White To Pale Yellow Powder
    Peso molecular:174.09
  • PfDHODH-IN-1

    CAS:
    <p>PfDHODH-IN-1 is an inhibitor of Plasmodium falciparum dihydroorotate dehydrogenase(PfDHODH) which catalyzes the rate-limiting step for DNA and RNA biosynthesis.</p>
    Fórmula:C14H11F3N2O2
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:296.24
  • Glycyl-L-leucine

    CAS:
    <p>Glycyl-L-leucine (Gly-Leu) is a substrate for the assay of glycyl-L-leucine dipeptidase.</p>
    Fórmula:C8H16N2O3
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:188.22
  • NRC-2694 dihydrochloride

    CAS:
    <p>NRC-2694 dihydrochloride is an epidermal growth factor receptor (EGFR) antagonist potentially for the treatment of solid tumors.</p>
    Fórmula:C24H28Cl2N4O3
    Cor e Forma:Solid
    Peso molecular:491.41
  • GeA-69

    CAS:
    <p>GeA-69 (GeA69) is a selective and allosteric PARP14 macrodomain 2 (MD2) inhibitor (Kd: 0.86 μM in ITC assays).</p>
    Fórmula:C20H16N2O
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:300.35
  • coreopsin

    CAS:
    <p>Coreopsin, from Coreopsis tinctoria, treats hypertension, diabetes, and helps in weight and fat reduction.</p>
    Fórmula:C21H22O10
    Pureza:99.47%
    Cor e Forma:Solid
    Peso molecular:434.39
  • Dimethylcurcumin

    CAS:
    <p>Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer.</p>
    Fórmula:C23H24O6
    Pureza:97.36% - 98.96%
    Cor e Forma:Solid
    Peso molecular:396.43
  • TH287

    CAS:
    <p>TH287 is a potent inhibitor of MTH1 (NUDT1), less potent for MTH2, NUDT5, NUDT12, NUDT14, and NUDT16.</p>
    Fórmula:C11H10Cl2N4
    Pureza:97.73% - 99%
    Cor e Forma:Solid
    Peso molecular:269.13
  • 1-Methyl-2-(Methylthio)iMidazole

    CAS:
    <p>1-Methyl-2-(methylthio)imidazole is an impurity of Methimazole and a thiourea antithyroid agent.</p>
    Fórmula:C5H8N2S
    Pureza:99.34%
    Cor e Forma:Solid
    Peso molecular:128.2
  • Oxibendazole

    CAS:
    <p>Oxibendazole: a benzimidazole antiparasitic for horses and pets against various worms.</p>
    Fórmula:C12H15N3O3
    Pureza:99.3% - 99.88%
    Cor e Forma:Crystalline Solid
    Peso molecular:249.27
  • Skepinone-L

    CAS:
    <p>Skepinone-L (CBS3830) is a selective p38 mitogen-activated protein kinase inhibitor.</p>
    Fórmula:C24H21F2NO4
    Pureza:99.56% - >99.99%
    Cor e Forma:Solid
    Peso molecular:425.42
  • MRE-269

    CAS:
    <p>MRE-269 (ACT-333679) is an orally available and long-acting prostacyclin receptor agonist prodrug, used for the treatment of pulmonary arterial hypertension.</p>
    Fórmula:C25H29N3O3
    Pureza:98.25%
    Cor e Forma:Solid
    Peso molecular:419.52
  • 4BP-TQS

    CAS:
    <p>4BP-TQS is an allosteric agonist of α7 nAChRs.</p>
    Fórmula:C18H17BrN2O2S
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:405.31
  • Secologanoside

    CAS:
    <p>Secologanoside shows anti-complementary, allelopathic, and anti-elastase activities.</p>
    Fórmula:C16H22O11
    Pureza:98.70% - 99.36%
    Cor e Forma:Solid
    Peso molecular:390.34
  • Cichoriin

    CAS:
    <p>Cichoriin is a photosensitive compound, it could be used as herbal photosensitizing agent in treating benign breast tumor in rats.</p>
    Fórmula:C15H16O9
    Pureza:99.75% - 99.99%
    Cor e Forma:Solid
    Peso molecular:340.28
  • Ochromycinone

    CAS:
    <p>Ochromycinone (STA 21) is a selective STAT3 inhibitor.</p>
    Fórmula:C19H14O4
    Pureza:99.21%
    Cor e Forma:Solid
    Peso molecular:306.31