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Inibidores

Inibidores

Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.

Subcategorias de "Inibidores"

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Foram encontrados 66676 produtos de "Inibidores"

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  • MELK-8a

    CAS:
    <p>MELK-8a inhibits MELK kinase crucial for cancer cell mitosis (IC50: 2 nM).</p>
    Fórmula:C25H32N6O
    Cor e Forma:Solid
    Peso molecular:432.56
  • Gynostemma Extract

    CAS:
    Gynostemma Extract (Gypenoside IX) is a saponins extract derived from the Gynostemma pentaphyllum.
    Fórmula:C47H80O17
    Pureza:98% - 99.6%
    Cor e Forma:Solid
    Peso molecular:917.13
  • PHGDH-inactive

    CAS:
    PHGDH inactive is inactive against PHGDH and serves as a negative control for NCT-502 and NCT-503 [1].
    Fórmula:C17H21N5S
    Pureza:99.83%
    Cor e Forma:Solid
    Peso molecular:327.45
  • DiD perchlorate

    CAS:
    DiD perchlorate is a lipophilic cyanine dye that can be used in cells tracking.
    Fórmula:C61H99ClN2O4
    Pureza:99.65%
    Cor e Forma:Solid
    Peso molecular:959.9
  • Nelociguat

    CAS:
    <p>Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.</p>
    Fórmula:C19H17FN8O2
    Pureza:99.19%
    Cor e Forma:Solid
    Peso molecular:408.39
  • Lophanthoidin E

    CAS:
    <p>Lophanthoidin E is a kind of natural product derived from the herbs of Rabdosia lophanthoides.</p>
    Fórmula:C22H30O7
    Pureza:98.00%
    Cor e Forma:Solid
    Peso molecular:406.47
  • NS309

    CAS:
    NS309 activates SK/KCa2, IK/KCa3.1 (0.12-1.2 μM EC50, 10-90 nM EC50), and Kv11.1 channels; doesn't affect BK/KCa1.1; modulates neuronal firing.
    Fórmula:C8H4Cl2N2O2
    Pureza:97.55%
    Cor e Forma:Solid
    Peso molecular:231.04
  • 6-Bromo-3-methyl-1,4-dihydroquinazolin-2-one

    CAS:
    CHEMBRDG-BB 7118966 is an inhibitor of Bromodomain-containing protein 4 (human).
    Fórmula:C9H9BrN2O
    Pureza:99.28%
    Cor e Forma:Solid
    Peso molecular:241.08
  • Procyanidin B1

    CAS:
    Procyanidin B1, isolated from commonly eaten fruits, binds to the TLR4/MD-2 complex and has anti-inflammatory activity.
    Fórmula:C30H26O12
    Pureza:98.00% - 99.91%
    Cor e Forma:Red-Brown Powder
    Peso molecular:578.52
  • Arachidonic acid

    CAS:
    Arachidonic acid: essential unsaturated fat, in liver/brain/organs, from linoleic acid, leads to prostaglandins, thromboxanes, leukotrienes.
    Fórmula:C20H32O2
    Pureza:99.21% - ≥98%
    Cor e Forma:Solid
    Peso molecular:304.47
  • Tyrphostin AG 528

    CAS:
    Tyrphostin AG 528 (Tyrphostin B66) is an inhibitor of EGFR (IC50: 4.9 μM) and ErbB2 (IC50: 2.1 μM).
    Fórmula:C18H14N2O3
    Pureza:99.64%
    Cor e Forma:Solid
    Peso molecular:306.32
  • PF-431396

    CAS:
    PF-431396 is a dual PYK2/FAK inhibitor (IC50: 11/2 nM).
    Fórmula:C22H21F3N6O3S
    Pureza:98.83% - 99.82%
    Cor e Forma:Solid
    Peso molecular:506.5
  • Methenamine Hippurate

    CAS:
    <p>Methenamine Hippurate is a component of Hiprex, with antibacterial activity.</p>
    Fórmula:C15H21N5O3
    Pureza:99.69% - 99.72%
    Cor e Forma:White Crystalline Powder
    Peso molecular:319.36
  • LF3

    CAS:
    LF3 is a specific inhibitor of canonical Wnt signaling by disrupting the interaction between β-catenin and TCF4 (IC50 < 2 μM)
    Fórmula:C20H24N4O2S2
    Pureza:99.63%
    Cor e Forma:Solid
    Peso molecular:416.56
  • 1,5-diphenylpyrazole-3-carboxylic acid

    CAS:
    1,5-diphenylpyrazole-3-carboxylic acid (1H-PYRAZOLE-3-CARBOXYLIC ACID, 1,5-DIPHENYL-) is a plant-physiologically tolerable salt radical or any desired ester
    Fórmula:C16H12N2O2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:264.28
  • [D-Phe12]-Bombesin acetate


    <p>[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.</p>
    Fórmula:C76H116N22O20S
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:1689.94
  • [D-Trp8]-γ-MSH acetate(321351-81-9 free base)


    [D-Trp8]-γ-MSH acetate(321351-81-9 free base) is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and
    Fórmula:C76H103N21O18S
    Pureza:99.75%
    Cor e Forma:Solid
    Peso molecular:1630.82
  • Deguelin

    CAS:
    Deguelin ((-)-Deguelin) is a PI3K/AKT Inhibitor, which is a natural product isolated from plants in the Mundulea sericea family.
    Fórmula:C23H22O6
    Pureza:96.39% - 99.29%
    Cor e Forma:Solid
    Peso molecular:394.42
  • GNF-5

    CAS:
    GNF-5, non-ATP Bcr-Abl inhibitor (IC50: 0.22±0.1 uM, wild-type), improves upon GNF-2 with better pharmacokinetics.
    Fórmula:C20H17F3N4O3
    Pureza:98% - 99.94%
    Cor e Forma:Solid
    Peso molecular:418.37
  • 2-Undecanol

    CAS:
    <p>2-Undecanol, a male pheromone from Lobiopa insularis, is also a floral volatile used by Hymenoptera species.</p>
    Fórmula:C11H24O
    Pureza:98%
    Cor e Forma:Clear Colorless Liquid
    Peso molecular:172.31
  • [(2-Methoxyphenoxy)Methyl]Oxirane

    CAS:
    [(2-Methoxyphenoxy)Methyl]Oxirane is a natural product.
    Fórmula:C10H12O3
    Pureza:97.61%
    Cor e Forma:White Solid Crystalline
    Peso molecular:180.2
  • Talinolol

    CAS:
    (±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
    Fórmula:C20H33N3O3
    Pureza:98.8%
    Cor e Forma:Solid
    Peso molecular:363.49
  • 1-​Furfurylpyrrole

    CAS:
    1-Furfurylpyrrole is a potential contributor of flavor and aroma to popcorn.
    Fórmula:C9H9NO
    Pureza:97.85%
    Cor e Forma:Liquid
    Peso molecular:147.17
  • Rhapontin

    CAS:
    Rhapontin may reduce liver fat and better blood sugar/lipids, showing potential for treating type 2 diabetes.
    Fórmula:C21H24O9
    Pureza:99% - 99.91%
    Cor e Forma:Light Yellow
    Peso molecular:420.41
  • 1-Dodecanol

    CAS:
    1-Dodecanol: a coconut-derived fatty alcohol with floral scent, used in detergents, lubricants, pesticides, and pharma.
    Fórmula:C12H26O
    Pureza:99.88%
    Cor e Forma:Colourless Solid Paraffin Like
    Peso molecular:186.33
  • PRIMA-1

    CAS:
    PRIMA-1 (NSC-281668) is a mutant p53 reactivator. It induces apoptosis and inhibits growth of human tumors with mutant p53.
    Fórmula:C9H15NO3
    Pureza:99.22%
    Cor e Forma:Solid
    Peso molecular:185.22
  • (2S)-2'-Methoxykurarinone

    CAS:
    (2S)-2'-Methoxykurarinone is isolated from the roots of Sophora flavescens.
    Fórmula:C27H32O6
    Pureza:97.00% - 99.44%
    Cor e Forma:Solid
    Peso molecular:452.54
  • Zebularine

    CAS:
    Zebularine (4-Deoxyuridine) is a DNA methylation inhibitor.
    Fórmula:C9H12N2O5
    Pureza:99.04% - >99.99%
    Cor e Forma:Solid
    Peso molecular:228.2
  • PS47

    CAS:
    PS-47(PS 47) is an inactive E-isomer of PS48. PS48 is an activator of PDK1.
    Fórmula:C17H15ClO2
    Pureza:99.09%
    Cor e Forma:Solid
    Peso molecular:286.75
  • RO495

    CAS:
    <p>RO495 (CS-2667), a potent inhibitor of TYK2, inhibits TYK2 with IC50 of 1.5nM as tested in cell-based pharmacological assays</p>
    Fórmula:C17H14Cl2N6O
    Pureza:97.94%
    Cor e Forma:Solid
    Peso molecular:389.24
  • Morpholinylmercaptobenzothiazole

    CAS:
    Morpholinylmercaptobenzothiazole is an aftereffect rapid vulcanization accelerator
    Fórmula:C11H12N2OS2
    Pureza:95%
    Cor e Forma:Light Tan Solid Powder
    Peso molecular:252.36
  • EDANS sodium

    CAS:
    EDANS sodium (5-(2-Aminoethylamino)-1-naphthalenesulfonic acid sodium salt) is a donor for developing FRET-based nucleic acid probes that is widely used in real
    Fórmula:C12H13N2NaO3S
    Pureza:98%
    Cor e Forma:Light Yellow Powder
    Peso molecular:288.3
  • Narirutin

    CAS:
    Narirutin combats cell growth, oxidation, allergies, and inflammation.
    Fórmula:C27H32O14
    Pureza:99.23% - 99.86%
    Cor e Forma:Off White Powder
    Peso molecular:580.53
  • Methyl cellulose

    CAS:
    Methylcellulose is a natural polymer that gels on heating. Methylcellulose is not toxic.
    Fórmula:C20H38O11
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:454.51(Monomer)
  • TP0463518

    CAS:
    TP-0463518 is a highly potent HIF prolyl hydroxylase (PHD) inhibitor (IC50s: 13 nM and 18 nM for human and rat PHD2, respectively).
    Fórmula:C20H18ClN3O6
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:431.83
  • RGFP966

    CAS:
    RGFP966 is an HDAC3 inhibitor (IC50: 0.08 μM) and does not affect other HDACs at concentrations up to 15 μM.
    Fórmula:C21H19FN4O
    Pureza:99.2% - 99.88%
    Cor e Forma:Solid
    Peso molecular:362.4
  • Biocytin

    CAS:
    <p>Biocytin, a D-biotin and L-lysine conjugate, maps brain connections via a secondary amide bond.</p>
    Fórmula:C16H28N4O4S
    Pureza:97.23%
    Cor e Forma:White Solid
    Peso molecular:372.48
  • Pseudolaric acid B β-D-glucoside

    CAS:
    Pseudolaric acid B β-D-glucoside (Pseudolaric acid B-glucopyranoside) is a natural product from Pseudolarix amabilis.
    Fórmula:C29H38O13
    Pureza:98.55% - ≥95%
    Cor e Forma:Solid
    Peso molecular:594.60
  • Nexturastat A

    CAS:
    Nexturastat A is an effective and specific HDAC6 inhibitor (IC50: 5 nM). Its selectivity is >190-fold than other HDACs.
    Fórmula:C19H23N3O3
    Pureza:99.40% - 99.57%
    Cor e Forma:Solid
    Peso molecular:341.4
  • Paris saponin VII

    CAS:
    <p>Paris saponin VII (Dioscini) shows inhibitory effects on cell proliferation.</p>
    Fórmula:C51H82O21
    Pureza:99.51% - 99.63%
    Cor e Forma:Solid
    Peso molecular:1031.18
  • MD2-IN-1

    CAS:
    MD2-IN-1 is a Myeloid differentiation protein 2 (MD2) inhibitor with a KD of 189  μM for the recombinant human MD2 (rhMD2).
    Fórmula:C20H22O6
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:358.39
  • Kansuinine A

    CAS:
    Kansuinine A, a 95% ethanol extract from the roots of E. kansui, possesses an inhibitory effect on IL-6-induced Stat3 activation by activating ERK1/2.
    Fórmula:C37H46O15
    Pureza:99.28%
    Cor e Forma:Solid
    Peso molecular:730.75
  • (S)-CPI203

    CAS:
    <p>CPI-203 is an effective BET bromodomain inhibitor (IC50: 37 nM for BRD4).</p>
    Fórmula:C19H18ClN5OS
    Pureza:99.01% - 99.92%
    Cor e Forma:Solid
    Peso molecular:399.9
  • CGS 21680 Hydrochloride

    CAS:
    CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.
    Fórmula:C23H29N7O6·HCl
    Pureza:96.74% - 99.53%
    Cor e Forma:Solid
    Peso molecular:535.98
  • Rabeprazole sodium

    CAS:
    <p>Rabeprazole sodium treats stomach ulcers and Zollinger-Ellison syndrome, blocking ATPase in gastric cells.</p>
    Fórmula:C18H20N3NaO3S
    Pureza:98% - 99.912%
    Cor e Forma:White Or Off White Crystalline Powder
    Peso molecular:381.42
  • Linocinnamarin

    CAS:
    <p>Linocinnamarin, from strawberries, blocks degranulation by inactivating Syk/PLCgamma.</p>
    Fórmula:C16H20O8
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:340.33
  • AP1189 acetate

    CAS:
    <p>AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.</p>
    Fórmula:C16H18N6O4
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:358.35
  • trans-Cinnamaldehyde

    CAS:
    Trans-Cinnamaldehyde (Phenylacrolein) exhibits anti-inflammatory activities and antidepressant-like effects in stressed mid-aged rats as a COX-2 inhibitor.
    Fórmula:C9H8O
    Pureza:98.07%
    Peso molecular:132.16
  • ICI 63197

    CAS:
    ICI 63197 (2-Amino-6-methyl-4-propyl-[1,2,4]triazolo[1,5-a]pyrimidin-5(4H)-one) is a PDE4 inhibitor.
    Fórmula:C9H13N5O
    Pureza:99.70%
    Cor e Forma:White Solid
    Peso molecular:207.23
  • SMIFH2

    CAS:
    <p>SMIFH2 is formin homology 2 (FH2) domains inhibitor.</p>
    Fórmula:C15H9BrN2O3S
    Pureza:97.41%
    Cor e Forma:Solid
    Peso molecular:377.21
  • Laurdan

    CAS:
    <p>Laurdan (6-Dodecanoyl-2-dimethylaminonaphthalene) is a fluorescent membrane probe that is spectrally sensitive to the phospholipid phase of the cell membrane to</p>
    Fórmula:C24H35NO
    Pureza:98.73% - 99.02%
    Cor e Forma:Solid
    Peso molecular:353.54
  • Esculentoside H

    CAS:
    Phytolaccaceae has anti-tumor activity, the mechanism may be related to the capacity of Esculentoside H for TNF release.
    Fórmula:C48H76O21
    Pureza:98.04% - 99.3%
    Cor e Forma:Solid
    Peso molecular:989.1
  • Cephapirin Benzathine

    CAS:
    <p>Cephapirin Benzathine is a semisynthetic, broad-spectrum, first-generation cephalosporin with antibacterial activity.</p>
    Fórmula:C17H17N3O6S2C16H20N2
    Pureza:98% - 99.38%
    Cor e Forma:Solid
    Peso molecular:543.63
  • Pempidine HCl

    CAS:
    Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.
    Fórmula:C10H22ClN
    Cor e Forma:Solid
    Peso molecular:191.74
  • NVP-BAW2881

    CAS:
    NVP-BAW2881 (BAW2881) is a potent and selective VEGFR inhibitor with activity to inhibit chronic and acute skin inflammation.
    Fórmula:C22H15F3N4O2
    Pureza:98.19% - 99.97%
    Cor e Forma:Solid
    Peso molecular:424.38
  • Autocamtide-2-related inhibitory peptide

    CAS:
    <p>Autocamtide-2-related inhibitory peptide is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.</p>
    Fórmula:C64H116N22O19
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:1497.74
  • Acid-C1-PEG5-Boc

    CAS:
    Acid-C1-PEG5-Boc is a PEG-based PROTAC linker that can be used in PROTAC synthesis.
    Fórmula:C17H32O9
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:380.43
  • ZINC00881524

    CAS:
    <p>ZINC00881524 (ROCK inhibitor) is an effective and specific ROCK inhibitor.</p>
    Fórmula:C21H20N2O3S
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:380.46
  • VUF 10166

    CAS:
    VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.
    Fórmula:C13H15ClN4
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:262.74
  • (+)-Columbianetin

    CAS:
    (+)-Columbianetin ((S)-Columbianetin) is a new phytoalexin associated with celery (Apium graveolens) resistance to pathogens during storage, it also has
    Fórmula:C14H14O4
    Pureza:99.27% - 99.85%
    Cor e Forma:Solid
    Peso molecular:246.26
  • Tussilagone

    CAS:
    Tussilagone has anti-cancer, anti-oxidant, anti-inflammatory effects and modulates dendritic cells, potentially treating colon cancer and neuro-inflammation.
    Fórmula:C23H34O5
    Pureza:98.17% - 99.63%
    Cor e Forma:Solid
    Peso molecular:390.51
  • Eformoterol Hemifumarate

    CAS:
    Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthma
    Fórmula:C19H24N2O4C4H4O4
    Pureza:99.86% - >99.99%
    Cor e Forma:White Powder
    Peso molecular:402.4
  • RG13022

    CAS:
    RG13022 (Tyrphostin RG13022) is a tyrosine kinase inhibitor; inhibits the autophosphorylation reaction of the EGF receptor (IC50: 4 μM).
    Fórmula:C16H14N2O2
    Pureza:98.38%
    Cor e Forma:Solid
    Peso molecular:266.29
  • 4μ8C

    CAS:
    4μ8C (IRE1 Inhibitor III)(IC50=76 nM) is an effective and specific IRE1 Rnase inhibitor.
    Fórmula:C11H8O4
    Pureza:97.48% - 98.45%
    Cor e Forma:Solid
    Peso molecular:204.18
  • 2'-FUCOSYLLACTOSE

    CAS:
    <p>2'-FUCOSYLLACTOSE (2'-Fucosyl-D-lactose) is a fucose-containing oligosaccharide.</p>
    Fórmula:C18H32O15
    Pureza:98.31% - 99.96%
    Cor e Forma:Solid
    Peso molecular:488.44
  • TPX-0046

    CAS:
    <p>TPX-0046 is a RET inhibitor designed to overcome resistance to Selpercatinib and Pralsetinib.</p>
    Fórmula:C21H21FN6O3
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:424.43
  • 1,2-Dipalmitoyl-sn-glycero-3-phosphoethanolamine

    CAS:
    <p>DPPE, a phospholipid, thickens membranes with Ca2+ and cholesterol.</p>
    Fórmula:C37H74NO8P
    Pureza:99.59% - 99.71%
    Cor e Forma:Solid
    Peso molecular:691.96
  • Bohemine

    CAS:
    Bohemine is a cyclin-dependent kinase inhibitor.
    Fórmula:C18H24N6O
    Pureza:99.09% - 99.53%
    Cor e Forma:Solid
    Peso molecular:340.42
  • 5-Methoxy-DL-tryptophan

    CAS:
    5-Methoxy-DL-tryptophan is a molecule produced by endothelial cells to modulate inflammatory responses and protect against systemic inflammation.
    Fórmula:C12H14N2O3
    Pureza:99.07% - 99.98%
    Cor e Forma:Off-White Powder
    Peso molecular:234.25
  • Scyllo-Inositol

    CAS:
    Scyllo-Inositol (Scyllitol) is one of the inositol stereoisomers, rare in the nature, and expected as a promising disease-modifying therapeutic agent for
    Fórmula:C6H12O6
    Pureza:99.95% - ≥95%
    Cor e Forma:Solid
    Peso molecular:180.16
  • 3-Methyltoxoflavin

    CAS:
    <p>3-Methyltoxoflavin (3-methyl toxoflavin) is an effective inhibitor of protein disulfide isomerase (PDI) and its IC50 value is 170 nM.</p>
    Fórmula:C8H9N5O2
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:207.19
  • PI-103

    CAS:
    <p>PI-103 is a potent, cell-permeable, ATP-competitive inhibitor of PI3K family members (IC50s: 2/3/3/15/30/23 nM for p110α/β/δ/γ, mTOR, and DNA-PK).</p>
    Fórmula:C19H16N4O3
    Pureza:97.79% - 99.3%
    Cor e Forma:Solid
    Peso molecular:348.36
  • Methyl 3-aminopropanoate hydrochloride

    CAS:
    Methyl 3-aminopropanoate hydrochloride (β-Alanine methyl ester hydrochloride) is the ethyl ester of the non-essential amino acid β-alanine.
    Fórmula:C4H10ClNO2
    Pureza:99.4%
    Cor e Forma:White To Off White Powder
    Peso molecular:139.58
  • Etidronic acid

    CAS:
    <p>Etidronic acid (HEDP) is a diphosphonate which affects calcium metabolism. It inhibits ectopic calcification and slows down bone resorption and bone turnover.</p>
    Fórmula:C2H8O7P2
    Pureza:99.93% - ≥95%
    Cor e Forma:Liquid Syrup
    Peso molecular:206.03
  • Edpetiline

    CAS:
    Edpetiline(Sipeimine-3β-D-glucoside), a principal alkaloid from P. eduardi., has significant anti-inflammatory effects.
    Fórmula:C33H53NO8
    Pureza:99.69% - 99.96%
    Cor e Forma:Solid
    Peso molecular:591.78
  • PF-06260933

    CAS:
    <p>PF-06260933 is a highly selective small-molecule MAP4K4 inhibitor with IC50s of 3.7 and 160 nM for kinase and cell, respectively.</p>
    Fórmula:C16H13ClN4
    Pureza:99.63% - 99.97%
    Cor e Forma:Solid
    Peso molecular:296.75
  • Adavivint

    CAS:
    <p>Adavivint (Adavivint (SM04690)) (SM04690) is a Wnt pathway inhibitor.</p>
    Fórmula:C29H24FN7O
    Pureza:98.27% - 98.6%
    Cor e Forma:Solid
    Peso molecular:505.55
  • CEP-28122

    CAS:
    <p>CEP-28122 is a highly potent and selective orally active ALK inhibitor.</p>
    Fórmula:C28H35ClN6O3
    Pureza:99.87% - >99.99%
    Cor e Forma:Solid
    Peso molecular:539.07
  • AX-024 hydrochloride

    CAS:
    AX-024 hydrochloride (AX-024 HCl) is an cytokine release inhibitor which can strongly inhibit the production of IL-6, TNFα, IFN-γ, IL-10 and IL-17A.
    Fórmula:C21H23ClFNO2
    Pureza:99.74%
    Cor e Forma:Solid
    Peso molecular:375.87
  • Edonerpic maleate

    CAS:
    Edonerpic maleate (T-817 maleate) is a neurotrophic agent which can inhibit amyloid-β peptides (Aβ).
    Fórmula:C20H25NO6S
    Pureza:98.24%
    Cor e Forma:Solid
    Peso molecular:407.48
  • Nigakinone

    CAS:
    <p>Nigakinone, isolated from Kumu, is an alkaloid with the pharmacological activity.</p>
    Fórmula:C15H10N2O3
    Pureza:98.66%
    Cor e Forma:Solid
    Peso molecular:266.25
  • RO8994

    CAS:
    RO8994: potent MDM2 spiroindolinone inhibitor, IC50: 20 nM (proliferation), 5 nM (binding).
    Fórmula:C31H31Cl2FN4O4
    Pureza:99.31% - 99.44%
    Cor e Forma:Solid
    Peso molecular:613.51
  • (Z)-LFM-A13

    CAS:
    (Z)-LFM-A13(IC50=2.5 μM), a specific Bruton's tyrosine kinase (BTK), is more than 100-fold specificity than other protein kinases, such as JAK1, JAK2, HCK, EGFR, and IRK.
    Fórmula:C11H8Br2N2O2
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:360
  • (R)-Propranolol hydrochloride

    CAS:
    (R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.
    Fórmula:C16H22ClNO2
    Pureza:98.63% - 99.01%
    Cor e Forma:Solid
    Peso molecular:295.8
  • Seladelpar

    CAS:
    <p>Seladelpar (MBX 8025) has been used in trials studying the treatment of Hyperlipidemia.</p>
    Fórmula:C21H23F3O5S
    Pureza:99.18% - 99.41%
    Cor e Forma:Solid
    Peso molecular:444.46
  • LDN-57444

    CAS:
    LDN-57444 is a reversible, competitive proteasome Uch-L1 inhibitor(IC50=0.88 μM) .
    Fórmula:C17H11Cl3N2O3
    Pureza:97.8% - 99.87%
    Cor e Forma:Solid
    Peso molecular:397.64
  • AL 082D06

    CAS:
    AL 082D06 (D-06), a selective nonsteroidal glucocorticoid receptor (GR) antagonist (Ki: 210 nM), exhibits outstanding selectivity against AR, ER, MR and PR.
    Fórmula:C23H24ClN3O2
    Pureza:99.05% - 99.06%
    Cor e Forma:Solid
    Peso molecular:409.91
  • Merestinib dihydrochloride

    CAS:
    Merestinib dihydrochloride (LY2801653 dihydrochloride) is a kinase inhibitor with antitumor activity that inhibits MET and MKNK1/2.
    Fórmula:C30H24Cl2F2N6O3
    Cor e Forma:Solid
    Peso molecular:625.45
  • AM92016

    CAS:
    AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.
    Fórmula:C26H30Cl2N2O6S
    Cor e Forma:Solid
    Peso molecular:569.49
  • Rhodiosin

    CAS:
    Rhodiosin is a compound with antioxidant activity.
    Fórmula:C27H30O16
    Pureza:98.57% - 99.55%
    Cor e Forma:Solid
    Peso molecular:610.52
  • Notoginsenoside Fe

    CAS:
    Notoginsenoside Fe (Ginsenoside Mb) is a natural compound found in Panax japlcus var.
    Fórmula:C47H80O17
    Pureza:99.43% - 99.93%
    Cor e Forma:Solid
    Peso molecular:917.13
  • Neoeriocitrin

    CAS:
    Neoeriocitrin, from Drynaria Rhizome, boosts MC3T3-E1 growth & bone differentiation; strong AChE inhibitor.
    Fórmula:C27H32O15
    Pureza:99.92% - 99.93%
    Cor e Forma:Solid
    Peso molecular:596.53
  • Jagged-1 (188-204) TFA(219127-21-6 free base)


    Jagged-1 (188-204) TFA, a JAG-1 skin protein fragment, induces epidermal maturation and keratinocyte stratification.
    Fórmula:C95H128F3N25O28S3
    Pureza:99.48%
    Cor e Forma:Solid
    Peso molecular:2221.37
  • Oxysanguinarine

    CAS:
    <p>Oxysanguinarine (Hydroxysanguinarine) possesses antiplatelet aggregation activity, it has potential inhibitory properties against the dengue virus.</p>
    Fórmula:C20H13NO5
    Pureza:99.57%
    Cor e Forma:Solid
    Peso molecular:347.32
  • Fmoc-Gly-Gly-OH

    CAS:
    Fmoc-Gly-Gly-OH is a cleavable ADC linker. Fmoc-Gly-Gly-OH can be used in the synthesis of antibody-drug conjugates (ADCs).
    Fórmula:C19H18N2O5
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:354.36
  • Sesamoside

    CAS:
    Sesamoside has antinociceptive activity.
    Fórmula:C17H24O12
    Pureza:99.47% - 99.87%
    Cor e Forma:Solid
    Peso molecular:420.37
  • Dimboa

    CAS:
    Dimboa (2,4-dihydroxy-7-methoxy-1,4-benzoxazin-3-one) is an antifungal compound used in crops.
    Fórmula:C9H9NO5
    Pureza:96.57% - 98.32%
    Cor e Forma:Solid
    Peso molecular:211.17
  • ML327

    CAS:
    <p>ML327 is a MYC blocker. ML327 can also de-repress E-cadherin transcription and reverse Epithelial-to-Mesenchymal Transition (EMT).</p>
    Fórmula:C19H18N4O4
    Pureza:98.47%
    Cor e Forma:Solid
    Peso molecular:366.37
  • Rubrofusarin gentiobioside

    CAS:
    <p>Rubrofusarin gentiobioside (Rubrofusarin-6-O-beta-D-gentiobioside) decreases the expression of TGF-beta1 and fibronectin and NF-kappaB DNA binding activity.</p>
    Fórmula:C27H32O15
    Pureza:99.91% - 99.93%
    Cor e Forma:Solid
    Peso molecular:596.53
  • ERK5-IN-1

    CAS:
    ERK5-IN-1 is a potent ERK5 inhibitor (IC50: 87 nM). It also inhibits LRRK2[G2019S] (IC50: 26 nM).
    Fórmula:C25H29N7O2
    Pureza:97.70%
    Cor e Forma:Solid
    Peso molecular:459.54