Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.786 produtos)
- Apoptose(6.265 produtos)
- Ciclo celular/Ponto de verificação(4.798 produtos)
- Cromatina/Epigenética(2.442 produtos)
- Sinalização Citoesquelética(1.530 produtos)
- Dano de DNA/Reparo de DNA(2.966 produtos)
- Endocrinologia/Hormónios(3.708 produtos)
- Enzima(3.669 produtos)
- GPCR/Proteína-G(9.018 produtos)
- Imunologia e Inflamação(3.883 produtos)
- Vírus da Influenza(301 produtos)
- Sinalização JAK/STAT(413 produtos)
- Sinalização MAPK(1.248 produtos)
- Transportador de Membranas/Canal Iónico(3.035 produtos)
- Metabolismo(10.214 produtos)
- Microbiologia/Virologia(7.604 produtos)
- Neurociência(10.384 produtos)
- Outros inibidores(36.027 produtos)
- Oxidação-Redução(42 produtos)
- Sinalização PI3K/Akt/mTOR(1.442 produtos)
- Proteases/Proteassoma(1.726 produtos)
- Células - tronco e Derivados(825 produtos)
- Tirosina Quinase/Adaptador(2.040 produtos)
- Ubiquitinação(1.718 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66684 produtos de "Inibidores"
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Carbonic anhydrase inhibitor 8
R-13, a carbonic anhydrase inhibitor, has Ki of 60.7 nM (hCA I), 320.7 nM (hCA II), and 2298 nM (hCA IV).Fórmula:C20H25N3O4SCor e Forma:SolidPeso molecular:403.5Antifungal agent 12
Antifungal agent 12 is a new fluconazole-like compound that exhibits good antifungal effects.Fórmula:C20H16F3N7O2S2Cor e Forma:SolidPeso molecular:507.51(±)-J 113397
CAS:(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM).Fórmula:C24H37N3O2Cor e Forma:SolidPeso molecular:399.57Aurora B inhibitor 1
CAS:Aurora B inhibitor 1 is an Aurora B (Aurora-1) inhibitor (Ki <0.010 uM) with potential anticancer activity for cancer research.Fórmula:C25H26ClF2N7O2Pureza:98.37%Cor e Forma:SolidPeso molecular:529.97Saprisartan potassium
CAS:Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.Fórmula:C25H21BrF3KN4O4SCor e Forma:SolidPeso molecular:649.52KIRA9
KIRA9 inhibits IRE1 with a 4.8 μM IC50, blocking ER-stress-induced mRNA decay and apoptosis by fully binding IRE1's ATP site.Fórmula:C27H27F3N6O3SCor e Forma:SolidPeso molecular:572.6GPR84 antagonist 3
CAS:Potent GPR84 antagonist 3 (compound 42), pIC50 8.28, inhibits GTPγS, with good pharmacokinetics.Fórmula:C29H27N5OCor e Forma:SolidPeso molecular:461.56MtDTBS-IN-1
MtDTBS-IN-1 is a notably potent binder (K_D = 57 nM) and inhibitor (K_i = 5 μM) of MtDTBS.Fórmula:C16H16N4O5Cor e Forma:SolidPeso molecular:344.32LSD1-IN-22
LSD1-IN-22: potent LSD1 inhibitor, K_i 98 nM, curbs cancer cell growth.Fórmula:C9H8BrF2NCor e Forma:SolidPeso molecular:248.07ATM Inhibitor-3
ATM Inhibitor-3 selectively inhibits ATM (IC50: 0.71 nM), targets PI3K kinase family, and is metabolically stable.Fórmula:C25H29FN6O3Cor e Forma:SolidPeso molecular:480.53CEP-7055
CAS:CEP-18770: oral proteasome inhibitor; blocks NF-kappaB; may cause cancer cell apoptosis; less toxic than bortezomib in normal cells.Fórmula:C32H35N3O4Cor e Forma:SolidPeso molecular:525.64Henagliflozin
CAS:Henagliflozin (SHR3824): an oral, selective SGLT2 inhibitor, weak on SGLT1.Fórmula:C22H24ClFO7Cor e Forma:SolidPeso molecular:454.87MI-1851
CAS:MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.Fórmula:C34H53N15O6Cor e Forma:SolidPeso molecular:767.88PIM-1/HDAC-IN-1
PIM-1/HDAC-IN-1 (4d): inhibits PIM-1 (IC50: 343.87nM), HDAC1 (63.65nM), HDAC6 (62.39nM); induces apoptosis in MCF-7 cells.Fórmula:C22H19N3O3Cor e Forma:SolidPeso molecular:373.4Amdinocillin methylacetate
CAS:Amdinocillin methylacetate is a Synthetic penicillin.Fórmula:C18H27N3O4SCor e Forma:SolidPeso molecular:381.49trans-Doxercalciferol
CAS:trans-Doxercalciferol is an isomer of Doxercalciferol. Doxercalciferol is an activator of the Vitamin D receptor and prevents renal disease.Fórmula:C28H44O2Pureza:98%Cor e Forma:SolidPeso molecular:412.65Antitumor agent-42
Antitumor agent-42 inhibits microtubule multimerisation and NO release, exhibiting anti-angiogenic, colony-forming and apoptosis-inducing effects.Fórmula:C24H19BrN2O8SCor e Forma:SolidPeso molecular:575.39Lafadofensine (D-(-)-Mandelic acid)
Lafadofensine D-(-)-Mandelic acid is a monoamines reuptake inhibitor with adequate effects when administered short-term.Fórmula:C32H32F2N2O6Cor e Forma:SolidPeso molecular:578.6Anti-inflammatory agent 23
Anti-inflammatory agent 23 blocks LPS-induced NO (IC50: 0.449 μM) and binds p65 well.Fórmula:C34H49NO6Cor e Forma:SolidPeso molecular:567.76Metocurine chloride
CAS:Metocurine: a muscle relaxant, not for kidney failure patients as it's kidney-excreted.Fórmula:C40H48Cl2N2O6Cor e Forma:SolidPeso molecular:723.72Anti-MRSA agent 2
CAS:Anti-MRSA agent 2 inhibits MRSA at 0.098 μg/ml, with low toxicity and disrupts bacterial membranes and DNA.Fórmula:C18H10Br2N2OCor e Forma:SolidPeso molecular:430.09IRAK4-IN-12
IRAK4-IN-12 (compound 37) is a potent inhibitor of IRAK4 (IC50: 0.015 μM) with cellular pIRAK4 potency (IC50: 0.5 μM).Fórmula:C24H31FN8OCor e Forma:SolidPeso molecular:466.55Mopivabil
Mopivabil is the angiotensin II receptor antagonist[1].Fórmula:C14H20O3Cor e Forma:SolidPeso molecular:236.31Norbinaltorphimine dihydrochloride
CAS:Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.Fórmula:C40H45Cl2N3O6Pureza:98.17% - 99.88%Cor e Forma:SolidPeso molecular:734.71Ref: TM-T12241
1mg38,00€5mg85,00€10mg120,00€25mg235,00€50mg409,00€100mg652,00€200mg908,00€1mL*10mM (DMSO)124,00€AChE/BChE-IN-1
<p>AChE/BChE-IN-1: dual AChE/BChE inhibitor, IC50 of 1.06 nM/7.3 nM, crosses blood-brain barrier, with antioxidant properties for Alzheimer's research.</p>Fórmula:C32H35ClN6O3Cor e Forma:SolidPeso molecular:587.11DS01080522
DS01080522: PRKACA inhibitor, IC50: kinase 0.8 nM, CREB 66 nM; potential for cancer research.Fórmula:C23H20Cl2N4O3Cor e Forma:SolidPeso molecular:471.34CXCR2 antagonist 6
CXCR2 antagonist 6: strong CXCR2 affinity (IC50=0.044 μM), hinders calcium mobilization (IC50=0.66 μM).Fórmula:C17H16F2N4OSCor e Forma:SolidPeso molecular:362.4Steroid sulfatase/17β-HSD1-IN-4
Steroid sulfatase/17β-HSD1-IN-4 (compound 37) is a potent dual inhibitor of steroid sulfatase ( STS ) and 17β-hydroxysteroid dehydrogenase type 1 ( 17β HSD1 ).Fórmula:C18H17N3O4S2Cor e Forma:SolidPeso molecular:403.48CHK-IN-1
CAS:CHK-IN-1 is a dual inhibitor of CHK1 and CHK2 with antiproliferative activity.Fórmula:C18H19ClFN5OSPureza:>99.99%Cor e Forma:SolidPeso molecular:407.89Isoleucyl tRNA synthetase-IN-2
CAS:Isoleucyl tRNA synthetase-IN-2 is a selective and potent inhibitor (Ki: 114 nM) that targets isoleucyl tRNA synthetase (IleRS).Fórmula:C22H33N5O8SCor e Forma:SolidPeso molecular:527.59Tribenuron
CAS:<p>Tribenuron, a slow acting sulfonylurea herbicide, controls broadleaf weed.</p>Fórmula:C14H15N5O6SCor e Forma:SolidPeso molecular:381.36BNTX maleate
CAS:δ1 opioid receptor antagonistFórmula:C31H31NO8Pureza:98%Cor e Forma:SolidPeso molecular:545.58BMS 310705
CAS:BMS 310705, an Epothilone B analog, targets ovarian/renal/bladder/lung cancer, inducing apoptosis via mitochondria.Fórmula:C27H42N2O6SCor e Forma:SolidPeso molecular:522.70AKR1C3-IN-7
AKR1C3-IN-7 (Compound 13) is an effective and selective AKR1C3 inhibitor (IC50=0.19 μM). AKR1C3-IN-7 has antitumor activity.Fórmula:C24H20N2O4Cor e Forma:SolidPeso molecular:400.43LY3020371 hydrochloride
CAS:LY3020371 HCl: potent mGlu2/3 antagonist, antidepressant-like; Ki: 5.3/2.5 nM, IC50: 16.2 nM for cAMP inhibition.Fórmula:C15H16ClF2NO5SCor e Forma:SolidPeso molecular:395.81Nrf2/HO-1 activator 2
Compound 13m, a difluoro derivative, activates Nrf2/HO-1, showing neuroprotective and antioxidant effects, useful in PD research.Fórmula:C20H16F2O5Cor e Forma:SolidPeso molecular:374.33Freselestat quarterhydrate
ONO-6818 quarterhydrate: oral neutrophil elastase inhibitor, Ki 12.2 nM; >100x less effective on other proteases; strong anti-inflammatory.Fórmula:C23H30N6O5Cor e Forma:SolidPeso molecular:457.03HER2-IN-6
CAS:HER2-IN-6, a potent HER2 inhibitor, may target wild/mutant EGFR and HER2-mediated tumors. (Patent WO2021164697A1, compound 11)Fórmula:C26H32N8O3Cor e Forma:SolidPeso molecular:504.58TMC353121
CAS:TMC353121 is an effective inhibitor of respiratory syncytial virus fusion (pEC50: 9.9).Fórmula:C32H42N6O3Pureza:≥98%Cor e Forma:SolidPeso molecular:558.71MRS2179 tetrasodium hydrate
MRS2179 blocks turkey P2Y1 receptor (Kb 102 nM, pA2 6.99), affects platelet aggregation, and has varying IC50s on P2 receptors.Fórmula:C11H15N5Na4O10P2Cor e Forma:SolidPeso molecular:576.21Fabimycin
CAS:Fabimycin, a FabI inhibitor, combats drug-resistant gram-negative bacterial infections effectively.Fórmula:C23H25ClN4O3Cor e Forma:SolidPeso molecular:440.92SID 26681509 quarterhydrate
SID 26681509 is a selective inhibitor of cathepsin L (IC50: 56 nM) and blocks Plasmodium falciparum (IC50: 15.4 μM) and Leishmania major (IC50: 12.5 μM).Fórmula:C27H35N5O6SCor e Forma:SolidPeso molecular:544.16Diospyrin
CAS:Diospyrin is a plant product that has significant inhibitory effect on the growth of Leishmania donovani promastigotes.Fórmula:C22H14O6Cor e Forma:SolidPeso molecular:374.34ABL-001-Amide-PEG3-acid
ABL-001-Amide-PEG3-acid, an analogue to ABL-001, primarily serves as a labeled chemical or fluorescent probe.Fórmula:C29H33ClF2N6O9Pureza:98%Cor e Forma:SolidPeso molecular:683.06IMR687
CAS:IMR687: a PDE9 inhibitor that could improve memory in Alzheimer's by slowing cGMP hydrolysis.Fórmula:C21H26N6O2Pureza:98%Cor e Forma:SolidPeso molecular:394.47ZBH-1205
CAS:ZBH-1205, a camptothecin derivative, shows strong antitumor effects via apoptosis, outperforming cpt-11 and sn38 in topoisomerase-1 inhibition.Fórmula:C29H31N3O8Cor e Forma:SolidPeso molecular:549.57ACSS2-IN-1
CAS:ACSS2-IN-1, a potent ACSS2 inhibitor, has IC50 0.01-<1 nM; useful in cancer research.Fórmula:C27H25ClN6O2Cor e Forma:SolidPeso molecular:500.98PD-1/PD-L1-IN-17
<p>PD-1/PD-L1-IN-17 (Compound P20) is a potent PD-1/PD-L1 inhibitor (IC50: 26.8 nM).</p>Fórmula:C23H20ClN3O4Cor e Forma:SolidPeso molecular:437.88Mevidalen HBA
CAS:Mevidalen (LY3154207), a potent D1 positive allosteric modulator, is in clinical trials for Lewy body dementia.Fórmula:C31H35Cl2NO6Cor e Forma:SolidPeso molecular:588.52BGC-638
CAS:BGC-638, an analogue of BGC-945, is a thymidylate synthase inhibitor specifically transported into α-folate receptor (α-FR)–overexpressing tumors.Fórmula:C32H33N5O9Cor e Forma:SolidPeso molecular:631.63RSV-IN-5
CAS:RSV-IN-5: Dual inhibitor for RSV fusion proteins, effective on wild-type A2 and D486N mutant with EC50s of 2.0 nM & 8.1 nM. Potent anti-RSV.Fórmula:C28H37N7O2Cor e Forma:SolidPeso molecular:503.64BTK-IN-6
BTK-IN-6, a potent BTK inhibitor, may treat immune, cardiac, cancer, viral, inflammatory, metabolic, and neurological disorders.Fórmula:C23H22FN5O3Cor e Forma:SolidPeso molecular:435.45BACE1-IN-8
BACE1-IN-8 is a potent inhibitor of BACE1 (β-site APP lyase 1) (IC50: 3.9 μM).Fórmula:C29H45N5O7Cor e Forma:SolidPeso molecular:575.7BRD4 D1-IN-2
BRD4 D1-IN-2 (compound 26), a BRD4 D1 inhibitor, IC50 <0.092 μM, 15 nM affinity, >500x selectivity over BRD2 D1/BRD4 D2.Fórmula:C33H39F3N6OCor e Forma:SolidPeso molecular:592.7TAK-915
CAS:TAK-915: potent, brain-ready PDE2A inhibitor, 0.61 nM IC50, 4100x selectivity over PDE1A.Fórmula:C19H18F4N4O5Pureza:98%Cor e Forma:SolidPeso molecular:458.36NLRP3-IN-4
NLRP3-IN-4 is an effective, oral NLRP3 inflammasome inhibitor with potent anti-inflammatory effects on colitis.Fórmula:C22H22N2O5Cor e Forma:SolidPeso molecular:394.42Nevirapine dimer
CAS:Nevirapine dimer is a non-nucleoside reverse transcriptase inhibitor (NNRTI).Fórmula:C30H26N8O2Cor e Forma:SolidPeso molecular:530.58Valopicitabine
CAS:<p>Valopicitabine is an effective prodrug of the effective anti-HCV drug 2'-C-methylcytidine and can be used as a promising antiviral drug for the study of chronic</p>Fórmula:C15H24N4O6Pureza:98%Cor e Forma:SolidPeso molecular:356.37Org-31710
CAS:Org-31710 is a progesterone receptor antagonist potentially for contraception.Fórmula:C30H39NO2Pureza:98%Cor e Forma:SolidPeso molecular:445.64ent-8-iso-15(S)-Prostaglandin F2α
CAS:Isoprostanes are produced by the non-enzymatic, free radical peroxidation of phospholipid-esterified arachidonic acid.Fórmula:C20H34O5Cor e Forma:SolidPeso molecular:354.48Moflomycin
CAS:Moflomycin is an anthracycline derivative. It exhibits a higher antileukemic activity compared to other anthracyclines.Fórmula:C25H25IO10Pureza:98%Cor e Forma:SolidPeso molecular:612.36IRAK4-IN-11
IRAK4-IN-11 (compound 6) is a potent inhibitor of IRAK4 with an IC 50 of 0.008 μM. IRAK4-IN-11 exhibits cell pIRAK4 potencies with an IC 50 of 0.19 μM [1].Fórmula:C16H19N7OCor e Forma:SolidPeso molecular:325.37MAO-B-IN-7
MAO-B-IN-7 inhibits MAO-B/AChE, crossing the blood-brain barrier; IC50: 41/87 nM (h/eel AChE), 0.3 μM (MAO-B). Reduces oxidative stress and neuroinflammation.Fórmula:C25H31NO4Cor e Forma:SolidPeso molecular:409.52ZK824859 hydrochloride (2271122-53-1 free base)
ZK824859 hydrochloride: oral, selective uPA inhibitor, IC50s: 79 nM (uPA), 1580 nM (tPA), 1330 nM (plasmin).Fórmula:C23H23ClF2N2O4Pureza:98%Cor e Forma:SolidPeso molecular:464.89PI3kδ inhibitor 1
CAS:<p>PI3kδ inhibitor 1 is a selective inhibitor of PI3Kδ (IC50 of 3.8 nM).</p>Fórmula:C28H33FN6O2Pureza:98%Cor e Forma:SolidPeso molecular:504.60MEIS-IN-1
CAS:<p>MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.</p>Fórmula:C24H21F3N2O4Cor e Forma:SolidPeso molecular:458.43UK-370106
CAS:UK-370106 is a potent and highly selective inhibitor of MMP-3 with IC50 of 23 nM and MMP-12 with IC50 of 42 nM, and potently inhibits cleavage of [3H]-Fórmula:C35H44N2O5Pureza:98%Cor e Forma:SolidPeso molecular:572.73Nikkomycin Z
CAS:Nikkomycin Z (Nikkomycin Z from Streptomyces tendae) is a competitive chitin synthase inhibitor.It inhibitor of the growth of filamentous fungi, insects,Fórmula:C20H25N5O10Pureza:98%Cor e Forma:SolidPeso molecular:495.44RET-IN-10
CAS:RET-IN-10: Potent RET inhibitor, may treat congenital megacolon and tumors (Patent WO2021135938A1, compound 18).Fórmula:C29H28N8OSCor e Forma:SolidPeso molecular:536.65HIF-1α-IN-5
HIF-1α-IN-5 is an inhibitor of HIF-1α with an IC 50 value of 24 nM in HEK293T cells that also inhibits the activity of MAO-A.Fórmula:C16H15N3O2Cor e Forma:SolidPeso molecular:281.31Anticancer agent 143
CAS:Anticancer Agent 143 (Compound 369), a potent dual inhibitor targeting PTPN2 and PTP1B, exhibits IC50 values below 2.5 nM.Fórmula:C19H15BrF2N3O6PS2Pureza:98%Cor e Forma:SolidPeso molecular:594.34Tandutinib (MLN518) HCl
Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.Fórmula:C31H43ClN6O4Pureza:98%Cor e Forma:SolidPeso molecular:599.16CI-1029
CAS:CI-1029: HIV protease inhibitor, combats mutant strains, high efficacy, good bioavailability in animals.Fórmula:C28H37NO4SCor e Forma:SolidPeso molecular:483.66Bulgecin A
CAS:Bulgecin A is an inhibitor of binuclear metallo-beta-lactamases and Lytic transglycosolase.Fórmula:C16H29N3O14S2Cor e Forma:SolidPeso molecular:551.54DNA Gyrase-IN-1
DNA Gyrase-IN-1: potent, selective promoter inhibitor. IC50: 2.6 μM, inhibits Mtb, MIC: 0.49 μM. Useful for tuberculosis research.Fórmula:C24H24FN7O6Cor e Forma:SolidPeso molecular:525.49TLR4/NF-κB/MAPK-IN-1
CAS:TLR4/NF-κB/MAPK-IN-1 is a novel antineuroinflammatory agent that functions by inhibiting the TLR4/NF-κB/MAPK pathways.Fórmula:C19H25BrO6Cor e Forma:SolidPeso molecular:429.3Nolpitantium besilate
CAS:Nolpitantium besilate is a neurokinin-1 receptor antagonist.Fórmula:C43H50Cl2N2O5SCor e Forma:SolidPeso molecular:777.849(S)-HETE
CAS:9(S)-HETE is an enantiomer of (±)9-HETE, not an enzymatic product, and doesn't promote cell adhesion like 12(S)-HETE. Identified by chiral HPLC.Fórmula:C20H32O3Cor e Forma:SolidPeso molecular:320.47CDK4/6-IN-10
CDK4/6-IN-10: Oral CDK4 (IC50: 22 nM) & CDK6 (IC50: 10 nM) inhibitor with anti-cancer potential for MM research.Cor e Forma:SolidKolavenic acid analog
CAS:KAA, an anticancer compound, inhibits centrosome clustering and targets HSET+ yeast and cancer cells.Fórmula:C25H38O4Cor e Forma:SolidPeso molecular:402.57LAF-153
CAS:LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.Fórmula:C18H32N2O7Cor e Forma:SolidPeso molecular:388.46BI-1388
CAS:BI-1388 is a potent HCV NS3 protease inhibitor; halts replication across genotypes, including D168V/R155K mutants.Fórmula:C41H53N7O9SCor e Forma:SolidPeso molecular:819.97STA 2
CAS:STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.Fórmula:C21H34O3SCor e Forma:SolidPeso molecular:366.56KRAS G12C inhibitor 33
CAS:KRAS G12C inhibitor 33 is a KRAS G12C inhibitor that can be used to study cancer.Fórmula:C30H33N7O3Cor e Forma:SolidPeso molecular:539.63Motuporin
CAS:Motuporin is an inhibitor of type-1 and type-2A protein phosphatase catalytic subunits (PP-1c and PP-2Ac).Fórmula:C40H57N5O10Cor e Forma:SolidPeso molecular:767.91Elocalcitol
CAS:Elocalcitol is a calcitriol analog for inhibition of prostate cell growth.Fórmula:C29H43FO2Cor e Forma:SolidPeso molecular:442.65Topo I-IN-1
Topo I-IN-1 (14d) is a powerful Topo I inhibitor with antitumor effects and DNA intercalation, inducing apoptosis.Fórmula:C20H14BrN3O2Cor e Forma:SolidPeso molecular:408.25Gabaculine HCl
CAS:Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.Fórmula:C7H10ClNO2Cor e Forma:SolidPeso molecular:175.61PDHK-IN-5
PDHK-IN-5, potent PDHK2 (0.006 μM IC50) & PDHK4 (0.0329 μM IC50) inhibitor, may be explored for cancer and diabetes treatment.Fórmula:C30H31N5O2Cor e Forma:SolidPeso molecular:493.6DS34942424
DS34942424 is an orally potent analgesic which did not exhibit mu opioid receptor agonist activity.Fórmula:C15H17FN2OCor e Forma:SolidPeso molecular:260.31SCH-1473759
CAS:SCH-1473759 is an inhibitor of the aurora (IC50s: 4 and 13 nM for Aurora A and B, respectively).Fórmula:C20H26N8OSPureza:98%Cor e Forma:SolidPeso molecular:426.54FXIa-IN-8
FXIa-IN-8: potent FXIa blocker (IC50: 14.2 nM), anti-thrombotic, low bleeding/toxicity risk.Cor e Forma:SolidDot1L-IN-1
CAS:The Ki value of DOT1L-in-1 is 2pm.It is a highly effective, selective and novel Dot1L inhibitor.Fórmula:C32H36ClN9O2SPureza:98%Cor e Forma:SolidPeso molecular:646.21Org-6906
CAS:DCB-3503, a tylophorine analog, may treat cancer and suppress immunity by blocking protein synthesis and modulating HSC70's ATPase activity.Fórmula:C13H16ClNPureza:98%Cor e Forma:SolidPeso molecular:221.73L 731735
CAS:L 731735 is a farnesyltransferase inhibitor.Fórmula:C19H40N4O4SPureza:98%Cor e Forma:SolidPeso molecular:420.61Pegcantratinib
CAS:Pegcantratinib is a tropomyosin receptor kinase inhibitor for treatment for inherited CYLD defective skin tumours.Fórmula:C32H28N4O7Cor e Forma:SolidPeso molecular:580.59Onfasprodil
CAS:Onfasprodil, NR2B inhibitor & GABA regulator, potential for Alzheimer's research. (Patent CN111481543A)Fórmula:C20H23FN2O3Cor e Forma:SolidPeso molecular:358.41Plumbemycin A
CAS:Plumbemycin A is isolated from Streptomyces plumbeus; an L-threonine antagonist.Fórmula:C12H20N3O9PCor e Forma:SolidPeso molecular:381.28L 702007
CAS:L 702007 is an inhibitor of HIV-1 reverse transcriptase.Fórmula:C18H25N3O2Pureza:98%Cor e Forma:SolidPeso molecular:315.41Furametpyr
CAS:Furametpyr is a kind of low toxicity pesticides used to control plant diseases caused by various pathogenic microorganisms.Fórmula:C17H20ClN3O2Pureza:98%Cor e Forma:SolidPeso molecular:333.81
