
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.861 produtos)
- Apoptose(6.355 produtos)
- Ciclo celular/Ponto de verificação(3.862 produtos)
- Cromatina/Epigenética(2.667 produtos)
- Sinalização Citoesquelética(1.578 produtos)
- Dano de DNA/Reparo de DNA(1.913 produtos)
- Endocrinologia/Hormónios(3.773 produtos)
- Enzima(3.748 produtos)
- GPCR/Proteína-G(9.184 produtos)
- Imunologia e Inflamação(3.663 produtos)
- Vírus da Influenza(297 produtos)
- Sinalização JAK/STAT(422 produtos)
- Sinalização MAPK(1.266 produtos)
- Transportador de Membranas/Canal Iónico(3.141 produtos)
- Metabolismo(9.717 produtos)
- Microbiologia/Virologia(7.173 produtos)
- Neurociência(10.597 produtos)
- Outros inibidores(36.280 produtos)
- Oxidação-Redução(44 produtos)
- Sinalização PI3K/Akt/mTOR(1.431 produtos)
- Proteases/Proteassoma(1.654 produtos)
- Células - tronco e Derivados(735 produtos)
- Tirosina Quinase/Adaptador(2.012 produtos)
- Ubiquitinação(1.772 produtos)
Exibir 16 mais subcategorias
Foram encontrados 65419 produtos para "Inibidores".
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Ciproquazone
CAS:Ciproquazone has analgesic activity and is used to treat spondylitis.Fórmula:C19H18N2O2Pureza:99.66%Cor e Forma:SolidPeso molecular:306.36Ostarine
CAS:Ostarine (MK-2866) is a non-steroidal SARM mimicking testosterone to boost muscle growth, libido, fertility, and may help prevent muscle wasting in cancer.Fórmula:C19H14F3N3O3Pureza:99.69% - 99.90%Cor e Forma:SolidPeso molecular:389.33Tiragolumab
CAS:Tiragolumab, a monoclonal antibody, targets TIGIT and is used with Atezolizumab to treat solid tumors like lung cancer.Pureza:SDS-PAGE:95.3%;SEC-HPLC:98.8%Cor e Forma:LiquidPeso molecular:148.3 kDaD-Glutamic acid
CAS:D-Glutamic acid ((R)-Glutamic acid), the enantiomer of L-glutamic acid, is widely used in medicine and food.Fórmula:C5H9NO4Pureza:99.24% - 99.33%Cor e Forma:SolidPeso molecular:147.13Captopril
CAS:Captopril (SA333) is a potent and specific inhibitor of peptidyl-dipeptidase A.Fórmula:C9H15NO3SPureza:98.34% - 99.85%Cor e Forma:SolidPeso molecular:217.29Broflanilide
CAS:Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.Fórmula:C25H14BrF11N2O2Pureza:99.82%Cor e Forma:SolidPeso molecular:663.29Ref: TM-T10618
1mg50,00€2mg71,00€5mg105,00€1mL*10mM (DMSO)124,00€10mg170,00€25mg339,00€50mg557,00€100mg792,00€2-Methylbenzene-1-sulfonamide
CAS:2-Methylbenzene-1-sulfonamide is used for saccharin, pharmaceutical intermediates, etc.Fórmula:C7H9NO2SPureza:99.25% - 99.43%Cor e Forma:SolidPeso molecular:171.22GSK-626616
CAS:GSK-626616: strong, oral DYRK3 inhibitor (IC50: 0.7 nM), affects DYRK family, may treat anemia.Fórmula:C18H10Cl2N4OSPureza:98.27%Cor e Forma:SolidPeso molecular:401.27Procodazole
CAS:Procodazole (2-Benzimidazolepropionic acid) is a non-specific active immunoprotective agent against viral and bacterial infections.Fórmula:C10H10N2O2Pureza:98% - 99.35%Cor e Forma:SolidPeso molecular:190.2L-Tyrosine
CAS:L-Tyrosine ((S)-Tyrosine) is a naturally occurring tyrosine and is synthesized in vivo from L-phenylalanine, considered a non-essential amino acid.Fórmula:C9H11NO3Pureza:99.82%Cor e Forma:SolidPeso molecular:181.19VU0134992 hydrochloride
CAS:VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).Fórmula:C20H32BrClN2O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:447.84FM4-64
CAS:FM4-64 (SynaptoRedTM C2) is a stylenoid dye. FM4-64 can be used to study endocytosis exocytosis and vesicle trafficking. High-Quality, Low-Cost!Fórmula:C30H45Br2N3Pureza:99.41% - 99.99%Cor e Forma:Green SolidPeso molecular:607.51Zileuton
CAS:Zileuton (A 64077) inhibits 5-lipoxygenase, reduces leukotrienes, aids bronchodilation, lessens mucus/edema, and helps manage asthma symptoms.Fórmula:C11H12N2O2SPureza:98.72% - 99.86%Cor e Forma:White SolidPeso molecular:236.29Eleclazine hydrochloride
CAS:Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).Fórmula:C21H17ClF3N3O3Pureza:99.86%Cor e Forma:SolidPeso molecular:451.83Ref: TM-T15207
1mg58,00€5mg110,00€1mL*10mM (DMSO)122,00€10mg166,00€25mg268,00€50mg403,00€100mg532,00€200mg705,00€Novobiocin Sodium
CAS:Novobiocin Sodium (Albamycinsodium) binds to DNA gyrase and blocks adenosine triphosphatase (ATPase) activity. Novobiocin sodium is an antibiotic compound.Fórmula:C31H35N2NaO11Pureza:99% - 99.51%Cor e Forma:SolidPeso molecular:634.61JW 642
CAS:JW 642 inhibits MAGL in mouse, rat, human brains (IC50: 7.6, 14, 3.7 nM).Fórmula:C21H20F6N2O3Pureza:99.28%Cor e Forma:SolidPeso molecular:462.39Dofequidar fumarate
CAS:Dofequidar fumarate (MS-209)(MS-209 fumarate), a quinoline-based compound administered orally, is known for counteracting multidrug resistance (MDR) through theFórmula:C34H35N3O7Pureza:99.93%Cor e Forma:SolidPeso molecular:597.66Ref: TM-T11071
1mg37,00€2mg52,00€5mg80,00€1mL*10mM (DMSO)90,00€10mg118,00€25mg233,00€50mg447,00€100mg650,00€500mg1.369,00€Tetrabenazine Metabolite
CAS:Tetrabenazine Metabolite ((-)-β-HTBZ), a vesicles monoamine transporter 2 (VMAT2) inhibitor, is an active metabolite of Tetrabenazine.Fórmula:C19H29NO3Pureza:97.09%Cor e Forma:SolidPeso molecular:319.44Ref: TM-T13133
1mg73,00€1mL*10mM (DMSO)146,00€5mg149,00€10mg212,00€25mg319,00€50mg447,00€100mg610,00€200mg822,00€Bromhexine hydrochloride
CAS:Bromhexine hydrochloride (Bisolvon) is a mucolytic agent used in the treatment of respiratory disorders associated with viscid or excessive mucus.Fórmula:C14H21Br2ClN2Pureza:99.98%Cor e Forma:SolidPeso molecular:412.59Tylosin tartrate
CAS:Tylosin tartrate, a macrolide antibiotic, is approved for the control of mycoplasmosis in poultry.Fórmula:C46H77NO17·C4H6O6Pureza:91.82% - 99.36%Cor e Forma:White SolidPeso molecular:1066.19Tobramycin
CAS:Tobramycin (NSC-180514) is an aminoglycoside, broad-spectrum antibiotic produced by Streptomyces tenebrarius.Fórmula:C18H37N5O9Pureza:99.21% - 99.87%Cor e Forma:SolidPeso molecular:467.51DTNB
CAS:DTNB, or Ellman's Reagent, quantifies thiol groups and measures low-mass thiols like glutathione in pure and biological samples.Fórmula:C14H8N2O8S2Pureza:97.11% - 99.51%Cor e Forma:SolidPeso molecular:396.35Adenosine 5'-monophosphate monohydrate
CAS:Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.Fórmula:C10H14N5O7P·H2OPureza:97.68% - 98.49%Cor e Forma:White SolidPeso molecular:365.24Clomiphene citrate
CAS:Clomiphene citrate (NSC 35770) is a selective estrogen receptor modulator.Fórmula:C32H36ClNO8Pureza:98.67% - >99.99%Cor e Forma:SolidPeso molecular:598.1Omeprazole metabolite Omeprazole sulfone
CAS:Omeprazole metabolite Omeprazole sulfone can inhibit proton pump.Fórmula:C17H19N3O4SPureza:99.87%Cor e Forma:SolidPeso molecular:361.42Ref: TM-T12309
1mg47,00€2mg62,00€5mg92,00€1mL*10mM (DMSO)101,00€10mg145,00€25mg281,00€50mg423,00€100mg608,00€500mg1.251,00€Linezolid
CAS:Linezolid (PNU-100766), the first of the oxazolidinone class, is a synthetic antibiotic used for the therapy of infections resulted from multi-resistantFórmula:C16H20FN3O4Pureza:99.73% - 99.99%Cor e Forma:SolidPeso molecular:337.35Ref: TM-T0391
1mL*10mM (DMSO)34,00€10mg48,00€25mg80,00€50mg90,00€100mg138,00€200mg172,00€500mg268,00€Pentetic Acid
CAS:Pentetic Acid (Detarex) is an edetate and a chelating agent used in preparing radiopharmaceuticals.Fórmula:C14H23N3O10Pureza:≥95%Cor e Forma:White Solid PowderPeso molecular:393.35GNF179
CAS:GNF179 is an optimized 8,8-dimethyl IP analog.Fórmula:C22H23ClFN5OPureza:97.80%Cor e Forma:White SolidPeso molecular:427.9Ref: TM-T15409
1mg109,00€2mg158,00€5mg260,00€1mL*10mM (DMSO)286,00€10mg430,00€25mg710,00€50mg973,00€100mg1.333,00€HLY78
CAS:HLY78, a Wnt/β-catenin activator, enhances Axin-LRP6 binding by targeting Axin's DIX domain.Fórmula:C17H17NO2Pureza:99.54%Cor e Forma:White SolidPeso molecular:267.32Tetraethylenepentamine Pentahydrochloride
CAS:Tetraethylenepentamine Pentahydrochloride is a high affinity copper and zinc chelator.Fórmula:C8H23N5·5HClPureza:≥95%Cor e Forma:SolidPeso molecular:371.61Oxybuprocaine hydrochloride
CAS:Oxybuprocaine hydrochloride (Oxybuprocaine HCl), a local anesthetic, is used especially in otolaryngology and ophthalmology.Fórmula:C17H29ClN2O3Pureza:>99.99%Cor e Forma:SolidPeso molecular:344.88Pyridoxine
CAS:Pyridoxine, or Vitamin B6, is a 4-methanol form, transformed to pyridoxal 5-phosphate in the body. Using both terms interchangeably is incorrect.Fórmula:C8H11NO3Pureza:97.58% - 99.83%Cor e Forma:SolidPeso molecular:169.18Niclosamide olamine
CAS:Niclosamide olamine (Niclosamide Ethanolamine salt) is an Repellent, Insect Attractant and Chemosterilant.Fórmula:C15H15Cl2N3O5Pureza:99.89%Cor e Forma:SolidPeso molecular:388.20AZD5904
CAS:AZD5904 is a potent and irreversible inhibitor of human Myeloperoxidase (MPO, IC50: 140 nM) which has similar potency in mouse and rat.Fórmula:C10H12N4O2SPureza:99.89%Cor e Forma:SolidPeso molecular:252.29DUPA(OtBu)-OH
CAS:DUPA(OtBu)-OH, a DUPA precursor, targets PSMA with high affinity (Ki=8nM) to deliver Docetaxel for prostate cancer therapy.Fórmula:C23H40N2O9Pureza:97.29%Cor e Forma:SolidPeso molecular:488.57Ref: TM-T11122
2mg34,00€5mg50,00€1mL*10mM (DMSO)54,00€10mg82,00€25mg123,00€50mg170,00€100mg235,00€200mg334,00€DMT1 blocker 2
CAS:Compound 12f, a DMT1 blocker, inhibits DMT1 with a 0.83 IC50, potentially blocking intestinal iron absorption.Fórmula:C16H13N3OPureza:99.68%Cor e Forma:SolidPeso molecular:263.29Ref: TM-T11064
1mg71,00€5mg155,00€1mL*10mM (DMSO)203,00€10mg222,00€25mg404,00€50mg607,00€100mg888,00€Diaveridine
CAS:Diaveridine (AI3-23935) (DVD) is a popular antibacterial synergist that is widely used in combination with sulfonamide.Fórmula:C13H16N4O2Pureza:99.10%Cor e Forma:SolidPeso molecular:260.29Levosulpiride
CAS:Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Fórmula:C15H23N3O4SPureza:98.20% - 99.88%Cor e Forma:White SolidPeso molecular:341.43Parsatuzumab
CAS:Parsatuzumab (RG 7414), a monoclonal antibody targeting EGFL7, an immunomodulator.Parsatuzumab inhibits the interaction of EGFL7 with endothelial cells.Pureza:> 95% - > 95%Cor e Forma:Transparent LiquidPeso molecular:148.22 kDaT3Inh-1
CAS:T3Inh-1 is a potent and selective ppGalNAc-T3 inhibitor with IC50 of 7 µM.Cost-effective and quality-assured.Fórmula:C27H20N6O3Pureza:97.21%Cor e Forma:SolidPeso molecular:476.49Ref: TM-T9720
1mg96,00€5mg205,00€1mL*10mM (DMSO)245,00€10mg344,00€25mg655,00€50mg973,00€100mg1.333,00€Prucalopride
CAS:Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.Fórmula:C18H26ClN3O3Pureza:99.99% - >99.99%Cor e Forma:White SolidPeso molecular:367.87Dehydroacetic acid
CAS:Dehydroacetic acid (Methylacetopyronone), a pyrone derivative, is served frequently as a fungicide and bactericide.Fórmula:C8H8O4Pureza:99.51%Cor e Forma:Yellow SolidPeso molecular:168.15Vitamin B6
CAS:Vitamin B6 aids metabolism, especially for amino acids, and helps prevent pregnancy-induced and radiation sickness vomiting.Fórmula:C8H12NO6PPureza:97.81%Cor e Forma:SolidPeso molecular:249.15PF429242 dihydrochloride
CAS:PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).Fórmula:C25H37Cl2N3O2Pureza:99.68%Cor e Forma:White ViscousPeso molecular:482.49Aminophylline
CAS:Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.Fórmula:C7H8O2·C2H8N2Pureza:99.31%Cor e Forma:SolidPeso molecular:420.43BI-1935
CAS:BI-1935 is an inhibitor of soluble epoxide hydrolase (sEH). For diseases related to cardiovascular disease.Fórmula:C24H21F3N6O3Pureza:97.55%Cor e Forma:SolidPeso molecular:498.46Ref: TM-T14557
1mg46,00€5mg94,00€1mL*10mM (DMSO)103,00€10mg148,00€25mg259,00€50mg360,00€100mg465,00€200mg625,00€GRP78-IN-3
CAS:GRP78-IN-3: Potent Hsp70 blocker, selective Grp78 (HSPA5) inhib., IC50 0.59 μM, 7x more vs HspA9, 20x vs HspA2.Fórmula:C17H18N4O2SPureza:99.49%Cor e Forma:SolidPeso molecular:342.42Ethylparaben
CAS:Ethylparaben (Ethyl parahydroxybenzoate) is a Standardized Chemical Allergen.Fórmula:C9H10O3Pureza:99.34%Cor e Forma:White SolidPeso molecular:166.17β-Elemene
CAS:β-Elemene (Levo-β-elemene) is a natural product isolated from Curcuma wenyujin, with an antitumor activity and induce cell apoptosis.Fórmula:C15H24Pureza:99.16% - 99.35%Cor e Forma:Transparent LiquidPeso molecular:204.35Ref: TM-T13476
1mL*10mM (DMSO)33,00€10mg46,00€25mg73,00€50mg104,00€100mg120,00€200mg173,00€500mg294,00€Terlipressin Acetate
CAS:Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).Fórmula:C56H82N16O19S2Pureza:98.50% - 99.69%Cor e Forma:SolidPeso molecular:1347.5
