
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.805 produtos)
- Apoptose(6.288 produtos)
- Ciclo celular/Ponto de verificação(4.815 produtos)
- Cromatina/Epigenética(2.486 produtos)
- Sinalização Citoesquelética(1.542 produtos)
- Dano de DNA/Reparo de DNA(2.945 produtos)
- Endocrinologia/Hormónios(3.706 produtos)
- Enzima(3.670 produtos)
- GPCR/Proteína-G(9.023 produtos)
- Imunologia e Inflamação(3.898 produtos)
- Vírus da Influenza(302 produtos)
- Sinalização JAK/STAT(415 produtos)
- Sinalização MAPK(1.248 produtos)
- Transportador de Membranas/Canal Iónico(3.071 produtos)
- Metabolismo(10.180 produtos)
- Microbiologia/Virologia(7.620 produtos)
- Neurociência(10.369 produtos)
- Outros inibidores(35.955 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.442 produtos)
- Proteases/Proteassoma(1.719 produtos)
- Células - tronco e Derivados(806 produtos)
- Tirosina Quinase/Adaptador(2.033 produtos)
- Ubiquitinação(1.719 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66631 produtos de "Inibidores"
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D-Mannitol
CAS:D-Mannitol (Mannitol) is a diuretic and renal diagnostic aid related to sorbitol.Fórmula:C6H14O6Pureza:99.66% - 99.68%Cor e Forma:Orthorhombic Needles From Alc (Ntp 1992)Peso molecular:182.17Fosamprenavir Calcium Salt
CAS:Fosamprenavir Calcium Salt (GW433908G) (GW433908G) is a phosphate ester prodrug of the antiretroviral protease inhibitor Amprenavir, with improved solubility.Fórmula:C25H34CaN3O9PSPureza:98.68% - 99.24%Cor e Forma:White Microcrystalline NeedlesPeso molecular:623.67Nidanilimab
CAS:<p>Nidanilimab (CAN04) is an IL1RAP antibody with 1.10 pM affinity and antitumor effects on NSCLC and PDAC.</p>Pureza:> 95%Cor e Forma:SoildPeso molecular:150 kDaKetanserin
CAS:Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Fórmula:C22H22FN3O3Pureza:99.19% - 99.73%Cor e Forma:SolidPeso molecular:395.43Aluminum Hydroxide
CAS:Aluminum Hydroxide: oral adjuvant, aids vaccine potency, enhances immune response.Fórmula:AlH3O3Pureza:98%Cor e Forma:White Solid PowderPeso molecular:78Nacubactam
CAS:Nacubactam (OP0595 free acid) is a potent inhibitor of non-β-lactam-β-lactamase with activity against class A and class C β-lactamases.Fórmula:C9H16N4O7SPureza:98.93%Cor e Forma:SolidPeso molecular:324.31Ref: TM-T12166
1mg59,00€5mg126,00€10mg207,00€25mg414,00€50mg622,00€100mg885,00€1mL*10mM (DMSO)140,00€Cloperastine hydrochloride
CAS:Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.Fórmula:C20H25Cl2NOPureza:97.74% - 99.42%Cor e Forma:SolidPeso molecular:366.33Azatadine dimaleate
CAS:<p>Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).</p>Fórmula:C28H30N2O8Pureza:99.7% - >99.99%Cor e Forma:PowderPeso molecular:522.55Olsalazine disodium
CAS:Olsalazine disodium (Dipentum) is bioconverted to 5-aminosalicylic acid (5-ASA) in the colon and has anti-inflammatory activity in ulcerative colitis.Fórmula:C14H8N2Na2O6Pureza:99.47% - 99.52%Cor e Forma:Yellow Crystalline PowderPeso molecular:346.2Ambroxol
CAS:Ambroxol treats respiratory diseases by thinning mucus. Active in Mucosolvan, it enhances mucus clearance and protects lungs.Fórmula:C13H18Br2N2OPureza:99.72%Cor e Forma:SolidPeso molecular:378.1Butylparaben
CAS:Butylparaben (Butyl 4-hydroxybenzoate) is a standardized chemical allergen, increasing histamine release, and cell-mediated immunity.Fórmula:C11H14O3Pureza:98.15%Cor e Forma:Small Colorless Crystals Or Powder Tongue Aqueous Solutions Slightly Acidic To Litmus (Ntp 1992)Peso molecular:194.232-Acetyl-4-butyramidophenol
CAS:2-Acetyl-4-butyramidophenol is gray crystalline powder.Fórmula:C12H15NO3Pureza:99.79%Cor e Forma:SolidPeso molecular:221.25ISRIB-A15
CAS:<p>ISRIB-A15 (ISR-IN-2) is an potent inhibitor of the integrated stress response with an EC50 of 0.8 nM.</p>Fórmula:C22H22Cl4N2O4Pureza:98.5%Cor e Forma:SoildPeso molecular:520.23Andecaliximab
CAS:<p>Andecaliximab: IgG4 antibody against MMP9, antifibrotic in mice, studies gastric cancer, IPF, dengue.</p>Pureza:> 95%Cor e Forma:LiquidPeso molecular:150 kDaTopilutamide
CAS:Topilutamide (Fluridil) is a topical nonsteroidal antiandrogen.Fórmula:C13H11F6N3O5Pureza:98.77% - 99.24%Cor e Forma:SolidPeso molecular:403.23Ref: TM-T13184
1mg56,00€5mg119,00€10mg188,00€25mg393,00€50mg615,00€100mg877,00€200mg1.198,00€1mL*10mM (DMSO)131,00€Nortropine
CAS:Nortropine (Nortropenol) is used as muscarinic receptor antagonists.Fórmula:C7H13NOPureza:99.18%Cor e Forma:Light Tan SolidPeso molecular:127.18Etofibrate
CAS:Etofibrate is a combination of clofibrate and niacin, used to treat hyperlipemia.Fórmula:C18H18ClNO5Pureza:98.74%Cor e Forma:White To Off-White SolidPeso molecular:363.79Clofazimine
CAS:Clofazimine, a phenazine dye, has anti-mycobacterial/inflammatory effects, targeting Mycobacterium leprae and others.Fórmula:C27H22Cl2N4Pureza:98.23% - 99.85%Cor e Forma:SolidPeso molecular:473.4Naringenin
CAS:<p>Naringenin (NSC-11855) is a bioactive flavanone with antioxidant, anti-inflammatory properties, aids in carbohydrate metabolism, immunity, and DNA repair.</p>Fórmula:C15H12O5Pureza:98.10% - 99.52%Cor e Forma:SolidPeso molecular:272.25Betaine chloride
CAS:Betaine chloride (Betaine hydrochloride) gains the amplification of DNA by decreasing the formation of secondary structure in GC-rich regions.Fórmula:C5H12ClNO2Pureza:99.98%Cor e Forma:Colorless To White CrystalsPeso molecular:153.61Sodium Nitroprusside
CAS:Sodium Nitroprusside (Ro 21-2498) is a potent vasodilator, releasing in blood with no spontaneously.Fórmula:Na2Fe(CN)5NOPureza:98%Cor e Forma:SolidPeso molecular:261.92Epertinib hydrochloride
CAS:Epertinib hydrochloride (S-22611 hydrochloride) shows potent antitumor activity.Fórmula:C30H28Cl2FN5O3Pureza:99.14%Cor e Forma:SolidPeso molecular:596.48Ref: TM-T11213
1mg92,00€5mg188,00€10mg311,00€25mg533,00€50mg755,00€100mg1.017,00€500mg2.043,00€1mL*10mM (DMSO)255,00€SAR405 R enantiomer
CAS:SAR405 R enantiomer is the less active enantiomer of SAR405. SAR405 is an inhibitor of PIK3C3/Vps34.Fórmula:C19H21ClF3N5O2Pureza:98.04%Cor e Forma:SolidPeso molecular:443.85Ref: TM-T12831
1mg48,00€5mg92,00€10mg158,00€25mg261,00€50mg379,00€100mg530,00€200mg722,00€1mL*10mM (DMSO)89,00€5-CFDA
CAS:5-CFDA is a cell-permeable compound that, once inside cells, is converted to 5-carboxyfluorescein for labeling cells in fluorescence microscopy.Fórmula:C25H16O9Pureza:97.16% - 97.51%Cor e Forma:SolidPeso molecular:460.39Rosiglitazone maleate
CAS:Rosiglitazone maleate (BRL 49653) is an oral antidiabetic and potential anticancer agent.Fórmula:C22H23N3O7SPureza:99.33% - 99.51%Cor e Forma:Off-White SolidPeso molecular:473.50Gestodene
CAS:Gestodene (WL 70) is a progestogen hormonal contraceptive.Fórmula:C21H26O2Pureza:98% - 99.68%Cor e Forma:White Crystalline SolidPeso molecular:310.43PF-3450074
CAS:PF-3450074 (PF-74) is a specific HIV-1 inhibitor, blocking viral replication and uncoating at submicromolar EC50=8-640 nM.Fórmula:C27H27N3O2Pureza:99.92%Cor e Forma:SolidPeso molecular:425.52Isatuximab
CAS:Isatuximab targets CD38 in blood cancers, with high expression in multiple myeloma, inducing apoptosis and impairing cellular functions.Pureza:SDS-PAGE:97.4%;SEC-HPLC:98.4%Cor e Forma:LiquidPeso molecular:145.21 kDa(25R)-3β,17α-dihydroxy-5α- spirostan-6-one3-O-α-L- rhamnopyranosyl-(1→2)-β- D-glucopyranoside
CAS:(25R)-3β,17α-dihydroxy-5α- spirostan-6-one3-O-α-L- rhamnopyranosyl-(1→2)-β- D-glucopyranoside is a natural product isolated from the bulbs of Lilium brownii varFórmula:C39H62O14Pureza:99.95%Cor e Forma:SolidPeso molecular:754.9Ethamsylate
CAS:Ethamsylate (Dicynene) 通常用作止血药,增加毛细血管内皮阻力和血小板粘附,抑制前列腺素的生物合成和作用。Fórmula:C10H17NO5SPureza:98.55%Cor e Forma:White Crystals Or Crystalline PowderPeso molecular:263.31CC-885
CAS:CC-885 is a modulator of cereblon (CRBN). It has potent anti-tumour activity.Fórmula:C22H21ClN4O4Pureza:99.08% - 99.83%Cor e Forma:SolidPeso molecular:440.88Ref: TM-T14893
1mg56,00€5mg119,00€10mg169,00€25mg305,00€50mg495,00€100mg722,00€1mL*10mM (DMSO)139,00€Metacavir
CAS:Metacavir, a reverse transcriptase inhibitor, is used potentially for the treatment of HBV infection.Fórmula:C11H15N5O3Pureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:265.27NBD-556
CAS:NBD-556 is a small molecule mimetic of CD4. NBD-556 recognizes the HIV-1 envelope protein gp120 and induces restructuring of gp120 analogous to CD4 binding.Fórmula:C17H24ClN3O2Pureza:99.79%Cor e Forma:SolidPeso molecular:337.845-hydroxytryptophan
CAS:5-hydroxytryptophan (NSC-92523) is the immediate precursor in the biosynthesis of SEROTONIN from tryptophan. It is used as an antiepileptic and antidepressant.Fórmula:C11H12N2O3Pureza:99.52%Cor e Forma:Minute Rods Or Needles From Ethanol White SolidPeso molecular:220.22Brodalumab
CAS:Brodalumab (AMG 827), a human IgG2 monoclonal antibody, inhibits IL-17R, treating psoriasis.Pureza:98.3%Cor e Forma:LiquidPeso molecular:144.06 kDaBMS-986158
CAS:BMS-986158: BET inhibitor, IC50 of 6.6 nM in SCLC, 5 nM in TNBC cells.Fórmula:C30H33N5O2Pureza:98.78%Cor e Forma:SolidPeso molecular:495.62Ref: TM-T14685
1mg87,00€5mg259,00€10mg465,00€25mg745,00€50mg1.026,00€100mg1.388,00€1mL*10mM (DMSO)283,00€Regorafénib N-oxyde (M2)
CAS:<p>Regorafénib N-oxyde M2 is an active metabolite of Regorafenib.</p>Fórmula:C21H15ClF4N4O4Pureza:98.03% - 98.26%Cor e Forma:SolidPeso molecular:498.812,5-Dihydroxybenzoic acid
CAS:2,5-Dihydroxybenzoic acid (Gentisic acid) is an active metabolite of salicylic acid degradation with a broad spectrum of biological activity.Fórmula:C7H6O4Pureza:99.63%Cor e Forma:SolidPeso molecular:154.12Risedronic Acid
CAS:Risedronic Acid (Risedronate), a pyridinyl biphosphonate, can inhibit osteoclast-mediated bone resorption.Fórmula:C7H11NO7P2Pureza:99.85% - 99.87%Cor e Forma:White Crystalline PowderPeso molecular:283.11TMN355
CAS:TMN355 is a potent chemical inhibitor of cyclophilin A and reduces foam cell formation and cytokine secretion,and is used for atherosclerosis.Fórmula:C21H14ClFN2O2Pureza:99.15%Cor e Forma:SolidPeso molecular:380.8Ref: TM-T13171
1mg42,00€2mg55,00€5mg88,00€10mg120,00€25mg235,00€50mg354,00€100mg520,00€500mg1.111,00€1mL*10mM (DMSO)87,00€Mucic Acid
CAS:Mucic Acid (Tetrahydroxyadipic acid) is an aldaric acid obtained by nitric acid oxidation of galactose or galactose-containing compounds.Fórmula:C6H10O8Pureza:99.31%Cor e Forma:Crystalline Powder SolidPeso molecular:210.14Nepafenac
CAS:Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.Fórmula:C15H14N2O2Pureza:98.94% - 99.43%Cor e Forma:SolidPeso molecular:254.289-Aminoacridine
CAS:9-Aminoacridine is a fluorescent anti-infective dye used clinically as a topical antiseptic and experimentally as a mutagen, due to its interaction with DNA.Fórmula:C13H10N2Pureza:98.74% - 99.93%Cor e Forma:Pale Yellow CrystalsPeso molecular:194.23Maritoclax
CAS:Maritoclax (Marinopyrrole A) (Marinopyrrole A) is a novel and specific Mcl-1 inhibitor, shows >8 fold selectivity than BCL-xl (IC50 > 80 μM),with an IC50 valueFórmula:C22H12Cl4N2O4Pureza:99.87%Cor e Forma:SolidPeso molecular:510.15Ref: TM-T11944
1mg46,00€2mg59,00€5mg87,00€10mg144,00€25mg279,00€50mg520,00€100mg725,00€1mL*10mM (DMSO)96,00€Cecropin B acetate
Cecropin B acetate activates NF-κB, inhibits CYP3A29, disrupts PXR/RXR-α-DNA binding, and has potent antimicrobial properties.Pureza:99.27%Cor e Forma:LiquidDegarelix acetate(214766-78-6 free base)
CAS:Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .Fórmula:C84H107ClN18O18Pureza:98.66%Cor e Forma:SolidPeso molecular:1692.34Aminothiazole
CAS:Aminothiazole (2-Aminothiazole), a thyroid inhibitor, displays antibacterial activity.Fórmula:C3H4N2SPureza:98.87%Cor e Forma:Physical Description Light Brown Crystals Or Brown Granular Solid (Ntp 1992)Peso molecular:100.14GSK256073
CAS:GSK256073 is an orally active GPR109A agonist.Fórmula:C10H13ClN4O2Pureza:98.46%Cor e Forma:SolidPeso molecular:256.69Ref: TM-T15432
1mg73,00€2mg97,00€5mg160,00€10mg250,00€25mg439,00€50mg647,00€100mg920,00€1mL*10mM (DMSO)170,00€Loxeen
CAS:Loxeen (Pridinol methanesulfonate) is used as an anticholinergic and as an antiparkinsonian agent.Fórmula:C20H25NO·CH4O3SPureza:99.46%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:391.52Theaflavin-3-gallate
CAS:Theaflavin-3-gallate reduces cholesterol absorption, has anticancer effects, and induces oxidative stress in lung cancer.Fórmula:C36H28O16Pureza:98.28% - 99.63%Cor e Forma:SolidPeso molecular:716.60

