
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.524 produtos)
- Apoptose(5.793 produtos)
- Ciclo celular/Ponto de verificação(4.452 produtos)
- Cromatina/Epigenética(2.242 produtos)
- Sinalização Citoesquelética(1.382 produtos)
- Dano de DNA/Reparo de DNA(2.826 produtos)
- Endocrinologia/Hormónios(3.507 produtos)
- Enzima(3.640 produtos)
- GPCR/Proteína-G(8.333 produtos)
- Imunologia e Inflamação(3.527 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(404 produtos)
- Sinalização MAPK(1.203 produtos)
- Transportador de Membranas/Canal Iónico(2.792 produtos)
- Metabolismo(9.449 produtos)
- Microbiologia/Virologia(6.981 produtos)
- Neurociência(9.926 produtos)
- Outros inibidores(37.921 produtos)
- Oxidação-Redução(41 produtos)
- Sinalização PI3K/Akt/mTOR(1.400 produtos)
- Proteases/Proteassoma(1.597 produtos)
- Células - tronco e Derivados(830 produtos)
- Tirosina Quinase/Adaptador(2.015 produtos)
- Ubiquitinação(1.650 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66639 produtos de "Inibidores"
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7-Aminoactinomycin D
CAS:<p>7-Aminoactinomycin D is a fluorescent DNA stain.</p>Fórmula:C62H87N13O16Pureza:98%Cor e Forma:Red To Dark Purple PowderPeso molecular:1270.453Neuronostatin-13 (human)
CAS:<p>Neuronostatin-13: human-conserved, 13-amino-acid peptide with amidated C-terminus.</p>Fórmula:C64H110N20O16Pureza:98%Cor e Forma:SolidPeso molecular:1415.68Asperosaponin IV
CAS:<p>Asperosaponin IV is a natural product for research related to life sciences. The catalog number is TN5282 and the CAS number is 126778-93-6.</p>Fórmula:C49H78O19Pureza:98%Cor e Forma:SolidPeso molecular:971.13N-(DBCO-PEG4)-N-Biotin-PEG4-NHS
CAS:<p>N-(DBCO-PEG4)-N-Biotin-PEG4-NHS is a PEG-based PROTAC linker suitable for synthesizing PROTACs[1].</p>Fórmula:C54H74N6O16SPureza:98%Cor e Forma:SolidPeso molecular:1095.265,7-Dimethoxy-4-methylcoumarin
CAS:<p>5,7-Dimethoxy-4-methylcoumarin has potential antioxidant antiproliferative and anticancer or activity.</p>Fórmula:C12H12O4Pureza:98.42%Cor e Forma:SoildPeso molecular:220.22ML267
CAS:<p>ML267 (4-(3-chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-methoxypyridin-2-yl)piperazine-1-carbothioamide trifluoroacetate) is a potent inhibitor of bacterial</p>Fórmula:C19H18ClF6N5O3SPureza:97.85%Cor e Forma:SolidPeso molecular:545.89Cefatrizine
CAS:<p>Cefatrizine inhibits eEF-2 kinase, affecting apoptosis, autophagy, and ER stress in cancers.</p>Fórmula:C18H18N6O5S2Pureza:98%Cor e Forma:SolidPeso molecular:462.5SMD-3040
CAS:<p>SMD-3040 is a potent and selective SMARCA2 PROTAC degrader (DC50: 12 nM), which consists of an SMARCA2/4 ligand, a linker, and a VHL ligand.</p>Fórmula:C52H66N10O5SPureza:98%Cor e Forma:SolidPeso molecular:943.21DGN462
CAS:<p>DGN462: DNA alkylator, anti-tumor, targets AML, for ADC cytotoxic parts.</p>Fórmula:C53H59N5O9SPureza:98%Cor e Forma:SolidPeso molecular:942.13UCL 1684 dibromide
CAS:<p>apamin-sensitive Ca2+-activated K+ channel (KCa2.1) blocker</p>Fórmula:C34H30Br2N4Pureza:98%Cor e Forma:SolidPeso molecular:654.45SPDP-C6-Gly-Leu-NHS ester
<p>SPDP-C6-Gly-Leu-NHS ester is a cleavable linker employed in the synthesis of antibody-drug conjugates (ADCs)[1].</p>Fórmula:C26H37N5O7S2Pureza:98%Cor e Forma:SolidPeso molecular:595.73ACTH 4-11 acetate
<p>ACTH 4-11 acetate, a fragment of adrenocorticotropin, matches α-MSH's sequence and has weak MSH potency at high doses (100-1000 nM).</p>Fórmula:C52H75N15O13SPureza:99.21%Cor e Forma:SolidPeso molecular:1150.31Angiotensinogen (1-14), human acetate
<p>Angiotensinogen (1-14), human acetate is a fragment of angiotensinogen which is a passive substrate of the renin-angiotensin system.</p>Fórmula:C85H126N24O21Pureza:98.4%Cor e Forma:SolidPeso molecular:1820.0626RFa Acetate (mouse,rat)
<p>Orphan GPCR SP9155 agonist P550 (mouse, rat) acetate (Orphan GPCR SP9155 agonist P550 ) is a member of the RFamide peptide family with orexigenic effects.</p>Fórmula:C128H199N37O39Pureza:98.49%Cor e Forma:SolidPeso molecular:2880.17Emoghrelin
CAS:<p>Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the ghrelin receptor [1].</p>Fórmula:C24H22O13Pureza:98%Cor e Forma:SolidPeso molecular:518.42Lanepitant
CAS:<p>Lanepitant (LY303870) is a non-peptide neurokinin-1 (NK-1) antagonist with analgesic activity for the prevention of migraine.</p>Fórmula:C33H45N5O3Pureza:97.71%Cor e Forma:SolidPeso molecular:559.74Strictosidine
CAS:<p>Strictosidine has DNA damaging activity in yeast RS 188N mutant, assessed as drug level required to produce 12 mm zone of inhibition.</p>Fórmula:C27H34N2O9Pureza:98%Cor e Forma:SolidPeso molecular:530.57Pristane
CAS:<p>Pristane (2,6,10,14-tetramethylpentadecane) is a natural product from shark liver oil and a non-antigenic adjuvant.</p>Fórmula:C19H40Pureza:98.67% - 99.47%Cor e Forma:Colorless Transparent; Stable Liquid SolidPeso molecular:268.52DL-m-Tyrosine
CAS:<p>DL-m-Tyrosine shows effects on Arabidopsis root growth.</p>Fórmula:C9H11NO3Pureza:98%Cor e Forma:White CrystalsPeso molecular:181.1885Sanshodiol
CAS:<p>Sanshodiol is a natural product of Zanthoxylum, Rutaceae.</p>Fórmula:C20H22O6Pureza:98%Cor e Forma:SolidPeso molecular:358.39Daphnilongeranin A
CAS:<p>Daphnilongeranin A is a natural product from Cimicifuga foetida L.</p>Fórmula:C23H29NO4Pureza:98%Cor e Forma:SolidPeso molecular:383.48Iodo-PEG4-N3
CAS:<p>Iodo-PEG4-N3 is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Fórmula:C8H16IN3O3Pureza:98%Cor e Forma:SolidPeso molecular:329.144'-O-Methylvitexin
CAS:<p>4'-O-Methylvitexin is a natural product for research related to life sciences. The catalog number is TN3064 and the CAS number is 2326-34-3.</p>Fórmula:C22H22O10Pureza:98%Cor e Forma:SolidPeso molecular:446.4[Orn8]-Urotensin II acetate
<p>[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.</p>Fórmula:C65H87N13O20S2Pureza:98.63%Cor e Forma:SolidPeso molecular:1434.59Lipofermata
CAS:<p>Lipofermata is a fatty acid transport protein (FATP) inhibitor that prevents lipid transport to melanoma cells and reduces melanoma growth and invasion.</p>Fórmula:C15H10BrN3OSPureza:99.22% - 99.57%Cor e Forma:SolidPeso molecular:360.23PD-1-IN-20
<p>PD-1-IN-20 is the less active enantiomer of PD-1-IN-1.</p>Fórmula:C12H20N6O7Pureza:98%Cor e Forma:SolidPeso molecular:360.32m-PEG7-CH2-OH
CAS:<p>m-PEG7-CH2-OH is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Fórmula:C16H34O8Pureza:98%Cor e Forma:SolidPeso molecular:354.44m-PEG4-amino-Mal
CAS:<p>m-PEG4-amino-Mal is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Fórmula:C16H26N2O7Pureza:98%Cor e Forma:SolidPeso molecular:358.39H 256
CAS:<p>H 256 is a pepsin heptapeptide inhibitor.</p>Fórmula:C43H62N10O12Pureza:98%Cor e Forma:SolidPeso molecular:911.0273MB-PP1
CAS:<p>3MB-PP1 is a bulky purine analog and a Polo-like kinase 1 (Plk1) inhibitor.</p>Fórmula:C17H21N5Pureza:99.96%Cor e Forma:White SolidPeso molecular:295.3820-Hydroxyaflavinine
CAS:<p>20-Hydroxyaflavinine is a natural product from the metabolites of the ascomycete fungus Tricladium sp.</p>Fórmula:C28H39NO2Pureza:98%Cor e Forma:SolidPeso molecular:421.61wt hMLN
<p>Wild-type human myoregulin (wt hMLN) is a microprotein that inhibits the sarcoplasmic reticulum Ca²⁺ pump (SERCA), playing a crucial role in the regulation of</p>Fórmula:C245H404N54O66SPureza:98%Cor e Forma:SolidPeso molecular:5194.22Impurity C of Alfacalcidol
CAS:<p>Impurity of Alfacalcidol is an impurity of Alfacalcidol. Alfacalcidol is a non-selective VDR activator medication.</p>Fórmula:C35H49N3O4Pureza:98%Cor e Forma:SolidPeso molecular:575.78N3-PEG6-Propanehydrazide
<p>N3-PEG6-Propanehydrazide: a PEG-based linker for PROTACs synthesis.</p>Fórmula:C15H31N5O7Pureza:98%Cor e Forma:SolidPeso molecular:393.44Sennidin A
CAS:<p>Sennidin A, has two hydroxyanthraquinone-like moieties, exerts inhibition on NS3 helicase with IC50 values of 0.8 μM.</p>Fórmula:C30H18O10Pureza:98%Cor e Forma:SolidPeso molecular:538.46(Iso)-RJW100
CAS:<p>Potent LRH-1/NR5A2 and SF-1/NR5A1 agonist; pEC50: 6.4 (LRH-1), 7.2 (SF-1).</p>Fórmula:C28H34OPureza:99.79%Cor e Forma:SoildPeso molecular:386.578-Deacetylyunaconitine
CAS:<p>8-Deacetylyunaconitine is a a diterpenoid alkaloid derived from Aconitum Vilmorinian Radix.</p>Fórmula:C33H47NO10Pureza:99.73%Cor e Forma:SolidPeso molecular:617.73Casein kinase 1δ-IN-3
CAS:<p>Casein kinase 1δ-IN-3 (Casein kinase 1δ-IN-3) (Compound 23a) is a casein kinase 1 delta (CK1d) inhibitor with a pIC50 of 6.5376 M.</p>Fórmula:C17H16N2O2SPureza:98.94%Cor e Forma:SoildPeso molecular:312.39AD57
CAS:<p>AD57 is a potent inhibitor of both c-Src and Abl with IC50 of 0.025 μM and 0.041 μM, respectively.</p>Fórmula:C22H20F3N7OPureza:99.05%Cor e Forma:SoildPeso molecular:455.44Dihydroepistephamiersine 6-acetate
CAS:<p>Dihydroepistephamiersine 6-acetate is a natural product for research related to life sciences. The catalog number is TN3850 and the CAS number is 57361-74-7.</p>Fórmula:C23H31NO7Pureza:98%Cor e Forma:SolidPeso molecular:433.501Biotin-PEG3-alcohol
CAS:<p>Biotin-PEG3-alcohol is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Fórmula:C16H29N3O5SPureza:98%Cor e Forma:SolidPeso molecular:375.48Syringin pentaacetate
CAS:<p>Syringin pentaacetate is a natural product for research related to life sciences. The catalog number is TN5087 and the CAS number is 92233-55-1.</p>Fórmula:C27H34O14Pureza:98%Cor e Forma:SolidPeso molecular:582.55DC-S239
CAS:<p>Ethyl 2-amino-4-methyl-5-thiophene carboxylate is a SETD7 inhibitor (IC50=4.59μM) with anticancer properties.</p>Fórmula:C15H15N3O5SPureza:99.37%Cor e Forma:SolidPeso molecular:349.36Senkyunolide A
CAS:<p>Senkyunolide A is a natural product isolated from Ligusticum chuanxiong Hort, with anti-tumor activity.</p>Fórmula:C12H16O2Pureza:99.52%Cor e Forma:SolidPeso molecular:192.258α-Methacryloyloxy-13-ethoxyvernojalcanolide
CAS:8alpha-Methacryloyloxy-13-ethoxyvernojalcanolide is a natural product for research related to life sciences.Fórmula:C25H34O11Pureza:98%Cor e Forma:SolidPeso molecular:510.5363α-Acetoxy-20(29)-lupene-23,28-dioic acid
CAS:<p>3alpha-Acetoxy-20(29)-lupene-23,28-dioic acid is a natural product for research related to life sciences.</p>Fórmula:C32H48O6Pureza:98%Cor e Forma:SolidPeso molecular:528.72BTK inhibitor 17
CAS:<p>BTK inhibitor 17 is a potent irreversible BTK inhibitor (IC50 = 2.1 nM). BTK inhibitor 17 can be used in rheumatoid arthritis studies.</p>Fórmula:C25H24N6O3Pureza:99.57% - 99.88%Cor e Forma:SolidPeso molecular:456.5Polyphyllin H
CAS:<p>Polyphyllin H can be extracted from loblolly pine and rhizomes, has antitumor activity, and is used in studies of inflammation, fractures, and convulsions.</p>Fórmula:C44H70O17Pureza:99.01%Cor e Forma:SolidPeso molecular:871.02Excisanin B
CAS:<p>Excisanin B shows inhibitory effects on LPS-induced production of nitric oxide in murine macrophage RAW264.7 cells.</p>Fórmula:C22H32O6Pureza:98%Cor e Forma:SolidPeso molecular:392.499α,13α-Epidioxyabiet-8(14)-en-18-oic acid
CAS:9alpha,13alpha-Epidioxyabiet-8(14)-en-18-oic acid shows potent inhibitory effects on Epstein-Barr virus early antigen (EBV-EA) activation induced by the tumorFórmula:C20H30O4Pureza:98%Cor e Forma:SolidPeso molecular:334.45

