
Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.542 produtos)
- Apoptose(5.816 produtos)
- Ciclo celular/Ponto de verificação(4.466 produtos)
- Cromatina/Epigenética(2.252 produtos)
- Sinalização Citoesquelética(1.381 produtos)
- Dano de DNA/Reparo de DNA(2.830 produtos)
- Endocrinologia/Hormónios(3.518 produtos)
- Enzima(3.640 produtos)
- GPCR/Proteína-G(8.362 produtos)
- Imunologia e Inflamação(3.540 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(405 produtos)
- Sinalização MAPK(1.201 produtos)
- Transportador de Membranas/Canal Iónico(2.809 produtos)
- Metabolismo(9.462 produtos)
- Microbiologia/Virologia(7.003 produtos)
- Neurociência(9.942 produtos)
- Outros inibidores(37.827 produtos)
- Oxidação-Redução(40 produtos)
- Sinalização PI3K/Akt/mTOR(1.399 produtos)
- Proteases/Proteassoma(1.598 produtos)
- Células - tronco e Derivados(830 produtos)
- Tirosina Quinase/Adaptador(2.012 produtos)
- Ubiquitinação(1.651 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66618 produtos de "Inibidores"
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N-DMTr-morpholino-T-5'-O-phosphoramidite
<p>N-DMTr-morpholino-T-5'-O-phosphoramidite is a Nucleoside Phosphoramidite.</p>Cor e Forma:SoildFluorizoline
CAS:<p>Fluorizoline is a PHB-binding compound with anticancer and antiproliferative activity and induces apoptosis.</p>Fórmula:C15H8Cl2F3NSPureza:98.22% - 99.52%Cor e Forma:SolidPeso molecular:362.20Propanil
CAS:Propanil is a widely used contact herbicide. It is mainly used in rice production.Fórmula:C9H9Cl2NOPureza:98%Cor e Forma:Propanil Is A Colorless To Brown Crystals Non Corrosive Used As An HerbicidePeso molecular:218.08Buparlisib Hydrochloride
CAS:<p>Buparlisib Hydrochloride is an inhibitor of pan-class I PI3K (IC50: 52 nM/166 nM/116 nM/262 nM for p110α/p110β/p110δ/p110γ, respectively).</p>Fórmula:C18H22ClF3N6O2Pureza:98.94%Cor e Forma:SolidPeso molecular:446.85Hexaethylene glycol monomethyl ether
CAS:Hexaethylene glycol monomethyl ether, a PEG-based PROTAC linker, facilitates the synthesis of PROTACs[1].Fórmula:C13H28O7Cor e Forma:SolidPeso molecular:296.362-Hydroxymethyltetrahydropyran
CAS:<p>2-Hydroxymethyltetrahydropyran is a volatile compound present in the seed oil of Sambucus williamsii (SW), which possesses promising antioxidant activity.</p>Fórmula:C6H12O2Cor e Forma:SolidPeso molecular:116.16Triptotriterpenic acid A
CAS:<p>Triptotriterpenic acid A (Abrusgenic acid) is isolated from Tripterygium wilfordii and has potential hepatotoxicity for the study of rheumatoid arthritis.</p>Fórmula:C30H48O4Pureza:98%Cor e Forma:SolidPeso molecular:472.79-Decyn-1-ol
CAS:9-Decyn-1-ol links GDC-0068 to Lenalidomide, forming INY-03-041, a selective Akt degrader with low IC50s.Fórmula:C10H18OCor e Forma:SolidPeso molecular:154.253'-Deoxy-3'-fluorocytidine
CAS:<p>3'-Deoxy-3'-fluorocytidine is a nucleoside, fluoro-modified nucleoside.</p>Fórmula:C9H12FN3O4Cor e Forma:SolidPeso molecular:245.21N4-(1,1,1,-Trifluoropropanoyl)cytidine
<p>N4-(1,1,1,-Trifluoropropanoyl)cytidine is a useful organic compound for research related to life sciences and the catalog number is TNU0842.</p>Cor e Forma:SoildThiol-PEG4-acid
CAS:Thiol-PEG4-acid is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.Fórmula:C11H22O6SPureza:98%Cor e Forma:SolidPeso molecular:282.355β-Dihydroprogesterone
CAS:5β-Dihydroprogesterone (5β-DHP) is a progesterone receptor agonist and metabolite of progesterone .1,2It is formed from progesterone by 5β-reductase.25β-DHPFórmula:C21H32O2Cor e Forma:SolidPeso molecular:316.4853'-O-Hexadecanyl adenosine
<p>3’-O-Hexadecanyl adenosine is a useful organic compound for research related to life sciences and the catalog number is TNU1650.</p>Cor e Forma:Soild5'-DMTr-T-Methyl phosphonamidite
CAS:<p>5'-DMTr-T-Methyl phosphonamidite is a Nucleoside Derivative - phosphonamidite.</p>Fórmula:C38H48N3O7PCor e Forma:SolidPeso molecular:689.781-[(5E)-5,6-Dideoxy-6-(diethoxyphosphinyl)-2-O-(2-methoxyethyl)-β-D-ribo-hex-5-enofuranosyl]uracil
<p>1-[(5E)-5,6-Dideoxy-6-(diethoxyphosphinyl)-2-O-(2-methoxyethyl)-β-D-ribo-hex-5-enofuranosyl]uracil is a useful organic compound for research related to life</p>Cor e Forma:Solid2',3'-Isopropylidene-isocytidine
CAS:<p>Nucleoside - isocytidine derivative</p>Fórmula:C12H17N3O5Cor e Forma:SolidPeso molecular:283.283',5'-Di-O-acetyl-2'-deoxy-5,N3-dimethyl uridine
CAS:<p>3',5'-Di-O-acetyl-2'-deoxy-5,N3-dimethyl uridine is a Nucleoside Derivative - N-Alkylated nucleoside.</p>Fórmula:C15H20N2O7Cor e Forma:SolidPeso molecular:340.33Lenalidomide-4-aminomethyl hydrochloride
CAS:<p>Lenalidomide-4-aminomethyl HCl, a CRBN ligand, aids in PROTAC formation by recruiting CRBN protein.</p>Fórmula:C14H16ClN3O3Cor e Forma:SolidPeso molecular:309.756-Chloro-7-fluoro-7-deazapurine
CAS:<p>6-Chloro-7-fluoro-7-deazapurine bolongs toIntermediates and Building Blocks - Nucleoside Base; Multi-functional; Heterocyclic Compounds - Purine; Scaffold and</p>Fórmula:C6H3ClFN3Cor e Forma:SolidPeso molecular:171.56N6-MethyladenosineN1-oxide
CAS:<p>Nucleoside Derivatives –6-Modified purine nucleosides;N-Methylated nucleosides; Drugs and Inhibitors; Antiviral agent</p>Fórmula:C11H15N5O5Cor e Forma:SolidPeso molecular:297.275-Fluorouracil-1-yl acetic acid
CAS:<p>5-Fluorouracil-1-yl acetic acid is a PNA-related Derivative.</p>Fórmula:C6H5FN2O4Cor e Forma:SolidPeso molecular:188.112',3',5'-Tri-O-acetyl-5-methoxycarbonylmethyl-2-thiouridine
CAS:<p>Nucleoside Derivatives - 5-Modified pyrimidine nucleosides; Thio-nucleosides</p>Fórmula:C18H22N2O10SCor e Forma:SolidPeso molecular:458.44Disitamab
CAS:<p>Disitamab (RC48-0) is a humanized anti-HER2 monoclonal antibody used in ADC synthesis.</p>Pureza:95.00%Cor e Forma:Liquid2'-Deoxy-2'-(N-trifluoroacetyl)amino-5'-O-DMTr-uridine 3'-CED phosphoramidite
CAS:<p>2’-Deoxy-2’-(N-trifluoroacetyl)amino-5’-O-DMTr-uridine 3’-CED phosphoramidite is a useful organic compound for research related to life sciences.</p>Fórmula:C41H47F3N5O9PCor e Forma:SolidPeso molecular:841.81N6-Benzoylarabinoadenosine
CAS:<p>Nucleoside Derivatives - Arabino-nucleosides</p>Fórmula:C17H17N5O5Cor e Forma:SolidPeso molecular:371.355'-Protected 2,2'-anhydrouridine
CAS:<p>Nucleoside Derivatives - Anhydro-nucleosides; Protected nucleosides with NH2/OH group</p>Fórmula:C30H28N2O7Cor e Forma:SolidPeso molecular:528.551,4-Dideoxy-1,4-epithio-D-ribitol
CAS:<p>1,4-Dideoxy-1,4-epithio-D-ribitol is a purine nucleoside analog that targets malignant tumors of the inert lymphatic system and possesses a broad spectrum of</p>Fórmula:C5H10O3SPureza:99.76%Cor e Forma:SolidPeso molecular:150.2Padsevonil
CAS:<p>Padsevonil (UCB-0942) is a potential GABA A receptor orthosteric modulator with antiepileptic activity for the treatment of epilepsy.</p>Fórmula:C14H14ClF5N4O2SPureza:99.63%Cor e Forma:SolidPeso molecular:432.801,10-Decanediamine, dihydrochloride
CAS:<p>1,10-Decanediamine, dihydrochloride is a biochemical.</p>Fórmula:C10H26Cl2N2Cor e Forma:SolidPeso molecular:245.23Loperamide-d6 hydrochloride
CAS:Loperamide D6 HCl: Deuterium-enriched opioid for diarrhea.Fórmula:C29H34Cl2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:519.545'-Deoxy-5-methyluridine
CAS:<p>5'-Deoxy-5-methyluridine is a Nucleoside Derivative - 5'-Modified nucleoside;5'-Deoxy nucleoside.</p>Fórmula:C10H14N2O5Cor e Forma:SolidPeso molecular:242.23(1,2-Dihydro-2-oxo-1,8-naphthyridin-3-yl)acetic acid ethyl ester
<p>(1,2-Dihydro-2-oxo-1,8-naphthyridin-3-yl)acetic acid ethyl ester is a PNA-related Derivative; Heterocyclic Compound - Fused polyheterocycle.</p>Cor e Forma:SoildTernidazole hydrochloride
CAS:<p>Ternidazole hydrochloride (Ternidazole HCl) is a 5-nitroimidazole antibiotic with antimicrobial antioxidant and antiprotozoal activity.</p>Fórmula:C7H12ClN3O3Pureza:99.70%Cor e Forma:SolidPeso molecular:221.64Biotin-C5-NHS Ester
CAS:Biotin-C5-NHS Ester is an alkyl/ether-based linker for PROTAC synthesis[1].Fórmula:C20H30N4O6SCor e Forma:White SolidPeso molecular:454.54Glyoxalase I inhibitor 6
CAS:<p>Compound 9j inhibits Glyoxalase I with 1.13 μM IC50, showing anticancer potential and low toxicity.</p>Fórmula:C18H15N3O5SCor e Forma:SolidPeso molecular:385.393-Deaza-4'-C-methyluridine
CAS:<p>Nucleoside Derivatives - 4’-Modified nucleosides; 3-Deazauridines</p>Fórmula:C11H15NO6Cor e Forma:SolidPeso molecular:257.24Cobimetinib hemifumarate
CAS:<p>Cobimetinib hemifumarate is a potent and selective MEK1 inhibitor with an IC50 value of 4.2 nM for MEK1.</p>Fórmula:C46H46F6I2N6O8Cor e Forma:SolidPeso molecular:1178.7074-(Phenylazo)diphenylamine
CAS:<p>4-(Phenylazo)diphenylamine serves as an effective colorimetric indicator for the precise quantification of strong bases, Lewis acids, and hydride reducing</p>Fórmula:C18H15N3Cor e Forma:SolidPeso molecular:273.337-TFA-ap-7-Deaza-dG
CAS:<p>5'-O-TBDMS-dG, a modified nucleoside, is utilized in the synthesis of deoxyribonucleic acid or nucleic acid.</p>Fórmula:C16H16F3N5O5Cor e Forma:SolidPeso molecular:415.329Bulleyaconitine A
CAS:<p>Bulleyaconitine A, an analgesic and antiinflammatory drug isolated from Aconitum plants, has several potential targets, such as voltage-gated Na+ channels.</p>Fórmula:C35H49NO9Pureza:99.56% - 99.76%Cor e Forma:SolidPeso molecular:627.76N4-Benzoyl-7'-OH-N-DMTr morpholino cytosine
<p>N4-Benzoyl-7'-OH-N-DMTr morpholino cytosine is a Nucleoside Derivative - Morpholino nucleoside.</p>Cor e Forma:Soild2-Amino-2'-deoxyadenosine
CAS:<p>2-Amino-2'-deoxyadenosine is a deoxyribonucleoside used for the oligonucleotide synthesis.</p>Fórmula:C10H14N6O3Cor e Forma:SolidPeso molecular:266.26Precyasterone
CAS:<p>Precyasterone is a natural compound extracted from the dried roots of Cyathula capitata.</p>Fórmula:C29H44O8Pureza:98%Cor e Forma:SolidPeso molecular:520.66L-Azidonorleucine hydrochloride
CAS:<p>L-Azidonorleucine HCl, unnatural amino acid, replaces Methionine, labels proteins, identifies MetRS mutants.</p>Fórmula:C6H13ClN4O2Cor e Forma:SolidPeso molecular:208.646NCGC00249987
CAS:<p>NCGC00249987 is a highly selective and allosteric Tyr phosphatase activity of inhibitor of Eya2(Eya2 ED and MBP-Eya2 FL with IC50s of 3 μM and 6.9 μM ).</p>Fórmula:C16H11FN4O2SPureza:98%Cor e Forma:SolidPeso molecular:342.35Isethionic acid
CAS:<p>Isethionic acid, organosulfur, in F. cylindrus, forms biodegradable surfactants; water-soluble, high-foaming.</p>Fórmula:C2H6O4SCor e Forma:SolidPeso molecular:126.13Boc-NH-PEG7-propargyl
CAS:<p>Boc-NH-PEG7-propargyl is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>Fórmula:C22H41NO9Cor e Forma:SolidPeso molecular:463.56Quinine HCl
CAS:Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.Fórmula:C20H25ClN2O2Pureza:98.00%Cor e Forma:SolidPeso molecular:360.88cGAMP
CAS:<p>cGAMP is an endogenous second messenger in metazoans and triggers interferon production in response to cytosolic DNA. It also is a STING ligand.</p>Fórmula:C20H24N10O13P2Pureza:98%Cor e Forma:SolidPeso molecular:674.41PI3K-IN-30
CAS:<p>PI3K-IN-30 (compound 6d) 是一种 PI3K 的有效抑制剂,能够作用于 PI3Kα (IC50: 5.1 nM)、PI3Kβ (IC50: 136 nM)、PI3Kγ (IC50: 30.7 nM) 和 PI3Kδ (IC50: 8.9 nM)。</p>Fórmula:C20H25F2N7O3Cor e Forma:SolidPeso molecular:449.45

