Inibidores
Os inibidores são moléculas que se ligam a enzimas, receptores ou outras proteínas para reduzir ou bloquear sua atividade biológica. Esses compostos são amplamente utilizados em pesquisas para estudar vias biológicas, entender mecanismos de doenças e desenvolver medicamentos terapêuticos. Os inibidores desempenham um papel crucial no tratamento de várias doenças, incluindo câncer, doenças cardiovasculares e infecções. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade para apoiar sua pesquisa em bioquímica, biologia celular e desenvolvimento farmacêutico.
Subcategorias de "Inibidores"
- Angiogénese(2.542 produtos)
- Apoptose(5.816 produtos)
- Ciclo celular/Ponto de verificação(4.466 produtos)
- Cromatina/Epigenética(2.252 produtos)
- Sinalização Citoesquelética(1.381 produtos)
- Dano de DNA/Reparo de DNA(2.830 produtos)
- Endocrinologia/Hormónios(3.518 produtos)
- Enzima(3.640 produtos)
- GPCR/Proteína-G(8.362 produtos)
- Imunologia e Inflamação(3.540 produtos)
- Vírus da Influenza(296 produtos)
- Sinalização JAK/STAT(405 produtos)
- Sinalização MAPK(1.201 produtos)
- Transportador de Membranas/Canal Iónico(2.809 produtos)
- Metabolismo(9.462 produtos)
- Microbiologia/Virologia(7.003 produtos)
- Neurociência(9.942 produtos)
- Outros inibidores(37.827 produtos)
- Oxidação-Redução(40 produtos)
- Sinalização PI3K/Akt/mTOR(1.399 produtos)
- Proteases/Proteassoma(1.598 produtos)
- Células - tronco e Derivados(830 produtos)
- Tirosina Quinase/Adaptador(2.012 produtos)
- Ubiquitinação(1.651 produtos)
Exibir 16 mais subcategorias
Foram encontrados 66618 produtos de "Inibidores"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
ML141
CAS:<p>ML141 (CID-2950007) is an effective, specific and reversible non-competitive inhibitor of Rho family GTPase cdc42 (IC50: 200 nM).</p>Fórmula:C22H21N3O3SPureza:99.36% - 99.56%Cor e Forma:SolidPeso molecular:407.49Nexturastat A
CAS:<p>Nexturastat A is an effective and specific HDAC6 inhibitor (IC50: 5 nM). Its selectivity is >190-fold than other HDACs.</p>Fórmula:C19H23N3O3Pureza:99.40% - 99.57%Cor e Forma:SolidPeso molecular:341.4Paris saponin VII
CAS:<p>Paris saponin VII (Dioscini) shows inhibitory effects on cell proliferation.</p>Fórmula:C51H82O21Pureza:99.51% - 99.63%Cor e Forma:SolidPeso molecular:1031.18PHGDH-inactive
CAS:<p>PHGDH inactive is inactive against PHGDH and serves as a negative control for NCT-502 and NCT-503 [1].</p>Fórmula:C17H21N5SPureza:99.83%Cor e Forma:SolidPeso molecular:327.45(S)-CPI203
CAS:<p>CPI-203 is an effective BET bromodomain inhibitor (IC50: 37 nM for BRD4).</p>Fórmula:C19H18ClN5OSPureza:99.01% - 99.92%Cor e Forma:SolidPeso molecular:399.9CGS 21680 Hydrochloride
CAS:<p>CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.</p>Fórmula:C23H29N7O6·HClPureza:96.74% - 99.53%Cor e Forma:SolidPeso molecular:535.98Procyanidin B1
CAS:Procyanidin B1, isolated from commonly eaten fruits, binds to the TLR4/MD-2 complex and has anti-inflammatory activity.Fórmula:C30H26O12Pureza:98.00% - 99.91%Cor e Forma:Red-Brown PowderPeso molecular:578.52AP1189 acetate
CAS:<p>AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.</p>Fórmula:C16H18N6O4Pureza:99.95%Cor e Forma:SolidPeso molecular:358.35LF3
CAS:LF3 is a specific inhibitor of canonical Wnt signaling by disrupting the interaction between β-catenin and TCF4 (IC50 < 2 μM)Fórmula:C20H24N4O2S2Pureza:99.63%Cor e Forma:SolidPeso molecular:416.56trans-Cinnamaldehyde
CAS:Trans-Cinnamaldehyde (Phenylacrolein) exhibits anti-inflammatory activities and antidepressant-like effects in stressed mid-aged rats as a COX-2 inhibitor.Fórmula:C9H8OPureza:98.07%Peso molecular:132.16ICI 63197
CAS:ICI 63197 (2-Amino-6-methyl-4-propyl-[1,2,4]triazolo[1,5-a]pyrimidin-5(4H)-one) is a PDE4 inhibitor.Fórmula:C9H13N5OPureza:99.70%Cor e Forma:White SolidPeso molecular:207.23Pantoprazole sodium
CAS:<p>Pantoprazole sodium is a proton pump inhibitor that irreversibly blocks gastric acid secretion by bonding with H+/K+-ATPase.</p>Fórmula:C16H14F2N3NaO4SPureza:96.92% - 99.81%Cor e Forma:White To Off-White SolidPeso molecular:405.35Laurdan
CAS:<p>Laurdan (6-Dodecanoyl-2-dimethylaminonaphthalene) is a fluorescent membrane probe that is spectrally sensitive to the phospholipid phase of the cell membrane to</p>Fórmula:C24H35NOPureza:98.73% - 99.02%Cor e Forma:SolidPeso molecular:353.54Sofalcone
CAS:<p>Sofalcone (SU-88), a gastric antiulcer agent in clinical use, is known to induce the expression of Heme oxygenase-1 (HO-1) in gastric epithelium.</p>Fórmula:C27H30O6Pureza:97.55%Cor e Forma:SolidPeso molecular:450.52Cephapirin Benzathine
CAS:<p>Cephapirin Benzathine is a semisynthetic, broad-spectrum, first-generation cephalosporin with antibacterial activity.</p>Fórmula:C17H17N3O6S2C16H20N2Pureza:98% - 99.38%Cor e Forma:SolidPeso molecular:543.63Magnesium Lithospermate B
CAS:<p>Magnesium Lithospermate B is a derivative of caffeic acid tetramer. Magnesium Lithospermate B inhibits neuroinflammation and reduces neurodegeneration.</p>Fórmula:C36H28MgO16Pureza:97.5% - 99.87%Cor e Forma:SolidPeso molecular:740.9NVP-BAW2881
CAS:NVP-BAW2881 (BAW2881) is a potent and selective VEGFR inhibitor with activity to inhibit chronic and acute skin inflammation.Fórmula:C22H15F3N4O2Pureza:98.19% - 99.97%Cor e Forma:SolidPeso molecular:424.38AGK2
CAS:<p>AGK2（IC50=3.5 μM） is an effective, and specific SIRT2 inhibitor.</p>Fórmula:C23H13Cl2N3O2Pureza:98.68% - 99.17%Cor e Forma:SolidPeso molecular:434.27Autocamtide-2-related inhibitory peptide
CAS:<p>Autocamtide-2-related inhibitory peptide is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.</p>Fórmula:C64H116N22O19Pureza:>99.99%Cor e Forma:SolidPeso molecular:1497.74GSK-1034702 HCl
CAS:<p>GSK-1034702 HCl is a potent M1 receptor allosteric agonist.</p>Fórmula:C18H25ClFN3O2Cor e Forma:SolidPeso molecular:369.87PS210
CAS:<p>PS210 selectively activates PDK1 (Kd: 3 μM), doesn't affect PDK1 downstream kinases. Prodrug PS423 inhibits PDK1-mediated S6K phosphorylation.</p>Fórmula:C19H15F3O5Pureza:99.78%Cor e Forma:SolidPeso molecular:380.31Jervine
CAS:<p>Jervine inhibits Smoothened, blocking Hedgehog signaling and GLI1 transcription activation.</p>Fórmula:C27H39NO3Pureza:99.20% - 99.86%Cor e Forma:Needles From Methanol + Water SolidPeso molecular:425.6Methyl cellulose
CAS:Methylcellulose is a natural polymer that gels on heating. Methylcellulose is not toxic.Fórmula:C20H38O11Pureza:≥98%Cor e Forma:SolidPeso molecular:454.51（Monomer）Thalidomide-4-OH
CAS:<p>Thalidomide-4-OH, a Thalidomide-derived Cereblon binder, recruits CRBN and serves as a PROTAC linker.</p>Fórmula:C13H10N2O5Pureza:99.59%Cor e Forma:SolidPeso molecular:274.23Eformoterol Hemifumarate
CAS:<p>Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthma</p>Fórmula:C19H24N2O4C4H4O4Pureza:99.86% - >99.99%Cor e Forma:White PowderPeso molecular:402.4RGFP966
CAS:<p>RGFP966 is an HDAC3 inhibitor (IC50: 0.08 μM) and does not affect other HDACs at concentrations up to 15 μM.</p>Fórmula:C21H19FN4OPureza:99.2% - 99.88%Cor e Forma:SolidPeso molecular:362.4γ-Cyclodextrin
CAS:<p>γ-Cyclodextrin (Ringdex C) is a cycloamylose composed of eight alpha-(1->4) linked D-glucopyranose units found in some foods.</p>Fórmula:C48H80O40Pureza:98.56%Cor e Forma:White Solid CrystallinePeso molecular:1297.12Efonidipine
CAS:Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.Fórmula:C34H38N3O7PPureza:98.35% - 99.47%Cor e Forma:SolidPeso molecular:631.66GNE-7915 tosylate
CAS:<p>GNE-7915 tosylate is a potent, selective, and brain-penetrant LRRK2 inhibitor, boasting an IC50 value of 9 nM.</p>Fórmula:C26H29F4N5O6SCor e Forma:SolidPeso molecular:615.6Amifostine thiol dihydrochloride
CAS:Amifostine (WR 1065) activates p53 via JNK and shields tissues from cancer drug toxicity.Fórmula:C5H16Cl2N2SPureza:>99.99%Cor e Forma:SolidPeso molecular:207.165IU1-248
CAS:<p>IU1-248 is a derivative of IU1. IU1-248 is a potent and selective USP14 inhibitor with an IC50 of 0.83 μM[1].</p>Fórmula:C20H23N3O2Pureza:99.3%Cor e Forma:SolidPeso molecular:337.42Pyrocatechuic acid
CAS:<p>Pyrocatechuic acid (Catecholcarboxylic acid), a normal human benzoic acid metabolite found in plasma, has increased levels after aspirin ingestion.</p>Fórmula:C7H6O4Pureza:98.10%Cor e Forma:SolidPeso molecular:154.12H-89 dihydrochloride
CAS:<p>H-89 dihydrochloride (5-Isoquinolinesulfonamide) is a potent inhibitor of protein kinase A (PKA; IC50: 0.14 μM, Ki: 48 nM).</p>Fórmula:C20H20BrN3O2S·2HClPureza:98.22% - >99.99%Cor e Forma:SolidPeso molecular:519.281400W dihydrochloride
CAS:<p>1400W dihydrochloride (N-(3-(Aminomethyl)benzyl)acetamidine) is a highly effective and specific inhibitor of inducible NOS2 (iNOS).</p>Fórmula:C10H17Cl2N3Pureza:98% - 99.94%Cor e Forma:SolidPeso molecular:250.17Nelociguat
CAS:<p>Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.</p>Fórmula:C19H17FN8O2Pureza:99.19%Cor e Forma:SolidPeso molecular:408.39VU0238441
CAS:<p>VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.</p>Fórmula:C16H9ClF3NO2Pureza:100%Cor e Forma:SolidPeso molecular:339.7Indican
CAS:<p>Indican (Indoxyl-β-D-glucoside) is a natural protective compound that is used to protect the liver.</p>Fórmula:C14H17NO6Pureza:99.78% - 99.92%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:295.29BI-6015
CAS:<p>BI 6015 is an antagonist of HNF4α. HNF4α is a nuclear receptor that regulates gene expression in the intestine cells, liver cells, and pancreas-β cells.</p>Fórmula:C15H13N3O4SPureza:99.81%Cor e Forma:SolidPeso molecular:331.35UMI-77
CAS:<p>UMI-77 is a selective Mcl-1 inhibitor. UMI-77 binds to the BH3-binding groove of Mcl-1.Cost-effective and quality-assured.</p>Fórmula:C18H14BrNO5S2Pureza:96% - 99.57%Cor e Forma:SolidPeso molecular:468.34Afimetoran
CAS:<p>Afimetoran (BMS-986256) is a toll-like receptor antagonist. Afimetoran can be used in the research of inflammatory and autoimmune diseases.</p>Fórmula:C26H32N6OPureza:99.81% - 99.94%Cor e Forma:SolidPeso molecular:444.57Thioflavine S
CAS:<p>Thioflavine S (Direct Yellow 7) is a fluorescent histochemical marker.</p>Pureza:98%Cor e Forma:SolidLinocinnamarin
CAS:<p>Linocinnamarin, from strawberries, blocks degranulation by inactivating Syk/PLCgamma.</p>Fórmula:C16H20O8Pureza:99.95%Cor e Forma:SolidPeso molecular:340.33BCI hydrochloride
CAS:<p>BCI hydrochloride ((E)-BCI hydrochloride) is a DUSP6 inhibitor that inhibits RANKL-mediated osteoclastogenesis and attenuates oophorectomy-induced bone loss.</p>Fórmula:C22H24ClNOPureza:99.95%Cor e Forma:SolidPeso molecular:353.89(2S,3R,4S,5R)-2-Amino-3,4,5,6-tetrahydroxyhexanal hydrochloride
CAS:<p>(2S,3R,4S,5R)-2-Amino-3,4,5,6-tetrahydroxyhexanal hydrochloride (D-Mannosamine hydrochloride) is a compound used in the development of mannosylated liposomes.</p>Fórmula:C6H14ClNO5Pureza:99.13% - 99.67%Cor e Forma:Powder To Fine Crystals White/ColorlessPeso molecular:215.63Pyrolin
CAS:<p>Pyrolin has a strong antifungal activity and exerts a potent impact on the ultrastructure of M.fructicola.</p>Fórmula:C7H8O2Pureza:99.38%Cor e Forma:Beige Solid CrystallinePeso molecular:124.14Lophanthoidin E
CAS:<p>Lophanthoidin E is a kind of natural product derived from the herbs of Rabdosia lophanthoides.</p>Fórmula:C22H30O7Pureza:98.00%Cor e Forma:SolidPeso molecular:406.47SSR504734
CAS:<p>SSR504734 is a novel potent glycine transporter 1 (GlyT1) inhibitor.</p>Fórmula:C20H20ClF3N2OCor e Forma:SolidPeso molecular:396.83Esculentoside H
CAS:<p>Phytolaccaceae has anti-tumor activity, the mechanism may be related to the capacity of Esculentoside H for TNF release.</p>Fórmula:C48H76O21Pureza:98.04% - 99.3%Cor e Forma:SolidPeso molecular:989.1Neoeriocitrin
CAS:Neoeriocitrin, from Drynaria Rhizome, boosts MC3T3-E1 growth & bone differentiation; strong AChE inhibitor.Fórmula:C27H32O15Pureza:99.92% - 99.93%Cor e Forma:SolidPeso molecular:596.532-Methylcyclohexanone
CAS:<p>2-Methylcyclohexanone is a human endogenous metabolite.</p>Fórmula:C7H12OPureza:97.16% - 99.60%Cor e Forma:SolidPeso molecular:112.17
