Derivados de Quinazolina e Quinolina
As quinazolinas e quinolinas são compostos heterocíclicos contendo nitrogénio, com estruturas aromáticas que desempenham um papel fundamental na síntese de fármacos com atividade anticancerígena, antimicrobiana e anti-inflamatória. Os seus derivados apresentam modificações estruturais que otimizam a biodisponibilidade e a seletividade, permitindo o desenvolvimento de novos princípios ativos para diversas aplicações terapêuticas. Estes compostos são utilizados na fabricação de APIs para o tratamento do câncer, infeções, doenças neurodegenerativas e cardiovasculares. Além disso, os derivados de quinazolina e quinolina são essenciais na investigação de inibidores enzimáticos e no desenvolvimento de moléculas bioativas inovadoras.
Na CymitQuimica, oferecemos derivados de quinazolina e quinolina de alta pureza para aplicações em síntese química, desenvolvimento farmacêutico e biotecnologia.
Foram encontrados 65630 produtos de "Derivados de Quinazolina e Quinolina"
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4-[(2,3,4-Trimethoxyphenyl)methyl]-1-piperazinecarboxylic acid ethyl ester
CAS:<p>4-[(2,3,4-Trimethoxyphenyl)methyl]-1-piperazinecarboxylic acid ethyl ester is an impurity standard for HPLC. It is a white or off-white solid that is soluble in organic solvents. The compound has been shown to be a metabolite of the drug product, and can also be found as an impurity in the API. 4-[(2,3,4-Trimethoxyphenyl)methyl]-1-piperazinecarboxylic acid ethyl ester can be synthesized from 2,3,4-trimethoxybenzoic acid and 1-(2-chloroethyl)piperazine.</p>Fórmula:C17H26N2O5Pureza:Min. 95%Peso molecular:338.4 g/molLoxoprofen Related Compound 2 - mixture of diastereomers
CAS:<p>Loxoprofen Related Compound 2 is a mixture of diastereomers that is an impurity in the drug product, Loxoprofen. Loxoprofen Related Compound 2 is a metabolite of loxoprofen and its concentration in blood plasma after administration of loxoprofen can be used as an indicator for pharmacokinetics. The compound has been shown to inhibit the activity of bacterial dna gyrase and topoisomerase IV, which are enzymes that maintain the integrity of bacterial DNA. Loxoprofen Related Compound 2 was found to be less active than loxoprofen against MRSA and Clostridium perfringens, although it was more active than loxoprofen against Mycobacterium tuberculosis, Mycobacterium avium complex, and methicillin-resistant Staphylococcus aureus (MRSA).</p>Fórmula:C15H18O4Pureza:Min. 95%Peso molecular:262.3 g/mol3’-Destrifluoromethyl 2’-trifluoromethyl cinacalcet
CAS:<p>3' - Destrifluoromethyl 2' - trifluoromethyl cinacalcet is a metabolite of cinacalcet, which is a drug used for the treatment of secondary hyperparathyroidism. It is an impurity in the drug product and can be identified by HPLC.</p>Fórmula:C22H22F3NPureza:Min. 95%Peso molecular:357.41 g/molMethyl 3-aminocrotonate
CAS:<p>Methyl 3-aminocrotonate is an intermediate in the synthesis of pyridinedicarboxylic acid. It is a white powder with a melting point of 160-165°C and a boiling point of 263°C. Methyl 3-aminocrotonate is soluble in water, alcohols, ethers, chloroform, and benzene. It has been detected by its UV absorption at 227 nm. The detection sensitivity for this compound was found to be 0.1 ppm. This product has shown to produce calcium stearate as an acid conjugate.<br>Methyl 3-aminocrotonate is a molecule that contains a hydrogen bond between the hydroxyl group and the amine group on C3, which are both in close proximity to the carbonyl group on C2. This molecule exhibits intramolecular hydrogen bonding between two hydrogen atoms on different molecules. <br>The IR spectrum for methyl 3-aminoc</p>Fórmula:C5H9NO2Pureza:Min. 95%Cor e Forma:White To Yellow SolidPeso molecular:115.13 g/molMethyl 4-[[1-(ethoxycarbonyl)-2-oxocyclopentyl]methyl]-α-methylbenzeneacetate
CAS:<p>Please enquire for more information about Methyl 4-[[1-(ethoxycarbonyl)-2-oxocyclopentyl]methyl]-α-methylbenzeneacetate including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C19H24O5Pureza:Min. 95%Peso molecular:332.39 g/mol2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperazinyl)ethoxy]ethanol N-oxide
CAS:<p>2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperazinyl)ethoxy]ethanol N-oxide is a peroxide that is used in pharmaceutical preparations as an antioxidant. It is a white solid that is insoluble in water and has a molecular weight of 168.13. 2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperazinyl)ethoxy]ethanol N-oxide has been shown to be effective against the development of cholesterol gallstones and can be used as a prophylactic agent against cardiovascular disease. This compound also inhibits the oxidation of drugs by hydrogen peroxide and other oxidizing agents. 2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperazinyl)eth</p>Fórmula:C21H25N3O3SPureza:Min. 95%Cor e Forma:Tan to pale orange solid.Peso molecular:399.51 g/mol1-[4-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-1-piperazinyl]-2-hydroxy-1-pentanone
CAS:<p>1-[4-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-1-piperazinyl]-2-hydroxy-1-pentanone (DMPP) is an analog of the antiarrhythmic drugs flecainide and propafenone. It has the same effects as these drugs, but with a longer duration of action. DMPP is a racemic mixture of two enantiomers, one of which is active against arrhythmias and the other inactive. The drug binds to the beta subunit of voltage gated potassium channels in cardiac muscle cells, preventing the flow of current through these channels. This results in prolongation of the action potential and suppression of arrhythmias. DMPP also inhibits cellulase activity and may be used as an agent for treatment of bacterial infections caused by methicillin resistant Staphylococcus aureus (MRSA).</p>Fórmula:C19H27N5O4Pureza:Min. 95%Peso molecular:389.45 g/molRisperidone N-oxide
CAS:<p>Risperidone N-oxide is a prodrug of risperidone. It is prepared by reacting risperidone with methanol and hydrogen peroxide in the presence of piperidine, followed by purification using preparative high-performance liquid chromatography. Risperidone N-oxide is a crystalline solid with a melting point of about 190 °C. Risperidone N-oxide has been shown to have antiemetic properties, which may be due to its ability to block dopamine receptors in the brain. The drug also shows some antipsychotic activity, and it has a constant therapeutic effect against schizophrenia. The major impurities found in risperidone N-oxide are hydroxylamine and piperidine.</p>Fórmula:C23H27FN4O3Pureza:Min. 95%Peso molecular:426.48 g/mol4'-[(1,4'-Dimethyl-2'-propyl[2,6'-bi-1H-benzimidazol]-1'-yl)methyl][1,1'-biphenyl]-2-carboxamide
CAS:<p>Imatinib is a drug substance that belongs to the class of imidazole and phenylpiperidine derivatives. It is used in the treatment of leukemia and other cancers. Imatinib has been shown to inhibit tumor cell proliferation by inhibiting protein synthesis via inhibition of ribosomal activity, leading to cell death. Imatinib also inhibits the activation of PPARγ, an important transcription factor involved in lipid metabolism. The presence of impurities may affect the therapeutic efficacy or safety of this drug, so it is important to know what impurities are present in order to avoid unexpected side effects.</p>Fórmula:C33H31N5OPureza:Min. 95%Peso molecular:513.63 g/mol1-[[3-Methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl]methyl]-2-[[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl]methyl]sulfinyl]-1H-b enzimidazole
CAS:<p>1-[[3-Methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl]methyl]-2-[[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl]methyl]sulfinyl]-1H-b enzimidazole is an impurity of a drug product. It is a metabolite that has been shown to be present in human plasma and urine. This compound is synthetically produced and is not found in nature. It has been shown to have niche applications in both analytical chemistry and pharmacopoeia.</p>Fórmula:C25H22F6N4O3SPureza:Min. 95%Peso molecular:572.52 g/mol1,3-bis(1,1-Dimethylpropyl) benzene
CAS:<p>1,3-bis(1,1-Dimethylpropyl) benzene is a synthetic compound that is used in drug product formulation. It is also used as an analytical standard for the determination of 1,3-bis(1,1-dimethylethyl)benzene in drug products and as a natural impurity in API preparations. This compound is metabolized to 1,3-dibromobenzene and 1,2-dibromoethane during its metabolic process. The chemical properties of this compound are similar to those of other alkylbenzenes and it has been shown to have pharmacological effects such as analgesic and antiinflammatory activities.</p>Fórmula:C16H26Pureza:Min. 95%Peso molecular:218.38 g/mol1-[4-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-1-piperazinyl]-5-hydroxy-1-pentanone
CAS:<p>1-[4-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-1-piperazinyl]-5-hydroxy-1-pentanone is a drug product that is used as an HPLC standard. It is a natural metabolite of the drug product 1-[4-(4-Amino-6,7-dimethoxyquinazolinyl)-1piperazinyl]-5hydroxypentane. The synthesis of this compound has been reported in the literature.<br>The impurity content of this compound meets the pharmacopoeia requirements for an analytical reference standard for API impurities.</p>Fórmula:C19H27N5O4Pureza:Min. 95%Peso molecular:389.45 g/mol(R)-1-Phenyl-1,2,3,4-tetrahydroisoquinoline
CAS:<p>(R)-1-Phenyl-1,2,3,4-tetrahydroisoquinoline is a chiral molecule with four stereocenters. It is synthesized by the reaction of sulfamic acid and cyclohexene in the presence of p-toluenesulfonic acid. The product formed is then dehydrogenated to produce (R)-1-phenyl-1,2,3,4-tetrahydroisoquinoline. This compound is soluble in organic solvents such as benzene and ethane and can be used as an acceptor for chiral stationary phases.</p>Fórmula:C15H15NPureza:Min. 95%Cor e Forma:PowderPeso molecular:209.29 g/molN,N-Bis[2-(2-hydroxyethoxy)ethyl] quetiapine chloride
<p>N,N-Bis[2-(2-hydroxyethoxy)ethyl] quetiapine chloride is a synthetic drug product with a purity of >98% and low impurity content, which is used in research and development. It can be custom synthesized to meet the needs of a particular research or development project. This compound has an analytical purity of >98% and low impurity content, making it suitable for use as an API impurity standard. N,N-Bis[2-(2-hydroxyethoxy)ethyl] quetiapine chloride is not currently regulated by any pharmacopoeia.</p>Fórmula:C25H34ClN3O4SPureza:Min. 95%Peso molecular:508.07 g/mol(S)-3-(Dimethylamino)-1-(2-thienyl)propan-1-ol
CAS:<p>(S)-3-(Dimethylamino)-1-(2-thienyl)propan-1-ol is a polymerase chain reaction (PCR) reagent that is used as a building block for the synthesis of five membered ring lactams and dihedral polymers. This compound is synthesized by chemoenzymatic coupling of propanamine with trifluoroacetic acid in the presence of methyl groups, followed by catalytic hydrogenation to yield the desired product. The asymmetric synthesis of this compound was achieved through chiral resolution using NMR spectroscopy.</p>Fórmula:C9H15NOSPureza:Min. 95%Peso molecular:185.29 g/molMirtazapine N-oxide
CAS:<p>Mirtazapine N-oxide is an antidepressant agent that is metabolized to mirtazapine. Mirtazapine N-oxide has been shown to have a linear response in the detection of serotonin in urine samples and has been used for pharmacokinetic studies, optimization, and clinical use. The enantiomer of mirtazapine N-oxide has been shown to be more potent than the racemic mixture. The drug is excreted unchanged into the urine with a half-life of 2 hours. Mirtazapine N-oxide can be detected in plasma for up to 24 hours after oral administration and may accumulate in certain tissues such as liver or kidney. This drug has also been shown to cause death in mice at very high doses.</p>Fórmula:C17H19N3OPureza:Min. 95%Peso molecular:281.35 g/mol2-Methyl-3,4-dimethoxy pyridine hydrochloride
CAS:<p>2-Methyl-3,4-dimethoxy pyridine hydrochloride is an analytical standard that is used as a reference compound in the pharmaceutical industry to identify impurities in drug products. It also has a niche use as an API impurity and HPLC standard. 2-Methyl-3,4-dimethoxy pyridine hydrochloride is used as an intermediate for the synthesis of other drugs, including benzodiazepines and beta blockers. It is also used in research and development for its high purity. This chemical is natural or synthetic in origin but can be custom synthesized to meet specific requirements. 2-Methyl-3,4-dimethoxy pyridine hydrochloride also has CAS number 1210824-88-6.</p>Fórmula:C8H11NO2HClPureza:Min. 95%Peso molecular:189.64 g/mol[6-Hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl](4-hydroxyphenyl)-methanone
CAS:<p>MDM2 inhibitors are a class of cancer drugs that inhibit the activity of MDM2, which is an oncoprotein that prevents the degradation of p53. This inhibition leads to increased levels of p53 and the activation of its tumor-suppressing functions. The anti-cancer activity of this drug has been shown in a number of cancer cells, including human colon cancer cells, human prostate cancer cells, and murine leukemia cells. Furthermore, this drug has been shown to have synergistic effects when combined with other chemotherapeutic agents such as cisplatin and vincristine.</p>Fórmula:C21H14O4SPureza:Min. 95%Peso molecular:362.4 g/molChlorhexidine diacetate EP Impurity O
CAS:<p>Chlorhexidine diacetate EP Impurity O is an analytical reference material that is used as a pharmaceutical impurity. It is a metabolite of chlorhexidine diacetate and has been shown to be present in the urine of patients who are taking chlorhexidine diacetate. Chlorhexidine diacetate EP Impurity O can be used for identification and quantification in HPLC analysis.</p>Fórmula:C22H30Cl2N10Pureza:Min. 95%Peso molecular:505.45 g/molN-Methyl omeprazole (Mixture of isomers with the methylated nitrogens of imidazole)
<p>Please enquire for more information about N-Methyl omeprazole (Mixture of isomers with the methylated nitrogens of imidazole) including the price, delivery time and more detailed product information at the technical inquiry form on this page</p>Fórmula:C18H21N3O3SPureza:Min. 95%Peso molecular:359.44 g/mol2-[3-[4-(3-Chloro-4-ethylphenyl)-1-piperazinyl]propyl]-1,2,4-triazolo[4,3-a]pyridin-3(2H)-one
CAS:<p>2-[3-[4-(3-Chloro-4-ethylphenyl)-1-piperazinyl]propyl]-1,2,4-triazolo[4,3-a]pyridin-3(2H)-one is a research and development impurity standard. Impurities are the substances that are not intentionally added to the drug product but can be generated from the synthesis process or from the raw materials. This substance has been used as a synthetic intermediate in the production of other drugs and as an analytical reference for HPLC analysis. It is used to help develop new drugs by providing data about metabolites and possible toxic effects on humans.</p>Pureza:Min. 95%(2R)-2-(3,4-Dimethoxyphenyl)-5-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-2-isopropylpentanenitrile hydrochloride
CAS:<p>(2R)-2-(3,4-Dimethoxyphenyl)-5-[2-(3,4-dimethoxyphenyl)ethyl-methylamino]-2-isopropylpentanenitrile hydrochloride (ZD4054) is a drug that has been shown to be sensitive to the efflux pump in Escherichia coli. It is also able to inhibit multidrug resistance in nematodes and cross-resistance in humans. ZD4054 inhibits multidrug resistance by inhibiting the efflux of drugs from cells. This prevents the development of resistance to antibiotics and other drugs. The mechanism of action for this drug is unknown, but it may affect chloride channels that are found on the cell membrane. ZD4054 has also been shown to be effective against C.elegans and Drosophila melanogaster, two species commonly used for research purposes.</p>Fórmula:C27H39ClN2O4Pureza:Min. 95%Peso molecular:491.06 g/mol1,4-Bis[(tetrahydro-2-furanyl)carbonyl]-piperazine
CAS:<p>1,4-Bis[(tetrahydro-2-furanyl)carbonyl]-piperazine is a synthetic drug product. It is used as an analytical standard to help elucidate the metabolic pathway of drugs and their metabolites. This compound has been shown to be metabolized by various enzymes including CYP450, glutathione reductase, and esterases. It can also be synthesized from 1,4-dihydropyridine and 2-furancarboxaldehyde. The physical properties of 1,4-bis[(tetrahydro-2-furanyl)carbonyl]-piperazine are: white powder; mp 178°C; IR max 1710 cm−1 (CO); UV max 221 nm (EtOH). The impurities in this product are: 1-(2H)-Quinolinone (CAS No. 2467-94-1) which may have a maximum concentration</p>Fórmula:C14H22N2O4Pureza:Min. 95%Peso molecular:282.34 g/molChloromethyl olanzapinium chloride
CAS:<p>Chloromethyl olanzapinium chloride is an analytical reference material that can be used as a standard for HPLC-UV analysis. It is also used in the development of new drugs and as an impurity standard during drug manufacturing. Chloromethyl olanzapinium chloride has been shown to be a metabolite of Olanzapine, which is a niche drug product that is not commercially available. Chloromethyl olanzapinium chloride is listed by the USP, EP and JP as a drug product impurity. It can be synthesized from natural or synthetic sources.</p>Fórmula:C18H22Cl2N4SPureza:Min. 95%Cor e Forma:PowderPeso molecular:397.37 g/mol4-Methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzamide
CAS:<p>4-Methyl-3-[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzamide is a synthetic compound that has been used as an impurity standard to determine the purity of drugs. It is also used in research and development, drug product, and custom synthesis. 4-Methyl-3-[4-(3-pyridinyl)-2-pyrimidinyl]amino]benzamide has a CAS number of 851137-91-2 and is on the list of pharmacopoeias. This compound is not found in nature, but it can be synthesized in the laboratory. Metabolism studies have been conducted for this drug to identify its metabolites, which can be determined through HPLC analysis.</p>Fórmula:C17H15N5OPureza:Min. 95%Peso molecular:305.33 g/molIndenolol
CAS:<p>Indenolol is a blocker of beta-adrenergic.</p>Fórmula:C15H21NO2Pureza:98%Cor e Forma:SolidPeso molecular:247.33CP 93129 dihydrochloride
CAS:<p>5-HT1B agonist, potent and highly selective</p>Fórmula:C12H14ClN3OPureza:98%Cor e Forma:SolidPeso molecular:251.71Benzatropine
CAS:<p>Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.</p>Fórmula:C21H25NOPureza:98%Cor e Forma:SolidPeso molecular:307.43GW-3333
CAS:<p>GW-3333 inhibits matrix metalloproteinases and TNF-Converting Enzyme, showing potential as an antiarthritic therapy.</p>Fórmula:C22H36N4O4Pureza:98%Cor e Forma:SolidPeso molecular:420.55Isothipendyl
CAS:Isothipendyl is the first generation of H1 antagonists (antihistamines) and anticholinergics and has an effect on itching.Fórmula:C16H19N3SCor e Forma:SolidPeso molecular:285.41Guanfacine
CAS:<p>Guanfacine is a selective agonist of the α2A receptor.</p>Fórmula:C9H9Cl2N3OPureza:98%Cor e Forma:SolidPeso molecular:246.09Blonanserin HCl
CAS:<p>Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.</p>Fórmula:C23H32Cl2FN3Pureza:98%Cor e Forma:SolidPeso molecular:440.42Deterenol Free Base
CAS:<p>Deterenol Free Base is a beta-adrenoceptor agonist.</p>Fórmula:C11H17NO2Cor e Forma:SolidPeso molecular:195.26Nifekalant hydrochloride
CAS:<p>Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.</p>Fórmula:C19H28ClN5O5Pureza:99.91%Cor e Forma:SolidPeso molecular:441.91Rolapitant
CAS:<p>Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.</p>Fórmula:C25H26F6N2O2Pureza:99.86%Cor e Forma:SolidPeso molecular:500.48Protriptyline
CAS:<p>Protriptyline: Antidepressant, AChE inhibitor (IC50 0.06 mM), prevents Aβ aggregation; potential for depression and Alzheimer's.</p>Fórmula:C19H21NCor e Forma:SolidPeso molecular:263.38Arasertaconazole
CAS:<p>Arasertaconazole, a sterol-14-alpha demethylation inhibitor, is used potentially for the treatment of vulvovaginal candcanidiasis.</p>Fórmula:C20H15Cl3N2OSCor e Forma:SolidPeso molecular:437.77(R)-Carvedilol
CAS:<p>(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Fórmula:C24H26N2O4Pureza:98%Cor e Forma:SolidPeso molecular:406.47Chlophedianol Hydrochloride
CAS:<p>Chlophedianol hydrochloride: a cough suppressant for dry cough with antihistamine and local anesthetic traits; possibly anticholinergic at high doses.</p>Fórmula:C17H21Cl2NOPureza:98%Cor e Forma:SolidPeso molecular:326.26BR351 precursor
CAS:<p>BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>Fórmula:C27H32N2O8S2Pureza:98%Cor e Forma:SolidPeso molecular:576.68Enadoline (Free Base)
CAS:<p>Enadoline is a K-opioid agonist with visual and dissociative effects, studied for pain but dropped due to dysphoria.</p>Fórmula:C24H32N2O3Cor e Forma:SolidPeso molecular:396.52Robenidine
CAS:<p>Robenidine, an anticoccidial guanidine, is used as an additive in rabbit fodder.</p>Fórmula:C15H13Cl2N5Pureza:98%Cor e Forma:SolidPeso molecular:334.2Levobetaxolol
CAS:<p>Levobetaxolol (AL-1577A/Betaxon) is a beta-blocker for ocular hypertension and glaucoma.</p>Fórmula:C18H29NO3Pureza:98%Cor e Forma:SolidPeso molecular:307.43Zuclopenthixol decanoate
CAS:<p>Zuclopenthixol decanoate is an anti-schizophrenia drug.</p>Fórmula:C32H43ClN2O2SPureza:98%Cor e Forma:SolidPeso molecular:555.21BP-5-087
CAS:<p>BP-5-087 is a STAT3 inhibitor, combining with BCR-ABL1 inhibition to overcome kinase-independent resistance in chronic myeloid leukemia.</p>Fórmula:C36H30F8N2O6SCor e Forma:SolidPeso molecular:770.69Hexazinone
CAS:<p>Hexazinone: a triazine herbicide blocks photosynthesis by binding to D-1 protein in photosystem II.</p>Fórmula:C12H20N4O2Pureza:99.99%Cor e Forma:SolidPeso molecular:252.31(R,R)-Glycopyrrolate
CAS:<p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>Fórmula:C19H28BrNO3Pureza:98%Cor e Forma:SolidPeso molecular:398.34PPNDS
CAS:<p>P2X1 receptor antagonist</p>Fórmula:C18H15N4NaO14PS2Pureza:98%Cor e Forma:SolidPeso molecular:629.42Gemigliptin Tartrate(911637-19-9 free base)
CAS:<p>Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).</p>Fórmula:C22H25F8N5O8Pureza:>99.99%Cor e Forma:SolidPeso molecular:639.45Carboxyamidotriazole
CAS:<p>Carboxyamidotriazole is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signaling pathways.</p>Fórmula:C17H12Cl3N5O2Pureza:98%Cor e Forma:SolidPeso molecular:424.67Lanicemine
CAS:<p>Lanicemine is a low-trapping NMDA channel blocker. It also has a binding (Ki: 0.56-2.1 μM).</p>Fórmula:C13H14N2Pureza:98%Cor e Forma:SolidPeso molecular:198.26Gallopamil hydrochloride
CAS:<p>Gallopamil hydrochloride (Methoxyverapamil hydrochloride) is an antagonist of phenylalkylamine calcium.</p>Fórmula:C28H41ClN2O5Pureza:99.86%Cor e Forma:SolidPeso molecular:521.09Afacifenacin
CAS:<p>Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.</p>Fórmula:C27H26F3N3O2Pureza:99.83%Cor e Forma:SolidPeso molecular:481.51Cibenzoline
CAS:Cibenzoline: antiarrhythmic, blocks KATP channels, minimizes LVPG, useful in hypertrophic cardiomyopathy studies.Fórmula:C18H18N2Cor e Forma:SolidPeso molecular:262.35Ivabradine
CAS:<p>Ivabradine: oral HCN blocker, lowers heart rate without affecting blood pressure, has anticonvulsant and anti-anginal properties.</p>Fórmula:C27H36N2O5Cor e Forma:SolidPeso molecular:468.59Batimastat sodium salt
CAS:<p>Batimastat (BB-94) sodium salt is a broad-spectrum MMP inhibitor (IC50s: 3, 4, 4, 6, and 20 nM for MMP-1, MMP-2, MMP-9, MMP-7, and MMP-3).</p>Fórmula:C23H31N3NaO4S2Pureza:98%Cor e Forma:SolidPeso molecular:500.63WAY-151693
CAS:<p>WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).</p>Fórmula:C21H22ClN3O5SCor e Forma:SolidPeso molecular:463.93MMP-1-IN-1
<p>MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .</p>Fórmula:C14H17ClN2O3Cor e Forma:SolidPeso molecular:296.75Vasicinone
CAS:<p>Vasicinone may act as a hepatoprotective agent.</p>Fórmula:C11H10N2O2Pureza:98.06%Cor e Forma:SolidPeso molecular:202.21Ivaltinostat
CAS:<p>CG-200745 is a potent inhibitor of HDAC. CG200745 induces apoptosis and also inhibits the deacetylation of histone H3 and tubulin.</p>Fórmula:C24H33N3O4Pureza:98%Cor e Forma:SolidPeso molecular:427.54Palonosetron
CAS:<p>Palonosetron, a 5-HT3 antagonist with Ki of 0.17 nM, is used in the prevention and treatment of chemotherapy-induced nausea and vomiting (CINV).</p>Fórmula:C19H24N2OPureza:98%Cor e Forma:SolidPeso molecular:296.41Safironil
CAS:<p>Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.</p>Fórmula:C15H23N3O4Pureza:99.83%Cor e Forma:SolidPeso molecular:309.36Riodoxol
CAS:<p>Riodoxol is an antiviral agent that effectively affects the reproduction and maturation of viruses.</p>Fórmula:C6H3I3O2Cor e Forma:SolidPeso molecular:487.8Piribedil dihydrochloride
CAS:<p>dopamine agonist</p>Fórmula:C16H20Cl2N4O2Pureza:98%Cor e Forma:SolidPeso molecular:371.26NNGH
CAS:<p>NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.</p>Fórmula:C13H20N2O5SPureza:98.41%Cor e Forma:SolidPeso molecular:316.37Vernakalant
CAS:<p>Vernakalant (RSD-1235) is a mixed ion channel blocker.</p>Fórmula:C20H31NO4Pureza:98%Cor e Forma:SolidPeso molecular:349.46Mizolastine dihydrochloride
CAS:<p>Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).</p>Fórmula:C24H27Cl2FN6OPureza:98%Cor e Forma:SolidPeso molecular:505.42PF-00356231 hydrochloride
CAS:<p>PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.</p>Fórmula:C25H21ClN2O3SPureza:98.39%Cor e Forma:SolidPeso molecular:464.96Rufloxacin hydrochloride
CAS:<p>Rufloxacin HCl (MF-934 HCl): a fluoroquinolone that inhibits topoisomerase and B-cell differentiation.</p>Fórmula:C17H19ClFN3O3SPureza:99.80%Cor e Forma:SolidPeso molecular:399.867Trifluperidol HCl
CAS:Trifluperidol, a dopamine D2-receptor antagonist, is used to treat schizophrenia.Fórmula:C22H24ClF4NO2Cor e Forma:SolidPeso molecular:445.88Thiochrome
CAS:<p>Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.</p>Fórmula:C12H14N4OSPureza:98%Cor e Forma:SolidPeso molecular:262.33Lorbamate
CAS:<p>Carbamate is a type of carbamate that has been studied as a muscle relaxant and sedative.</p>Fórmula:C12H22N2O4Cor e Forma:SolidPeso molecular:258.31Tiropramide
CAS:<p>Tiropramide is an antispasmodic drug. It also useful to inhibit the contractile response of the urinary bladder and in managing abdominal pain in IBS.</p>Fórmula:C28H41N3O3Pureza:98%Cor e Forma:SolidPeso molecular:467.64U 27391
CAS:<p>U 27391 is a metalloproteinase inhibitor. It acts by inhibits the action of human recombinant interleukin-1beta and glycosaminoglycan synthesis.</p>Fórmula:C23H36N4O5Pureza:98%Cor e Forma:SolidPeso molecular:448.56Carisbamate
CAS:<p>CarisbAMate (JNJ-10234094, RWJ 333369, YKP-509) is an antiepileptic drug candidate.</p>Fórmula:C9H10ClNO3Cor e Forma:SolidPeso molecular:215.63Vapendavir
CAS:<p>Vapendavir binds enterovirus capsids; effective against EV71 with EC50 of 0.5-1.4 μM.</p>Fórmula:C21H26N4O3Pureza:98%Cor e Forma:SolidPeso molecular:382.46Vandetanib Fumarate
CAS:<p>Oral tyrosine kinase inhibitor Vandetanib Fumarate targets RET, VEGFRs, EGFR in thyroid cancer.</p>Fórmula:C26H28BrFN4O6Pureza:98%Cor e Forma:SolidPeso molecular:591.43(R)-Afatinib
CAS:<p>(R)-Afatinib: oral ErbB inhibitor (EGFR/HER2), IC50 ≤14 nM. For ESCC, NSCLC, gastric cancer research.</p>Fórmula:C24H25ClFN5O3Cor e Forma:SolidPeso molecular:485.94cis-Tadalafil
CAS:<p>Cis-Tadalafil is a potent inhibitor of phosphodiesterase 5, which is used to treat erectile dysfunction (ED) and primary pulmonary hypertension (PPH). It works by increasing blood flow to the penis, allowing men with ED to achieve and maintain an erection. Cis-Tadalafil is also used to treat symptoms of prostatic hyperplasia (enlarged prostate) in men. This drug has been shown to be effective in treating PPH by reducing pulmonary arterial pressure and improving exercise capacity. Cis-Tadalafil belongs to the carboline class of drugs and is a phosphodiesterase 5 inhibitor that selectively inhibits cGMP-specific phosphodiesterase type 5 (PDE5). This drug has been shown to be highly effective in treating both ED and PPH with minimal side effects.</p>Fórmula:C22H19N3O4Pureza:Min. 95%Cor e Forma:White/Off-White SolidPeso molecular:389.4 g/molBifeprunox
CAS:<p>Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.</p>Fórmula:C24H23N3O2Pureza:98%Cor e Forma:SolidPeso molecular:385.46(R)-Mequitazine
CAS:<p>(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.</p>Fórmula:C20H22N2SCor e Forma:SolidPeso molecular:322.47Alimemazine
CAS:<p>Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.</p>Fórmula:C18H22N2SPureza:98%Cor e Forma:Crystals SolidPeso molecular:298.45Landiolol
CAS:<p>Landiolol is used as a highly cardioselective ultra short-acting beta-blocker.</p>Fórmula:C25H39N3O8Pureza:98%Cor e Forma:White Crystalline PowderPeso molecular:509.59TAPI-1
CAS:<p>TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.</p>Fórmula:C26H37N5O5Pureza:≥95%Cor e Forma:SolidPeso molecular:499.6(S)-Carvedilol
CAS:<p>(S)-Carvedilol is a non-selective β/α-1 blocker.It exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).</p>Fórmula:C24H26N2O4Pureza:98%Cor e Forma:Less Crystalline Solid Colourless Crystalline SolidPeso molecular:406.47WAY 629
CAS:<p>WAY 629 is a selective SR-2C agonist that also act as potent 5-HT2C receptor agonists.</p>Fórmula:C15H18N2Cor e Forma:SolidPeso molecular:226.32Tanomastat
CAS:<p>Tanomastat is an orally bioavailable and non-peptidic biphenyl matrix metalloproteinases inhibitor.</p>Fórmula:C23H19ClO3SPureza:98%Cor e Forma:SolidPeso molecular:410.91(Rac)-Tanomastat
CAS:<p>Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.</p>Fórmula:C23H19ClO3SCor e Forma:SolidPeso molecular:410.91Bornaprine
CAS:<p>Bornaprine is an anticholinergic drug used to treat Parkinson's disease due to inhibition of muscarinic or nicotinic transmission.</p>Fórmula:C21H31NO2Cor e Forma:SolidPeso molecular:329.48(S)-Propafenone
CAS:<p>(S)-Propafenone, or (S)-SA-79, is an S-enantiomer with beta-blocking effects and sodium channel blocking class 1 antiarrhythmic properties.</p>Fórmula:C21H27NO3Pureza:98%Cor e Forma:SolidPeso molecular:341.44Daltroban
CAS:<p>Daltroban (SKF 96148) is a specific thromboxane A2 (TXA2) receptor antagonist.</p>Fórmula:C16H16ClNO4SPureza:99.74%Cor e Forma:SolidPeso molecular:353.82(S)-Azelastine
CAS:<p>(S)-Azelastine is an antihistamine reducing receptors H1R, M1R, M3R, and inhibiting HNEpC cell growth.</p>Fórmula:C22H24ClN3OCor e Forma:SolidPeso molecular:381.9Phenindamine
CAS:<p>Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].</p>Fórmula:C19H19NCor e Forma:SolidPeso molecular:261.36(S)-Pomalidomide
CAS:<p>(S)-Pomalidomide is an inhibitor of angiogenesis and growth of B-cell neoplasias, which induces complete regressions of Burkitt's lymphoma cell tumors.</p>Fórmula:C13H11N3O4Cor e Forma:SolidPeso molecular:273.24(S)-Hydroxychloroquine
CAS:(S)-Hydroxychloroquine is the enantiomer of Hydroxychloroquine. Hydroxychloroquine shows efficiently inhibits SARS-CoV-2 infection in vitro.Fórmula:C18H26ClN3OPureza:98%Cor e Forma:SolidPeso molecular:335.87Medroxalol
CAS:<p>Medroxalol (RMI81968), an oral α- & β-adrenergic blocker, has antihypertensive and vasodilatory effects.</p>Fórmula:C20H24N2O5Cor e Forma:SolidPeso molecular:372.42(R)-Hydroxychloroquine
CAS:<p>(R)-Hydroxychloroquine is the enantiomer of Hydroxychloroquine. Hydroxychloroquine is an agent of synthetic antimalarial.</p>Fórmula:C18H26ClN3OPureza:98%Cor e Forma:SolidPeso molecular:335.87Bifeprunox Mesylate
CAS:<p>Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.</p>Fórmula:C25H27N3O5SPureza:98%Cor e Forma:SolidPeso molecular:481.56Omeprazole Sodium
CAS:<p>Omeprazole Sodium is a proton pump inhibitor(PPI) and suppresses gastric acid secretion.</p>Fórmula:C17H18N3NaO3SPureza:99.84%Cor e Forma:Clear In WaterPeso molecular:367.4ND-322 HCl
CAS:<p>ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.</p>Fórmula:C15H16ClNO3S2Pureza:99.49%Cor e Forma:SolidPeso molecular:357.88
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