Derivados de Quinazolina e Quinolina
As quinazolinas e quinolinas são compostos heterocíclicos contendo nitrogénio, com estruturas aromáticas que desempenham um papel fundamental na síntese de fármacos com atividade anticancerígena, antimicrobiana e anti-inflamatória. Os seus derivados apresentam modificações estruturais que otimizam a biodisponibilidade e a seletividade, permitindo o desenvolvimento de novos princípios ativos para diversas aplicações terapêuticas. Estes compostos são utilizados na fabricação de APIs para o tratamento do câncer, infeções, doenças neurodegenerativas e cardiovasculares. Além disso, os derivados de quinazolina e quinolina são essenciais na investigação de inibidores enzimáticos e no desenvolvimento de moléculas bioativas inovadoras.
Na CymitQuimica, oferecemos derivados de quinazolina e quinolina de alta pureza para aplicações em síntese química, desenvolvimento farmacêutico e biotecnologia.
Foram encontrados 65630 produtos de "Derivados de Quinazolina e Quinolina"
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Pemigatinib
CAS:<p>Pemigatinib (INCB054828) is an orally active, selective inhibitor of FGFR(IC50s of 0.4 nM, 0.5 nM, 1.2 nM, 30 nM for FGFR1, FGFR2, FGFR3, FGFR4, respectively).</p>Fórmula:C24H27F2N5O4Pureza:99.57% - 99.95%Cor e Forma:SolidPeso molecular:487.5Tetrahydrozoline
CAS:<p>Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the study of nasal and conjunctival congestion.</p>Fórmula:C13H16N2Pureza:97.85% - 99.77%Cor e Forma:SolidPeso molecular:200.28Deracoxib
CAS:<p>Deracoxib (SC 46) is a selective COX-2 inhibitor, non-steroidal, non-narcotic anti-inflammatory drug with an IC50 of 70-150 μM for osteosarcoma cells.</p>Fórmula:C17H14F3N3O3SPureza:98.94% - 99.81%Cor e Forma:SolidPeso molecular:397.37Nefopam hydrochloride
CAS:<p>Nefopam hydrochloride (Nefopam HCl) is the hydrochloride salt form of nefopam, a centrally-acting, non-opioid benzoxazocine with analgesic activity.</p>Fórmula:C17H20ClNOPureza:99.32% - 99.85%Cor e Forma:SolidPeso molecular:289.8Trazodone hydrochloride
CAS:<p>Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.</p>Fórmula:C19H23Cl2N5OPureza:99.5% - 99.52%Cor e Forma:SolidPeso molecular:408.33Dasatinib monohydrate
CAS:<p>Dasatinib monohydrate, an oral SRC-kinase inhibitor, counters imatinib-resistant chronic myeloid leukemia.</p>Fórmula:C22H28ClN7O3SPureza:99.68% - >99.99%Cor e Forma:SolidPeso molecular:506.03Ribociclib succinate
CAS:<p>Ribociclib succinate (LEE011 succinate) is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively).</p>Fórmula:C27H36N8O5Pureza:99.9%Cor e Forma:SolidPeso molecular:552.63Mianserin hydrochloride
CAS:<p>Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.</p>Fórmula:C18H21ClN2Pureza:99.63% - 99.82%Cor e Forma:White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedPeso molecular:300.83Lercanidipine
CAS:<p>Lercanidipine (Masnidipine) is a calcium channel blocker of the dihydropyridine class.</p>Fórmula:C36H41N3O6Pureza:99.92%Cor e Forma:White To Light Yellow SolidPeso molecular:611.73Alosetron hydrochloride
CAS:<p>Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.</p>Fórmula:C17H19ClN4OPureza:99.90%Cor e Forma:Off-White PowderPeso molecular:330.813-Aminopropionitrile fumarate (2:1)
CAS:<p>3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) is an organic compound and antirheumatic agent used in veterinary medicine.</p>Fórmula:C4H4O4·2C3H6N2Pureza:99.76% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:256.26Ambroxol
CAS:<p>Ambroxol treats respiratory diseases by thinning mucus. Active in Mucosolvan, it enhances mucus clearance and protects lungs.</p>Fórmula:C13H18Br2N2OPureza:99.72%Cor e Forma:SolidPeso molecular:378.1Sitagliptin
CAS:<p>Sitagliptin (MK0431), an oral DPP-4 inhibitor, treats type 2 diabetes alone or with metformin/thiazolidinedione by increasing incretins and insulin.</p>Fórmula:C16H15F6N5OPureza:99.33% - 99.83%Cor e Forma:Yellow GreasePeso molecular:407.31Chlorhexidine dihydrochloride
CAS:Chlorhexidine dihydrochloride (NSC-185) is a disinfectant and topical anti-infective agent used also as mouthwash to prevent oral plaque.Fórmula:C22H32Cl4N10Pureza:97.51% - 98.32%Cor e Forma:White To Pale Yellow PowderPeso molecular:578.38Tafenoquine Succinate
CAS:<p>Tafenoquine Succinate (WR 238605 (Succinate)) is an 8-aminoquinoline. and is an agent of anti-malarial prophylactic.</p>Fórmula:C28H34F3N3O7Pureza:99.77%Cor e Forma:SolidPeso molecular:581.58Linagliptin
CAS:<p>Linagliptin (BI 1356) is a potent, orally bioavailable dihydropurinedione-based inhibitor of dipeptidyl peptidase 4 (DPP-4), with hypoglycemic activity.</p>Fórmula:C25H28N8O2Pureza:99.15% - >99.99%Cor e Forma:SolidPeso molecular:472.54Ticagrelor
CAS:<p>Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.</p>Fórmula:C23H28F2N6O4SPureza:98.08% - 99.77%Cor e Forma:SolidPeso molecular:522.57Chlorhexidine
CAS:<p>Chlorhexidine is a biguanide antiseptic targeting bacteria, damaging cell membranes and causing cell death, more effective against gram-positive types.</p>Fórmula:C22H30Cl2N10Pureza:98% - 99.85%Cor e Forma:Crystals From Methanol SolidPeso molecular:505.45Venlafaxine hydrochloride
CAS:<p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>Fórmula:C17H28ClNO2Pureza:97.32% - 99.86%Cor e Forma:White Crystalline PowderPeso molecular:313.86Raloxifene hydrochloride
CAS:<p>Raloxifene HCl treats postmenopausal osteoporosis, acts as estrogen on bone/cholesterol, and blocks it in breast/uterus.</p>Fórmula:C28H28ClNO4SPureza:98% - 99.97%Cor e Forma:Light Yellow SolidPeso molecular:510.044Ranitidine Hydrochloride
CAS:<p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>Fórmula:C13H23ClN4O3SPureza:99.30% - 99.49%Cor e Forma:SolidPeso molecular:350.86Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Fórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Cor e Forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53Flubendazole
CAS:<p>Flubendazole (Flumoxane) is available OTC in Europe that is an anthelmintic using to treat worm infection in humans.</p>Fórmula:C16H12FN3O3Pureza:98.47% - 99.30%Cor e Forma:White To Pale Yellow PowderPeso molecular:313.28Nifuratel
CAS:<p>Nifuratel (SAP 113) is a local antiprotozoal and antifungal agent that may also be given orally.</p>Fórmula:C10H11N3O5SPureza:99.76% - 99.87%Cor e Forma:Fresh Yellow Crystalline Or Yellow PowderPeso molecular:285.28Carebastine
CAS:<p>Carebastine, the active metabolite of Ebastine, is an antagonist of the histamine H1 receptor.</p>Fórmula:C32H37NO4Pureza:99.16%Cor e Forma:Off-White SolidPeso molecular:499.64Ramelteon
CAS:<p>Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.</p>Fórmula:C16H21NO2Pureza:97.21% - 99.92%Cor e Forma:Crystalline SolidPeso molecular:259.34Telmisartan
CAS:<p>Telmisartan (BIBR 277) is an Angiotensin 2 Receptor Blocker. The mechanism of action of telmisartan is as an Angiotensin 2 Receptor Antagonist.</p>Fórmula:C33H30N4O2Pureza:99.88% - 99.97%Cor e Forma:White Or Off White Crystalline PowderPeso molecular:514.62Primidone
CAS:<p>Primidone (NCI-C56360) is a potent anticonvulsant agent.</p>Fórmula:C12H14N2O2Pureza:99.91%Cor e Forma:Crystals (Ntp 1992)Peso molecular:218.25BI-1935
CAS:<p>BI-1935 is an inhibitor of soluble epoxide hydrolase (sEH). For diseases related to cardiovascular disease.</p>Fórmula:C24H21F3N6O3Pureza:97.55%Cor e Forma:SolidPeso molecular:498.46Iproniazid Phosphate
CAS:<p>Iproniazid Phosphate is a non-selective, irreversible monoamine oxidase inhibitor (MAOI).</p>Fórmula:C9H13N3O·H3PO4Pureza:99.6% - 99.87%Cor e Forma:SolidPeso molecular:277.21O-Desmethyl gefitinib
CAS:<p>O-Desmethyl gefitinib is an active EGFR inhibitor (IC50: 36 nM), a metabolite of Gefitinib, formed by CYP2D6.</p>Fórmula:C21H22ClFN4O3Pureza:97.17%Cor e Forma:SolidPeso molecular:432.88Benazepril hydrochloride
CAS:<p>Benazepril hydrochloride (CGS 14824A HCl) is an angiotensin-converting enzyme (ACE) inhibitor widely used in the therapy of hypertension.</p>Fórmula:C24H29ClN2O5Pureza:99.68% - ≥95%Cor e Forma:Crystalline SolidPeso molecular:460.95Molidustat
CAS:<p>Molidustat (BAY 85-3934) 是新型HIF-PH 抑制剂，对PHD1(IC50:480 nM)、PHD2(IC50:280 nM)、PHD3(IC50:450 nM)。</p>Fórmula:C13H14N8O2Pureza:98.79%Cor e Forma:SolidPeso molecular:314.3Fosinopril sodium
CAS:<p>Fosinopril sodium: ACE inhibitor prodrug for hypertension, becomes active metabolite fosinoprilat.</p>Fórmula:C30H45NO7P·NaPureza:99.37% - 99.40%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:585.65Hydralazine hydrochloride
CAS:<p>Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.</p>Fórmula:C8H9ClN4Pureza:99.85% - 99.86%Cor e Forma:Yellow Crystals White Crystalline SolidPeso molecular:196.64Deferiprone
CAS:<p>Deferiprone (Deferidone) is an Iron Chelator. The mechanism of action of deferiprone is as an Iron Chelating Activity.</p>Fórmula:C7H9NO2Pureza:99.58% - ≥95%Cor e Forma:White NeedlesPeso molecular:139.15Pipemidic acid
CAS:<p>Pipemidic acid (Acido pipemidico), a new antibacterial agent, inhibits the activity of Pseudomonas aeruginosa.</p>Fórmula:C14H17N5O3Pureza:99.65%Cor e Forma:SolidPeso molecular:303.32Lacidipine
CAS:<p>Lacidipine (SN-305) is a slow-acting, long-duration lipophilic dihydropyridine calcium blocker that prevents reflex tachycardia and lowers blood pressure.</p>Fórmula:C26H33NO6Pureza:99.98%Cor e Forma:White-To-Off-White Crystalline SolidPeso molecular:455.54Nifedipine
CAS:<p>Nifedipine (Procardia) is a dihydropyridine calcium channel blocking agent.</p>Fórmula:C17H18N2O6Pureza:99.39% - 99.49%Cor e Forma:Yellow Crystals Physical Description Odorless Yellow Crystals Or Powder Tasteless (Ntp 1992)Peso molecular:346.33Imiquimod
CAS:<p>Imiquimod (R 837) is an immune response modifier that acts as a toll-like receptor 7 agonist.</p>Fórmula:C14H16N4Pureza:99.62% - >99.99%Cor e Forma:White To Off White Crystalline PowderPeso molecular:240.30Hydroxyzine Pamoate
CAS:<p>Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria and histamine-mediated pruritus.</p>Fórmula:C44H43ClN2O8Pureza:99.49%Cor e Forma:SolidPeso molecular:763.27Irbesartan
CAS:<p>Irbesartan (SR-47436) is an Angiotensin 2 Receptor Blocker. The mechanism of action of irbesartan is as an Angiotensin 2 Receptor Antagonist.</p>Fórmula:C25H28N6OPureza:99.79% - 99.81%Cor e Forma:White Crystalline PowderPeso molecular:428.53Captopril
CAS:<p>Captopril (SA333) is a potent and specific inhibitor of peptidyl-dipeptidase A.</p>Fórmula:C9H15NO3SPureza:98.34% - 99.85%Cor e Forma:White To Off-White Crystalline Powder SolidPeso molecular:217.29Erlotinib hydrochloride
CAS:<p>Erlotinib hydrochloride (NSC 718781) is an EGFR inhibitor (IC50: 2 nM). It is used for the treatment of non-small cell lung cancer.</p>Fórmula:C22H23N3O4·HClPureza:99.78% - 99.85%Cor e Forma:White Or Off-White PowderPeso molecular:429.9Phenylbutazone
CAS:<p>Phenylbutazone, an anti-inflammatory, reduces fever and pain, used for spondylitis and arthritis.</p>Fórmula:C19H20N2O2Pureza:99.70% - 99.93%Cor e Forma:SolidPeso molecular:308.37Dimetridazole
CAS:<p>Dimetridazole (1, 2-Dimethyl-5-nitroimidazole) is a agent that combats protozoan infections. Dimetridazole is a nitroimidazole class drug.</p>Fórmula:C5H7N3O2Pureza:99.88%Cor e Forma:SolidPeso molecular:141.13Ketoconazole
CAS:<p>Ketoconazole (R-41400), a CYP3A4 inhibitor, is an imidazole anti-fungal agent.</p>Fórmula:C26H28Cl2N4O4Pureza:99.53% - 99.62%Cor e Forma:Crystals From 4-Methylpentanone SolidPeso molecular:531.43Haloperidol
CAS:Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function.Fórmula:C21H23ClFNO2Pureza:98.69% - 98.97%Cor e Forma:Crystals SolidPeso molecular:375.86Phenytoin
CAS:<p>Phenytoin: a non-sedative hydantoin, antiepileptic with anticonvulsant effects, stabilizes neurons, prevents seizure spread, and relaxes muscles.</p>Fórmula:C15H12N2O2Pureza:99.95%Cor e Forma:Needles (Alcohol) Tasteless (Ntp 1992)Peso molecular:252.27
