Derivados de Quinazolina e Quinolina
As quinazolinas e quinolinas são compostos heterocíclicos contendo nitrogénio, com estruturas aromáticas que desempenham um papel fundamental na síntese de fármacos com atividade anticancerígena, antimicrobiana e anti-inflamatória. Os seus derivados apresentam modificações estruturais que otimizam a biodisponibilidade e a seletividade, permitindo o desenvolvimento de novos princípios ativos para diversas aplicações terapêuticas. Estes compostos são utilizados na fabricação de APIs para o tratamento do câncer, infeções, doenças neurodegenerativas e cardiovasculares. Além disso, os derivados de quinazolina e quinolina são essenciais na investigação de inibidores enzimáticos e no desenvolvimento de moléculas bioativas inovadoras.
Na CymitQuimica, oferecemos derivados de quinazolina e quinolina de alta pureza para aplicações em síntese química, desenvolvimento farmacêutico e biotecnologia.
Foram encontrados 65630 produtos de "Derivados de Quinazolina e Quinolina"
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Asenapine Maleate
CAS:Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.Fórmula:C21H20ClNO5Pureza:99.28%Cor e Forma:SolidPeso molecular:401.84Febantel
CAS:<p>Febantel is an anthelmintic. It is used for veterinary use on dogs, cats, cattle, sheep, goats, pig, and poultry against roundworms and tapeworms.</p>Fórmula:C20H22N4O6SPureza:99.85%Cor e Forma:White To Off-White PowderPeso molecular:446.48Tadalafil
CAS:Tadalafil (IC-351) is a carboline-based compound with vasodilatory activity.Fórmula:C22H19N3O4Pureza:97.03%Cor e Forma:Off-White Cyrstalline SolidPeso molecular:389.40Deferiprone
CAS:<p>Deferiprone (Deferidone) is an Iron Chelator. The mechanism of action of deferiprone is as an Iron Chelating Activity.</p>Fórmula:C7H9NO2Pureza:99.58% - ≥95%Cor e Forma:White NeedlesPeso molecular:139.15Flutamide
CAS:<p>Flutamide (SCH 13521) is an antiandrogen with about the same potency as cyproterone in rodent and canine species.</p>Fórmula:C11H11F3N2O3Pureza:99.6% - 99.96%Cor e Forma:SolidPeso molecular:276.21Chlorhexidine
CAS:<p>Chlorhexidine is a biguanide antiseptic targeting bacteria, damaging cell membranes and causing cell death, more effective against gram-positive types.</p>Fórmula:C22H30Cl2N10Pureza:98% - 99.85%Cor e Forma:Crystals From Methanol SolidPeso molecular:505.45Clofazimine
CAS:<p>Clofazimine, a phenazine dye, has anti-mycobacterial/inflammatory effects, targeting Mycobacterium leprae and others.</p>Fórmula:C27H22Cl2N4Pureza:98.23% - 99.79%Cor e Forma:SolidPeso molecular:473.4Perhexiline maleate
CAS:<p>Perhexiline maleate is an orally active inhibitor of CPT1 and CPT2 that reduces fatty acid metabolism.</p>Fórmula:C23H39NO4Pureza:99.77% - ≥98%Cor e Forma:SolidPeso molecular:393.56Clomipramine hydrochloride
CAS:<p>Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.</p>Fórmula:C19H23ClN2·HClPureza:99.04% - 99.47%Cor e Forma:White To Slightly Yellow Crystalline PowderPeso molecular:351.31Amiodarone hydrochloride
CAS:<p>Amiodarone HCl: Antianginal, class III antiarrhythmic. Lengthens heart muscle action, slows heart rate, reduces vascular resistance.</p>Fórmula:C25H29I2NO3·HClPureza:99.82% - ≥95%Cor e Forma:White To Cream Crystalline PowderPeso molecular:681.78Mexiletine hydrochloride
CAS:<p>Mexiletine hydrochloride is a lidocaine-like antiarrhythmic (Class IB) and anesthetic, stabilizing heartbeats by inhibiting sodium in cardiac cells.</p>Fórmula:C11H18ClNOPureza:99.88%Cor e Forma:White To Off-White SolidPeso molecular:215.72Doxylamine succinate
CAS:<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Fórmula:C21H28N2O5Pureza:99.61%Cor e Forma:5 1 (Ntp 1992)Peso molecular:388.46Diphenidol hydrochloride
CAS:<p>Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.</p>Fórmula:C21H28ClNOPureza:99.15% - 99.33%Cor e Forma:Crystals Soluble In Methanol WaterPeso molecular:345.91Clonidine hydrochloride
CAS:<p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>Fórmula:C9H10Cl3N3Pureza:99.16% - 99.86%Cor e Forma:SolidPeso molecular:266.55Hydralazine hydrochloride
CAS:<p>Hydralazine hydrochloride, an antihypertensive phthalazine, induces vasodilation and may inhibit tumor DNA methylation.</p>Fórmula:C8H9ClN4Pureza:99.85% - 99.86%Cor e Forma:Yellow Crystals White Crystalline SolidPeso molecular:196.64Afoxolaner
CAS:<p>Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs.</p>Fórmula:C26H17ClF9N3O3Pureza:99.1% - 99.38%Cor e Forma:SolidPeso molecular:625.87Mefloquine hydrochloride
CAS:Mefloquine hydrochloride (Mefloquin hydrochloride) is a quinoline derivative used for the prevention and therapy of P. falciparum malaria.Fórmula:C17H17ClF6N2OPureza:99% - 99.99%Cor e Forma:Off-White To Yellow SolidPeso molecular:414.77Balofloxacin
CAS:<p>Balofloxacin, a quinolone antibiotic, can inhibit the synthesis of bacterial DNA by interfering with the DNA gyrase.</p>Fórmula:C20H24FN3O4Pureza:99.62% - 99.98%Cor e Forma:Crystalline SolidPeso molecular:389.42Nilotinib
CAS:<p>Nilotinib (AMN107) is a Bcr-Abl tyrosine kinase inhibitor. Nilotinib has antitumor activity and may be used in CML. Cost-effective and quality-assured.</p>Fórmula:C28H22F3N7OPureza:99.89% - >99.99%Cor e Forma:Off-White SolidPeso molecular:529.52Olanzapine
CAS:<p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>Fórmula:C17H20N4SPureza:99.86% - ≥95%Cor e Forma:Yellowish Crystalline PowderPeso molecular:312.43Norfloxacin
CAS:<p>Norfloxacin (MK-0366)(Norxacin) is a broad-spectrum antibiotic that is active against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C16H18FN3O3Pureza:98.54% - 99.83%Cor e Forma:White To Light-Yellow Crystalline Powder SolidPeso molecular:319.33Olopatadine hydrochloride
CAS:<p>Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.</p>Fórmula:C21H23NO3·HClPureza:99.62% - 99.64%Cor e Forma:White SolidPeso molecular:373.87Droperidol
CAS:<p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>Fórmula:C22H22FN3O2Pureza:97.16% - 98%Cor e Forma:SolidPeso molecular:379.43Levofloxacin hydrate
CAS:<p>Levofloxacin hydrate (Cravit hydrate) is a third-generation fluoroquinolone antibiotic and optically active L-isomer of ofloxacin with antibacterial activity.</p>Fórmula:C18H20FN3O4H2OPureza:98.26%Cor e Forma:Pale Yellow SolidPeso molecular:370.38Sertraline hydrochloride
CAS:<p>Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.</p>Fórmula:C17H18Cl3NPureza:99.12% - 99.89%Cor e Forma:Solid PowderPeso molecular:342.691Amisulpride
CAS:<p>Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.</p>Fórmula:C17H27N3O4SPureza:99.97%Cor e Forma:White Or Almost White Crystalline PowderPeso molecular:369.48Ritodrine hydrochloride
CAS:<p>Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.</p>Fórmula:C17H21NO3·HClPureza:99% - 99.52%Cor e Forma:SolidPeso molecular:323.82Venlafaxine hydrochloride
CAS:<p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>Fórmula:C17H28ClNO2Pureza:97.32% - 99.86%Cor e Forma:White Crystalline PowderPeso molecular:313.864-Methylamino antipyrine
CAS:<p>4-Methylamino antipyrine, a Metamizole metabolite, is an analgesic and antipyretic with mild anti-inflammatory effects, also inhibits COX.</p>Fórmula:C12H15N3OPureza:99.67%Cor e Forma:SolidPeso molecular:217.27Rebamipide
CAS:<p>Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.</p>Fórmula:C19H15ClN2O4Pureza:99.48% - 99.61%Cor e Forma:White PowderPeso molecular:370.79Ezlopitant
CAS:<p>Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.</p>Fórmula:C31H38N2OPureza:97.49%Cor e Forma:SolidPeso molecular:454.65Bromopride
CAS:<p>Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.</p>Fórmula:C14H22BrN3O2Pureza:99.95%Cor e Forma:SolidPeso molecular:344.25Raloxifene hydrochloride
CAS:<p>Raloxifene HCl treats postmenopausal osteoporosis, acts as estrogen on bone/cholesterol, and blocks it in breast/uterus.</p>Fórmula:C28H28ClNO4SPureza:98% - 99.97%Cor e Forma:Light Yellow SolidPeso molecular:510.044Fluoxetine hydrochloride
CAS:Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.Fórmula:C17H19ClF3NOPureza:99.6% - 99.98%Cor e Forma:White To Off-White Crystalline Solid White To Off-White PowderPeso molecular:345.787Lansoprazole
CAS:<p>Lansoprazole (A-65006) is a 2, 2, 2-trifluoroethoxypyridyl derivative of timoprazole that is used in the therapy of STOMACH ULCERS and ZOLLINGER-ELLISON</p>Fórmula:C16H14F3N3O2SPureza:99.18% - 99.84%Cor e Forma:White Crystalline PowderPeso molecular:369.36Ranitidine Hydrochloride
CAS:<p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>Fórmula:C13H23ClN4O3SPureza:99.30% - 99.49%Cor e Forma:SolidPeso molecular:350.86Pemirolast potassium
CAS:<p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>Fórmula:C10H7KN6OPureza:98.91% - 99.63%Cor e Forma:Crystals From Dimethylformamide Crystalline SolidPeso molecular:266.31Sorafenib
CAS:<p>Sorafenib (Bay 43-9006) is a multikinase inhibitor that inhibits Raf-1, B-Raf, VEGFR2, VEGFR3, VEGFR4, PDGFRβ, FLT3, c-Kit, and others (IC50=6/22/90/15/20/20/57</p>Fórmula:C21H16ClF3N4O3Pureza:98% - 99.89%Cor e Forma:SolidPeso molecular:464.82Amitriptyline hydrochloride
CAS:<p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>Fórmula:C20H24ClNPureza:97% - 99.94%Cor e Forma:Crystals White To Off-White PowderPeso molecular:313.86O-Desmethyl gefitinib
CAS:<p>O-Desmethyl gefitinib is an active EGFR inhibitor (IC50: 36 nM), a metabolite of Gefitinib, formed by CYP2D6.</p>Fórmula:C21H22ClFN4O3Pureza:97.17%Cor e Forma:SolidPeso molecular:432.88Methocarbamol
CAS:<p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>Fórmula:C11H15NO5Pureza:99.96%Cor e Forma:Crystals From Benzene SolidPeso molecular:241.24Tiapride hydrochloride
CAS:<p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>Fórmula:C15H24N2O4S·HClPureza:99.4% - 99.77%Cor e Forma:SolidPeso molecular:364.89Amlexanox
CAS:<p>Amlexanox (AA673) treats ulcers by blocking leukotrienes, histamine, reducing inflammation, pain, and healing time.</p>Fórmula:C16H14N2O4Pureza:99.67% - ≥95%Cor e Forma:White Crystalline SolidPeso molecular:298.29Doxazosin mesylate
CAS:Doxazosin mesylate (UK 33274 mesylate)(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.Fórmula:C24H29N5O8SPureza:99.92%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:547.58Dacarbazine
CAS:<p>Dacarbazine (DTIC-Dome) is an antineoplastic agent. It has significant activity against melanomas.</p>Fórmula:C6H10N6OPureza:99.78% - 99.87%Cor e Forma:Ivory Microcrystaline Substance Physical Description White To Ivory Microcrystals Or Off-White Crystalline Solid (Ntp 1992)Peso molecular:182.18Nadifloxacin
CAS:<p>Nadifloxacin (OPC7251) has been used in trials studying the treatment of Acne Vulgaris.</p>Fórmula:C19H21FN2O4Pureza:99.03% - 99.7%Cor e Forma:Off-White Crystalline SolidPeso molecular:360.38Robenidine hydrochloride
CAS:<p>Robenidine hydrochloride (Robenidine Hydrochoride) is an anticoccidial agent mainly used in poultry.</p>Fórmula:C15H14Cl3N5Pureza:>99.99%Cor e Forma:Off-White SolidPeso molecular:370.66Benztropine mesylate
CAS:<p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>Fórmula:C21H25NO·CH4SO3Pureza:98.41% - 99.96%Cor e Forma:White Crystalline Powder; Odourless Or Almost OdourlessPeso molecular:403.53Dasatinib
CAS:<p>Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive.</p>Fórmula:C22H26ClN7O2SPureza:99.59% - 99.86%Cor e Forma:Pale-Yellow SolidPeso molecular:488.01
