Derivados de Quinazolina e Quinolina
As quinazolinas e quinolinas são compostos heterocíclicos contendo nitrogénio, com estruturas aromáticas que desempenham um papel fundamental na síntese de fármacos com atividade anticancerígena, antimicrobiana e anti-inflamatória. Os seus derivados apresentam modificações estruturais que otimizam a biodisponibilidade e a seletividade, permitindo o desenvolvimento de novos princípios ativos para diversas aplicações terapêuticas. Estes compostos são utilizados na fabricação de APIs para o tratamento do câncer, infeções, doenças neurodegenerativas e cardiovasculares. Além disso, os derivados de quinazolina e quinolina são essenciais na investigação de inibidores enzimáticos e no desenvolvimento de moléculas bioativas inovadoras.
Na CymitQuimica, oferecemos derivados de quinazolina e quinolina de alta pureza para aplicações em síntese química, desenvolvimento farmacêutico e biotecnologia.
Foram encontrados 65630 produtos de "Derivados de Quinazolina e Quinolina"
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Dimetridazole
CAS:<p>Dimetridazole (1, 2-Dimethyl-5-nitroimidazole) is a agent that combats protozoan infections. Dimetridazole is a nitroimidazole class drug.</p>Fórmula:C5H7N3O2Pureza:99.88%Cor e Forma:SolidPeso molecular:141.13Racecadotril
CAS:<p>Racecadotril (Acetorphan) has been investigated for the basic science and treatment of Diarrhea, Acute Diarrhea, and Acute Gastroenteritis.</p>Fórmula:C21H23NO4SPureza:98.86% - 99.66%Cor e Forma:White To Off-White Crystalline PowerPeso molecular:385.48Incyclinide
CAS:<p>Incyclinide (COL-3) is a matrix metalloproteinase (MMP) inhibitor.</p>Fórmula:C19H17NO7Pureza:97.99%Cor e Forma:SolidPeso molecular:371.34Ramatroban
CAS:<p>Ramatroban (BAY u3405) (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.</p>Fórmula:C21H21FN2O4SPureza:98.75% - >99.99%Cor e Forma:Crystalline SolidPeso molecular:416.47Niclosamide
CAS:<p>Niclosamide (Niclocide)(BAY2353) is used to treat most tapeworm infections by inhibiting DNA replication.</p>Fórmula:C13H8Cl2N2O4Pureza:98.47% - 99.1%Cor e Forma:Pale Yellow Crystals SolidPeso molecular:327.12Losartan potassium
CAS:<p>Losartan potassium (DuP-753 potassium) , an Angiotensin II Receptor Blocker, selectively and competitively blocks the binding of angiotensin II to the</p>Fórmula:C22H22ClKN6OPureza:99.9% - >99.99%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:461.01Thioridazine hydrochloride
CAS:Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4Fórmula:C21H27ClN2S2Pureza:99.55% - 99.957%Cor e Forma:White To Off-White SolidPeso molecular:407.04Fluoxetine
CAS:<p>Fluoxetine (LY-110140), a specific serotonin inhibitor, serves as an antidepressant with fewer side-effects.</p>Fórmula:C17H18F3NOPureza:99.07% - 99.28%Cor e Forma:SolidPeso molecular:309.33Rupatadine Fumarate
CAS:<p>Rupatadine Fumarate (Rinialer) (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 uM.</p>Fórmula:C26H26ClN3·C4H4O4Pureza:99.86%Cor e Forma:White Or Almost-White PowderPeso molecular:532.03Chlorpheniramine maleate
CAS:<p>Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.</p>Fórmula:C20H23ClN2O4Pureza:99.64% - 99.98%Cor e Forma:Odorless White Crystalline Solid Or White Powder With A Bitter TastePeso molecular:390.87Bupivacaine hydrochloride
CAS:Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.Fórmula:C18H28N2O·HClPureza:99.89% - 99.9%Cor e Forma:SolidPeso molecular:324.89Tamsulosin hydrochloride
CAS:<p>Tamsulosin hydrochloride (Flomax hydrochloride) is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.</p>Fórmula:C20H29ClN2O5SPureza:95.45% - 99.95%Cor e Forma:White To Off-White SolidPeso molecular:444.97Fluorofenidone
CAS:<p>Fluorofenidone (AKF-PD) slows kidney fibrosis by inhibiting NADPH oxidase/ECM via PI3K/Akt, akin to AMR69 but less toxic with a longer half-life.</p>Fórmula:C12H10FNOPureza:99.85%Cor e Forma:SolidPeso molecular:203.21Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Fórmula:C21H25N3O2SPureza:99.14% - 99.63%Cor e Forma:White To Off-White Crystalline PowderPeso molecular:383.51Acetamide, 2,2-dichloro-N-[(1S,2R)-1-(fluoromethyl)-2-hydroxy-2-[4-(methylsulfonyl)phenyl]ethyl]-
CAS:Fórmula:C12H14Cl2FNO4SPureza:%Cor e Forma:SolidPeso molecular:358.2133Benazepril hydrochloride
CAS:<p>Benazepril hydrochloride (CGS 14824A HCl) is an angiotensin-converting enzyme (ACE) inhibitor widely used in the therapy of hypertension.</p>Fórmula:C24H29ClN2O5Pureza:99.68% - ≥95%Cor e Forma:Crystalline SolidPeso molecular:460.95Phenformin hydrochloride
CAS:<p>Phenformin hydrochloride (Phenformin HCl) is an agent belonging to the biguanide class of antidiabetics with antihyperglycemic activity.</p>Fórmula:C10H16ClN5Pureza:97.11% - 99.80%Cor e Forma:Lactic AcidosisPeso molecular:241.72Nifuratel
CAS:<p>Nifuratel (SAP 113) is a local antiprotozoal and antifungal agent that may also be given orally.</p>Fórmula:C10H11N3O5SPureza:99.76% - 99.87%Cor e Forma:Fresh Yellow Crystalline Or Yellow PowderPeso molecular:285.28Dasatinib
CAS:<p>Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive.</p>Fórmula:C22H26ClN7O2SPureza:99.59% - 99.86%Cor e Forma:Pale-Yellow SolidPeso molecular:488.01Diphenidol hydrochloride
CAS:Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.Fórmula:C21H28ClNOPureza:99.15% - 99.33%Cor e Forma:Crystals Soluble In Methanol WaterPeso molecular:345.91Levamlodipine
CAS:<p>Levamlodipine (S-amlodipine) belongs to the dihydropyridine group of calcium channel blockers.</p>Fórmula:C20H25ClN2O5Pureza:97.21%Cor e Forma:White Crystal PowderPeso molecular:408.88Norfloxacin
CAS:<p>Norfloxacin (MK-0366)(Norxacin) is a broad-spectrum antibiotic that is active against both Gram-positive and Gram-negative bacteria.</p>Fórmula:C16H18FN3O3Pureza:98.54% - 99.83%Cor e Forma:White To Light-Yellow Crystalline Powder SolidPeso molecular:319.33Epalrestat
CAS:<p>Epalrestat (ONO2235), an aldose reductase inhibitor, helps manage diabetic neuropathy symptoms and slows disease progression.</p>Fórmula:C15H13NO3S2Pureza:99.2% - 99.54%Cor e Forma:Deep Red Acicular CrystalPeso molecular:319.4Dipyridamole
CAS:Dipyridamole (Persantin) is a Platelet Aggregation Inhibitor. The physiologic effect of dipyridamole is by means of Decreased Platelet Aggregation.Fórmula:C24H40N8O4Pureza:99.47% - 99.84%Cor e Forma:SolidPeso molecular:504.63Cimetidine
CAS:<p>Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS.</p>Fórmula:C10H16N6SPureza:99.82%Cor e Forma:Crystals Physical Description White Crystals With A Slight Sulfur-Mercaptan Odor (Ntp 1992)Peso molecular:252.34Salmeterol
CAS:<p>Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.</p>Fórmula:C25H37NO4Pureza:99.2% - 99.9%Cor e Forma:SolidPeso molecular:415.57Ticagrelor
CAS:<p>Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.</p>Fórmula:C23H28F2N6O4SPureza:98.08% - 99.77%Cor e Forma:SolidPeso molecular:522.57Olodaterol
CAS:Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptorsFórmula:C21H26N2O5Pureza:98.9%Cor e Forma:SolidPeso molecular:386.45Orbifloxacin
CAS:<p>Orbifloxacin (CP-104354) is a broad-spectrum fluoroquinolone antibiotic.</p>Fórmula:C19H20F3N3O3Pureza:99.46% - 99.58%Cor e Forma:SolidPeso molecular:395.38(R)-Terazosin
CAS:<p>R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 nM, α1d 1.97 nM).</p>Fórmula:C19H25N5O4Pureza:98.87% - 98.96%Cor e Forma:SolidPeso molecular:387.43Clidinium bromide
CAS:<p>Clidinium bromide (Ro 2-3773), a synthetic anticholinergic, treats peptic ulcers and alleviates abdominal cramps and IBS symptoms.</p>Fórmula:C22H26BrNO3Pureza:98.89% - 99.86%Cor e Forma:White Crystalline SolidPeso molecular:432.35DHODH-IN-11
CAS:<p>DHODH-IN-11 is a leflunomide derivative and weak dihydroorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.03.</p>Fórmula:C15H11N3O2Pureza:98.14%Cor e Forma:SolidPeso molecular:265.27Deracoxib
CAS:<p>Deracoxib (SC 46) is a selective COX-2 inhibitor, non-steroidal, non-narcotic anti-inflammatory drug with an IC50 of 70-150 μM for osteosarcoma cells.</p>Fórmula:C17H14F3N3O3SPureza:98.94% - 99.81%Cor e Forma:SolidPeso molecular:397.37Chlorambucil
CAS:Chlorambucil (CB-1348) is an orally-active antineoplastic aromatic nitrogen mustard.Fórmula:C14H19Cl2NO2Pureza:97.37% - 98.45%Cor e Forma:Off-White Slightly Granular Powder Melting Point 65-69°CPeso molecular:304.21Nithiamide
CAS:<p>Nithiamide (CL-5279) is an orally available antiprotozoan agent used in the treatment of vaginal trichomoniasis.</p>Fórmula:C5H5N3O3SPureza:99.85%Cor e Forma:SolidPeso molecular:187.18O-Desmethyl gefitinib
CAS:O-Desmethyl gefitinib is an active EGFR inhibitor (IC50: 36 nM), a metabolite of Gefitinib, formed by CYP2D6.Fórmula:C21H22ClFN4O3Pureza:97.17%Cor e Forma:SolidPeso molecular:432.88Nicorandil
CAS:<p>Nicorandil (SG-75)(Ikorel) acts by relaxing the smooth muscle of the blood vessels, especially those of the venous system.</p>Fórmula:C8H9N3O4Pureza:98.14% - >99.99%Cor e Forma:White Or Off-White PowderPeso molecular:211.17Duloxetine hydrochloride
CAS:<p>Duloxetine hydrochloride is an SNRI used for depression, anxiety, and pain in diabetes and fibromyalgia.</p>Fórmula:C18H20ClNOSPureza:99.93% - >99.99%Cor e Forma:White Or White Crystalline PowderPeso molecular:333.88Azelastine hydrochloride
CAS:<p>Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.</p>Fórmula:C22H24ClN3O·HClPureza:98% - >99.99%Cor e Forma:White Crystalline PowderPeso molecular:418.36Vigabatrin
CAS:<p>Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-</p>Fórmula:C6H11NO2Pureza:99.47% - 99.88%Cor e Forma:SolidPeso molecular:129.16Dapoxetine hydrochloride
CAS:<p>Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature ejaculation.</p>Fórmula:C21H23NO·HClPureza:99.70% - 99.91%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:341.87Phenoxybenzamine hydrochloride
CAS:<p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>Fórmula:C18H23Cl2NOPureza:98.04% - >99.99%Cor e Forma:Antihypertensive DrugPeso molecular:340.3Ethionamide
CAS:Ethionamide: antibacterial used to treat TB; may block mycolic acid synthesis, disrupting bacterial walls. Its effect varies with concentration and organism.Fórmula:C8H10N2SPureza:99.45% - 99.92%Cor e Forma:Yellow Crystals From Ethanol Odor (Ntp 1992)Peso molecular:166.24Ethambutol dihydrochloride
CAS:Ethambutol dihydrochloride (CL40881) is a bacteriostatic antimycobacterial agent, which obstructs the formation of cell wall by inhibiting arabinosylFórmula:C10H26Cl2N2O2Pureza:98% - 99.95%Cor e Forma:Crystals White PowderPeso molecular:277.24Azelnidipine
CAS:<p>Azelnidipine (UR-12592) is a dihydropyridine used as calcium channel blocker.</p>Fórmula:C33H34N4O6Pureza:99.78%Cor e Forma:Light Yellowish PowderPeso molecular:582.65Tropisetron hydrochloride
CAS:<p>Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.</p>Fórmula:C17H21ClN2O2Pureza:99.72% - 99.83%Cor e Forma:SolidPeso molecular:320.82Meclofenamic acid sodium
CAS:<p>Meclofenamic acid sodium (Movens), a non-steroidal anti-inflammatory agent, has properties of antipyretic and antigranulation activities.</p>Fórmula:C14H10Cl2NNaO2Pureza:98% - 98.96%Cor e Forma:SolidPeso molecular:318.14Pyrantel pamoate
CAS:<p>Pyrantel pamoate (Pyrantel embonate) is a depolarizing neuromuscular blocking agent.</p>Fórmula:C34H30N2O6SPureza:99.71%Peso molecular:594.69Salbutamol
CAS:<p>Salbutamol (Albuterol) 是短效的 β2 肾上腺素受体激动剂，用于哮喘和慢性阻塞性肺疾病(COPD) 引发的支气管痉挛的研究。</p>Fórmula:C13H21NO3Pureza:91.59% - 99.9%Cor e Forma:White To Off-White Crystalline Solid SolidPeso molecular:239.31Zomepirac sodium salt
CAS:<p>Zomepirac sodium salt (McN-2783-21-98) is a prostaglandin synthetase inhibitor.</p>Fórmula:C15H13ClNNaO3Pureza:98.65% - ≥95%Cor e Forma:SolidPeso molecular:313.71
