Moduladores enzimáticos
Moduladores de enzimas são compostos que podem aumentar ou inibir a atividade de enzimas, regulando assim a taxa de reações bioquímicas. Esses moduladores desempenham um papel crucial no controle de vias metabólicas, sinalização celular e vários processos fisiológicos. Os moduladores de enzimas são amplamente utilizados em pesquisa e desenvolvimento de medicamentos para estudar as funções enzimáticas e desenvolver agentes terapêuticos. Na CymitQuimica, oferecemos uma ampla gama de moduladores de enzimas de alta qualidade para apoiar sua pesquisa em regulação enzimática e descoberta de medicamentos.
Subcategorias de "Moduladores enzimáticos"
Foram encontrados 693 produtos de "Moduladores enzimáticos"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Camostat mesylate - Bio-X ™
CAS:Camostat is a serine protease inhibitor that is used for the treatment of chronic pancreatitis. This drug has shown to reduce inflammation and pain. Studies have shown that Camostat has also inhibited the entry of SARS-CoV-2 in lung cells by inhibiting the priming process of S-protein, necessary for the viral entry into host cells.Fórmula:C20H22N4O5•CH4O3SPureza:Min. 95%Cor e Forma:PowderPeso molecular:494.52 g/molTivozanib
CAS:Inhibitor of VEGF receptorsFórmula:C22H19ClN4O5Pureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:454.86 g/molGefitinib - Bio-X ™
CAS:Gefitinib is an inhibitor of the epidermal growth factor receptor (EGFR) protein. This inhibition is on the EGFR tyrosine kinase domain, where Gefitinib bindings to the ATP-binding site. As a a tyrosine kinase inhibitor, Gefitinib blocks tumor growth and has led to its use in slowing the progression of non-small cell lung cancer. Gefitinib also inhibits invasion and metastasis through inhibition of macrophage receptor interacting protein kinase 2 (RIPK2), rather than EGFR.Fórmula:C22H24ClFN4O3Pureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:446.9 g/molPentoxifylline
CAS:Produto ControladoPhosphodiesterase inhibitorFórmula:C13H18N4O3Pureza:Min. 95%Cor e Forma:White PowderPeso molecular:278.31 g/molO6-Benzylguanine - Bio-X ™
CAS:O6-Benzylguanine is a guanine analog that is an antineoplastic agent. It works by acting as a suicide inhibitor of the enzyme O6-alkylguanine-DNA alkyltransferase. This results to an interruption of DNA repair so that damage can occur to local tumor targets.Fórmula:C12H11N5OPureza:Min. 95%Cor e Forma:PowderPeso molecular:241.25 g/mol3-(4-Phenylbutyl)-4-propyloxetan-2-one
CAS:Cis/trans-form of GK 563 [2351820-19-2]Fórmula:C16H22O2Pureza:Min. 95%Cor e Forma:SolidPeso molecular:246.34 g/molTrilostane
CAS:Produto ControladoInhibitor of 3β-hydroxysteroid dehydrogenase in steroid biosynthesis
Fórmula:C20H27NO3Pureza:Min. 95%Cor e Forma:White PowderPeso molecular:329.43 g/molMK 4827
CAS:Inhibitor of PARP1 and PARP2 enzymes
Fórmula:C19H20N4OPureza:Min. 96 Area-%Cor e Forma:White PowderPeso molecular:320.39 g/molRucaparib camsylate
CAS:Inhibitor of poly (ADP-ribose) polymerase enzyme; antineoplasticFórmula:C19H18FN3O•C10H16O4SPureza:Min. 95%Cor e Forma:Off-White To Yellow SolidPeso molecular:555.66 g/molAbiraterone acetate - Bio-X ™
CAS:Produto ControladoAbiraterone is an antiandrogen drug used in the treatment of metastatic prostate cancer. It is a derivative of steroidal progesterone. This drug inhibits the enzyme CYP17 irreversibly, thus inhibiting the synthesis of androgen. It specifically inhibits the conversion of 17-hydroxyprognenolone to dehydroepiandrosterone to decrease serum levels of testosterone and other androgens.Fórmula:C26H33NO2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:391.55 g/molEtoposide phosphate
CAS:Topoisomerase II inhibitor; chemotherapeutic drugFórmula:C29H33O16PPureza:Min. 95%Cor e Forma:PowderPeso molecular:668.54 g/molDiacerein - Bio-X ™
CAS:Diacerein is a slow-onset anthraquinone IL-1 inhibitor that is used in the treatment of joint diseases such as osteoarthritis. This drug is also being studied for the treatment of insulin resistance and diabetes mellitus. Diacerein works to decrease inflammation and cartilage destruction by reducing the level of interleukin-1.Fórmula:C19H12O8Pureza:Min. 95%Cor e Forma:PowderPeso molecular:368.29 g/molFlurbiprofen
CAS:Inhibitor of cytochrome P450; inhibitor of prostaglandin synthesis
Fórmula:C15H13FO2Pureza:Min. 98 Area-%Cor e Forma:PowderPeso molecular:244.26 g/molImiquimod - Bio-X ™
CAS:Imiquimod is a toll-like receptor 7 agonist drug that is used for the treatment of genital warts, basal cell carcinoma and condyloma acuminata. This drug works by relieving and controlling wart production. Studies in mice have shown that this drug may induce cytokines such as interleukins. Imiquimod helps to increase apoptosis of diseased tissues and an infiltration of lymphocytes into tumor lesions.Fórmula:C14H16N4Pureza:Min. 95%Cor e Forma:PowderPeso molecular:240.3 g/molBrivanib alaninate
CAS:VEGFR2 a tyrosine kinase receptor inhibitor; antineoplasticFórmula:C22H24FN5O4Pureza:Min. 95%Cor e Forma:PowderPeso molecular:441.18123Lenalidomide - Bio-X ™
CAS:Produto ControladoLenalidomide is a thalidomide derivative that is used to treat multiple myeloma and anemia. This drug exerts immunomodulatory effects by altering cytokine production. Lenalidomide also directly inhibits the cullin ring E3 ubiquitin ligase complex.Fórmula:C13H13N3O3Pureza:Min. 95%Cor e Forma:PowderPeso molecular:259.26 g/molLeflunomide - Bio-X ™
CAS:Produto ControladoLeflunomide is a pyrimidine synthesis inhibitor drug that is used to treat rheumatoid arthritis. Although its mechanism of action is not fully determined, this drug has shown to interfere with cell cycle progression by inhibiting dihydroorotate dehydrogenase and has shown antiproliferative activity. As a result of this, it interferes with the expansion of activated autoimmune lymphocytes. Additionally, Leflunomide is a tyrosine kinase inhibitor.Fórmula:C12H9F3N2O2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:270.21 g/molSU 0268
CAS:Inhibitor of 8-oxoguanine DNA glycosylase OGG1 with IC50 of 0.059 μM and excellent specificity over other DNA repair enzymes. OGG1 and its substrate 8-oxoguanine are involved in mutagenesis, genotoxicity, inflammation and cancer. The compound can cause accumulation of 8-oxoguanine in DNA in vitro and is a potent tool for the study of OGG1 biology.Fórmula:C26H25N3O4SPureza:Min. 95%Cor e Forma:White PowderPeso molecular:475.56 g/molGboxin
CAS:Inhibitor of oxidative phosphorylation which acts on the F0F1 ATP synthase in the inner mitochondrial membrane and causes acute increase in mitochondrial membrane potential. Gboxin was shown to accumulate in mitochondria of cancer cells, to cause cellular toxicity and cell growth inhibition in mouse glioblastoma. However, Gboxin did not inhibit growth of mouse embryonic fibroblasts or neonatal astrocytes.Fórmula:C22H33N2O2•ClPureza:Min. 95%Cor e Forma:SolidPeso molecular:392.96 g/molMLN120B
CAS:Inhibitor of IKKβ serine kinaseFórmula:C19H15ClN4O2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:366.8 g/mol
