Moduladores enzimáticos
Moduladores de enzimas são compostos que podem aumentar ou inibir a atividade de enzimas, regulando assim a taxa de reações bioquímicas. Esses moduladores desempenham um papel crucial no controle de vias metabólicas, sinalização celular e vários processos fisiológicos. Os moduladores de enzimas são amplamente utilizados em pesquisa e desenvolvimento de medicamentos para estudar as funções enzimáticas e desenvolver agentes terapêuticos. Na CymitQuimica, oferecemos uma ampla gama de moduladores de enzimas de alta qualidade para apoiar sua pesquisa em regulação enzimática e descoberta de medicamentos.
Subcategorias de "Moduladores enzimáticos"
Foram encontrados 693 produtos de "Moduladores enzimáticos"
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Mirodenafil dihydrochloride - Bio-X ™
CAS:<p>This product is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready-to-use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.</p>Fórmula:C26H37N5O5S•(HCl)2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:604.59 g/molDarapladib - Bio-X ™
CAS:<p>This product is part of our Bio-X ™ Range. These products are aimed at life science researchers who need high quality ready-to-use products for assay development, screening or other R&D work. With a solubility datasheet and convenient vials, all of our Bio-X ™ products are in stock across our global warehouses for rapid delivery and ease of use.</p>Fórmula:C36H38F4N4O2SPureza:Min. 95%Cor e Forma:PowderPeso molecular:666.77 g/molFlavoxate HCl - Bio-X ™
CAS:<p>Flavoxate is a muscarinic antagonist and spasmolytic drug that is used for the relief of conditions associatied with a lack of muscle control in the bladder such as urine urgency. This drug acts as a direct antagonist on acetylcholine receptors. This action reduces the tonus of smooth muscles in the bladder.</p>Fórmula:C24H25NO4•HClPureza:Min. 95%Cor e Forma:PowderPeso molecular:427.92 g/molAG 490
CAS:<p>A tyrosine kinase inhibitor with potent activity against EGFR, STAT3, JAK3/STAT, JAK3/AP-1 and JAK3/MAPK. Suppresses IL-2 signaling pathway, inhibits T-cell growth and activation of JAK3, AP-1, STAT, MAPK. Has anti-proliferative and anti-invasive effect on cancer cells.</p>Fórmula:C17H14N2O3Pureza:Min. 95%Cor e Forma:Yellow PowderPeso molecular:294.3 g/molGabexate mesylate
CAS:<p>Serine protease inhibitor</p>Fórmula:C17H27N3O7SPureza:Min. 95%Peso molecular:417.15697SB 61211 hydrochloride
CAS:<p>Nociceptin/orphanin FQ peptide receptor antagonist</p>Fórmula:C24H29Cl2NO·HClPureza:Min. 95%Peso molecular:454.86 g/molBML 257
CAS:<p>Inhibits Akt translocation by targeting the pleckstrin homology (PH) domain. Inhibits hepatitis C virus NS5B RNA-dependent RNA polymerase (IC50 = 79 µM). Attenuates cannabinoid agonist-mediated proliferation of neural stem/precursor cells.</p>Fórmula:C21H14N2O2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:326.35 g/molRegorafenib
CAS:<p>Multi-kinase inhibitor; inhibits epoxide hydrolase; antineoplastic</p>Fórmula:C21H15ClF4N4O3Pureza:Min. 95%Cor e Forma:White PowderPeso molecular:482.82 g/molSU 3327
CAS:<p>SU 3327, originally introduced as a thiadiazole JNK inhibitor (De et al. 2009) has recently been identified as having antibiotic activity against a broad range of bacteria including drug-resistant gram positive and negative strains (Strokes et al. 2020). This molecule has been given the fictional name ‘Halicin’ inspired by the AI approach used to discover its novel biological activity.</p>Fórmula:C5H3N5O2S3Pureza:Min. 95%Cor e Forma:PowderPeso molecular:261.31 g/molZofenopril calcium
CAS:<p>Angiotensin-converting enzyme inhibitor; antioxidant</p>Fórmula:C44H46N2O8S4•CaPureza:Min. 95%Cor e Forma:PowderPeso molecular:899.17 g/molMG 132
CAS:<p>MG 132 is a modified tripeptide that acts as proteasomal inhibitor. In 2006, MG 132 has been experimentally tested in in vitro cell-based and in vivo models for to assess its use in the medical treatment of Parkinson's disease.</p>Fórmula:C26H41N3O5Pureza:Min. 95%Cor e Forma:PowderPeso molecular:475.304621-NM-PP1
CAS:<p>1-NM-PP1, also known as 1NM-PP1, is an inhibitor of the Src kinase. Studies have shown that 1-NM-PP1 inhibits analog-sensitive kinases (as-kinases) characterised by a small amino acid as gatekeeper of the ATP binding site. Tested to prevent parasitic infections, 1-NM-PP1 inhibited the Toxoplasma gondii life cycle when used at a higher concentration than 500 nM.</p>Fórmula:C20H21N5Pureza:Min. 95%Cor e Forma:PowderPeso molecular:331.1797SB 271046 hydrochloride
CAS:<p>5-HT6 serotonin receptor antagonist; anti-convulsant</p>Fórmula:C20H22CIN3O3S2·HClPureza:Min. 95%Peso molecular:591.91 g/molTiludronic acid disodium
CAS:<p>Farnesyltransferase inhibitor</p>Fórmula:C7H9ClO6P2S•Na2Pureza:Min. 95%Cor e Forma:PowderPeso molecular:364.59 g/molApatinib
CAS:<p>Apatinib, also known as rivoceranib, is an inhibitor of the vascular endothelial growth factor receptor 2 (VEGFR2) tyrosine kinase. Apatinib targets VEGFR2 with its action and has proven to have strong anti-tumor effects in human cancers. In studies in mice, apatinib acted as an Inhibitor of VEGFR2 and played an antiangiogenic effect. Apatinib has been suggested for the treatment of ischemia-induced proliferative retinopathy and neovascular age-related macular degeneration.</p>Fórmula:C24H23N5OPureza:Min. 95%Cor e Forma:PowderPeso molecular:397.47 g/molPitofenone hydrochloride
CAS:<p>Inhibits acetylcholinesterase (AChE); antispasmodic agent</p>Fórmula:C22H25NO4·ClHPureza:Min. 95%Peso molecular:403.9 g/molA 922500
CAS:<p>Inhibits human and mouse diacylglycerol O-acyltransferase 1 (DGAT-1) with IC50 values of 9 and 22 nM, respectively. Selective for DGAT-1 over DGAT-2 (IC50 = 53 µM), acyl coenzyme A transferase (IC50 = 296 µM) and other acyltransferases. Reduces plasma and liver triglycerides, FFA, chylomicron secretion and increases HDL cholesterol in vivo.</p>Fórmula:C26H24N2O4Pureza:Min. 95%Peso molecular:428.48 g/molStaurosporine
CAS:Produto Controlado<p>Inhibitor of protein kinases; induces apoptosis; anti-cancer</p>Fórmula:C28H26N4O3Pureza:Min. 98 Area-%Cor e Forma:Off-White PowderPeso molecular:466.53 g/molTolrestat
CAS:<p>Aldose reductase AKR1B10 inhibitor; hepatotoxic</p>Fórmula:C16H14F3NO3SPureza:Min. 95%Peso molecular:357.35 g/molCyclosporin B
CAS:<p>Cyclosporin B is an antifungal and immunosuppressive cyclic peptide, which is derived from the fungus *Tolypocladium inflatum*. The compound is a member of the cyclosporin family, characterized by cyclic polypeptides with a unique arrangement of amino acids that enable its biological activity. Though its precise mode of action is not completely delineated, it is observed to influence cell growth and viability by potentially disrupting cellular communication or signal transduction pathways.</p>Fórmula:C61H109N11O12Pureza:Min. 95%Cor e Forma:PowderPeso molecular:1,188.59 g/mol
