Histamine H3 antagonist-1, identified by its CAS number 1000392-25-5, is a chemical compound that functions primarily as an antagonist of the histamine H3 receptor. This receptor is involved in various physiological processes, including the regulation of neurotransmitter release in the central nervous system. As an H3 antagonist, this compound may enhance the release of histamine and other neurotransmitters, potentially leading to increased alertness and cognitive function. The compound's structure typically includes features that allow it to effectively bind to the H3 receptor, blocking its activity. This can have implications in treating conditions such as sleep disorders, cognitive deficits, and certain neurodegenerative diseases. Additionally, histamine H3 antagonists are being explored for their potential in managing obesity and metabolic disorders due to their influence on appetite regulation. Overall, the pharmacological profile of Histamine H3 antagonist-1 suggests it may have therapeutic applications, although further research is necessary to fully understand its efficacy and safety in clinical settings.

Histamine H3 antagonist-1

1000392-25-5: Histamine H3 antagonist-1, identified by its CAS number 1000392-25-5, is a chemical compound that functions primarily as an antagonist of the histamine H3 receptor. This receptor is involved in various physiological processes, including the regulation of neurotransmitter release in the central nervous system. As an H3 antagonist, this compound may enhance the release of histamine and other neurotransmitters, potentially leading to increased alertness and cognitive function. The compound's structure typically includes features that allow it to effectively bind to the H3 receptor, blocking its activity. This can have implications in treating conditions such as sleep disorders, cognitive deficits, and certain neurodegenerative diseases. Additionally, histamine H3 antagonists are being explored for their potential in managing obesity and metabolic disorders due to their influence on appetite regulation. Overall, the pharmacological profile of Histamine H3 antagonist-1 suggests it may have therapeutic applications, although further research is necessary to fully understand its efficacy and safety in clinical settings.

<p>Compound 10o, a histamine H3 antagonist-1, functions as both a histamine H3 antagonist and a serotonin reuptake inhibitor, making it useful for research in depression [1].</p>

CAS 1000392-25-5

Histamine H3 antagonist-1

Histamine H3 antagonist-1

Ref: TM-T86579