CAS 100938-10-1

AMASTATIN HYDROCHLORIDE

Description:

Amastatin hydrochloride is a synthetic compound primarily known for its role as a potent inhibitor of aminopeptidases, particularly in the context of biochemical research and potential therapeutic applications. It is characterized by its ability to selectively inhibit the activity of these enzymes, which are involved in protein metabolism and processing. The compound is typically presented as a hydrochloride salt, enhancing its solubility in aqueous solutions, which is advantageous for laboratory use. Amastatin hydrochloride is often utilized in studies related to peptide synthesis, enzyme kinetics, and the modulation of various biological pathways. Its structural features include a specific arrangement of functional groups that contribute to its inhibitory activity. As with many chemical substances, safety precautions should be observed when handling Amastatin hydrochloride, as it may pose risks if ingested or improperly managed. Overall, its unique properties make it a valuable tool in biochemical research, particularly in the study of proteolytic enzymes and their roles in cellular processes.

Formula: C₂₁H₃₉ClN₄O₈

InChI: InChI=1/C21H38N4O8.ClH/c1-9(2)7-12(22)17(28)20(31)25-16(11(5)6)19(30)24-15(10(3)4)18(29)23-13(21(32)33)8-14(26)27;/h9-13,15-17,28H,7-8,22H2,1-6H3,(H,23,29)(H,24,30)(H,25,31)(H,26,27)(H,32,33);1H/t12-,13+,15+,16+,17+;/m1./s1

Synonyms:

• H-(2S,3R)-Ahmh-Val-Val-Asp-Oh Hcl
• [(2S,3R)-3-Amino-2-Hydroxy-5-Methylhexanoyl]-Val-Val-Asp Hydrochloride
• (2S,3R)-[3-Amino-2-Hydroxy-5-Methylhexanoyl]-Val-Val-Asp-Oh Hcl
• Amastatin
• Amastatin Hcl
• Amastatin Hydrochloride Hydrate
• N((2S 3R)3-Amino-2-Hxy-5-Me.Hexanoyl)-L&
• N-[(2S,3R)-3-amino-2-hydroxy-5-methylhexanoyl]-L-valyl-L-valyl-L-aspartic acid hydrochloride (1:1)

Amastatin · HCl

CAS: 100938-10-1

Amastatin has originally been isolated from the culture filtrate of Streptomyces sp. ME98-M3 and is a competitive inhibitor of human serum aminopeptidase A (Ki = 1.1 · 10⁻⁶ M) and of pig kidney leucine aminopeptidase (Ki = 1.6 · 10⁻⁶ M).

Formula: C₂₁H₃₈N₄O₈·HCl

Purity: 96.3%

Color and Shape: White Powder

Molecular weight: 511.02

Ref: 01-4025800

L-Aspartic acid, N-[(2S,3R)-3-amino-2-hydroxy-5-methyl-1-oxohexyl]-L-valyl-L-valyl-, monohydrochloride (9CI)

CAS: 100938-10-1

Formula: C₂₁H₃₉ClN₄O₈

Color and Shape: Solid

Molecular weight: 511.0094

Ref: IN-DA00039N

Amastatin hydrochloride

CAS: 100938-10-1

Amastatin hydrochloride

Formula: C₂₁H₃₈N₄O₈·ClH

Purity: By hplc: >99% (Typical Value in Batch COA)

Color and Shape: white powder

Molecular weight: 511.00935g/mol

Ref: 54-BIMI1803

Amastatin hydrochloride

CAS: 100938-10-1

Amastatin HCl is an inhibitor of aminopeptidase. It also induces vasoconstriction.

Formula: C₂₁H₃₉ClN₄O₈

Color and Shape: White To Off-White Powder

Molecular weight: 511.01

Ref: TM-T19665

Amastatin hydrochloride

CAS: 100938-10-1

Formula: C₂₁H₃₈N₄O₈·HCl·xH₂O

Purity: ≥ 97%

Color and Shape: White or almost white powder

Molecular weight: 511.01 (anhydrous)

Ref: 7W-GA1330

Amastatin Hydrochloride

Controlled Product

CAS: 100938-10-1

Formula: C₂₁H₃₉ClN₄O₈

Color and Shape: Neat

Molecular weight: 622.77

Ref: TR-A575950