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CAS 101975-10-4

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Zardaverine

Description:
Zardaverine, with the CAS number 101975-10-4, is a chemical compound that has been studied primarily for its potential therapeutic applications. It is classified as a selective phosphodiesterase (PDE) inhibitor, specifically targeting PDE4, which plays a crucial role in the regulation of intracellular signaling pathways involving cyclic adenosine monophosphate (cAMP). By inhibiting this enzyme, Zardaverine can enhance cAMP levels, leading to various physiological effects, including anti-inflammatory and bronchodilator activities. This makes it of interest in the treatment of respiratory conditions such as asthma and chronic obstructive pulmonary disease (COPD). Zardaverine is also noted for its ability to modulate smooth muscle relaxation and has been investigated for its potential in cardiovascular applications. Its chemical structure features a unique arrangement of functional groups that contribute to its biological activity. As with many pharmacological agents, the safety profile, pharmacokinetics, and specific therapeutic uses are subjects of ongoing research to fully understand its efficacy and potential side effects.
Formula:C12H10F2N2O3
InChI:InChI=1S/C12H10F2N2O3/c1-18-10-6-7(2-4-9(10)19-12(13)14)8-3-5-11(17)16-15-8/h2-6,12H,1H3,(H,16,17)
InChI key:InChIKey=HJMQDJPMQIHLPB-UHFFFAOYSA-N
SMILES:O(C)C=1C=C(C=CC1OC(F)F)C=2C=CC(=O)NN2
Synonyms:
  • 3(2H)-Pyridazinone, 6-[4-(difluoromethoxy)-3-methoxyphenyl]-
  • 6-(4-(Difluoromethoxy)-3-methoxyphenyl)-3(2H)-pyridazinone
  • 6-[4-(difluoromethoxy)-3-methoxyphenyl]pyridazin-3(2H)-one
  • Unii-Tq358Gwh6Y
  • Zardaverina
  • Zardaverina [INN-Spanish]
  • Zardaverine [INN]
  • Zardaverinum
  • Zardaverinum [INN-Latin]
  • Zardaverine
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