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CAS 103255-66-9

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Pazinaclone

Description:
Pazinaclone is a chemical compound classified as a benzodiazepine derivative, primarily known for its anxiolytic and sedative properties. It acts on the central nervous system by enhancing the effects of the neurotransmitter gamma-aminobutyric acid (GABA) at the GABA-A receptor, leading to increased inhibitory neurotransmission. This mechanism contributes to its potential use in treating anxiety disorders and sleep disturbances. Pazinaclone is characterized by its relatively rapid onset of action and a shorter duration of effects compared to some other benzodiazepines, which may reduce the risk of dependence. The compound is typically administered in oral form and has been studied for its pharmacokinetic properties, including absorption, distribution, metabolism, and excretion. As with other benzodiazepines, potential side effects may include drowsiness, dizziness, and cognitive impairment. Due to its pharmacological profile, pazinaclone is subject to regulatory controls in many countries, reflecting the need for careful management in clinical use.
Formula:C25H23ClN4O4
InChI:InChI=1S/C25H23ClN4O4/c26-20-7-5-16-6-8-21(28-23(16)27-20)30-19(17-3-1-2-4-18(17)24(30)32)15-22(31)29-11-9-25(10-12-29)33-13-14-34-25/h1-8,19H,9-15H2
InChI key:InChIKey=DPGKFACWOCLTCA-UHFFFAOYSA-N
SMILES:C(C(=O)N1CCC2(CC1)OCCO2)C3N(C(=O)C=4C3=CC=CC4)C5=NC6=C(C=C5)C=CC(Cl)=N6
Synonyms:
  • (±)-2-(7-Chloro-1,8-naphthyridin-2-yl)-3-[(1,4-dioxa-8-azaspiro[4.5]dec-8-yl)carbonylmethyl]isoindolin-1-one
  • (±)-8-[[2-(7-Chloro-1,8-naphthyridin-2-yl)-3-oxo-1-isoindolinyl]acetyl]-1,4-dioxa-8-azaspiro[4.5]decane
  • 1,4-Dioxa-8-azaspiro[4.5]decane, 8-[[2-(7-chloro-1,8-naphthyridin-2-yl)-2,3-dihydro-3-oxo-1H-isoindol-1-yl]acetyl]-
  • 103255-66-9
  • 1H-Isoindol-1-one, 2-(7-chloro-1,8-naphthyridin-2-yl)-3-[2-(1,4-dioxa-8-azaspiro[4.5]dec-8-yl)-2-oxoethyl]-2,3-dihydro-
  • 2-(7-Chloro-1,8-naphthyridin-2-yl)-3-[2-(1,4-dioxa-8-azaspiro[4.5]dec-8-yl)-2-oxoethyl]isoindolin-1-one
  • 2-(7-chloro-1,8-naphthyridin-2-yl)-3-[2-(1,4-dioxa-8-azaspiro[4.5]dec-8-yl)-2-oxoethyl]-2,3-dihydro-1H-isoindol-1-one
  • 8-[[2-(7-Chloro-1,8-naphthyridin-2-yl)-2,3-dihydro-3-oxo-1H-isoindol-1-yl]acetyl]-1,4-dioxa-8-azaspiro[4.5]decane
  • A 77000
  • Dn 2327
  • Pazinaclone
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