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CAS 103614-28-4

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dynorphin A ethylamide (1-9), MeTyr(1)-MeArg(7)-Leu(8)-

Description:
Dynorphin A ethylamide (1-9), specifically the variant MeTyr(1)-MeArg(7)-Leu(8)-, is a synthetic peptide derived from the dynorphin family, which are endogenous opioid peptides. This compound is characterized by its structure, which includes modifications such as the methylation of the tyrosine and arginine residues, enhancing its stability and receptor affinity. Dynorphins primarily interact with the kappa-opioid receptors in the central nervous system, influencing pain modulation, stress response, and various neurophysiological processes. The ethylamide modification contributes to its bioavailability and potential therapeutic applications. As a research chemical, it is often studied for its effects on pain relief, mood regulation, and its role in addiction and neurodegenerative diseases. The specific sequence and modifications of this peptide can significantly affect its pharmacological properties, making it a subject of interest in neuropharmacology and peptide research. However, detailed studies are necessary to fully elucidate its mechanisms of action and potential clinical applications.
Formula:C56H93N19O10
InChI:InChI=1/C56H93N19O10/c1-8-75(56(62)63)26-14-18-38(47(57)79)70-49(81)42(28-34(4)5)73-52(84)44(19-13-25-66-55(60)61)74(7)53(85)39(17-12-24-65-54(58)59)71-50(82)41(27-33(2)3)72-51(83)43(30-35-15-10-9-11-16-35)69-46(78)32-67-45(77)31-68-48(80)40(64-6)29-36-20-22-37(76)23-21-36/h9-11,15-16,20-23,33-34,38-44,64,76H,8,12-14,17-19,24-32H2,1-7H3,(H2,57,79)(H3,62,63)(H,67,77)(H,68,80)(H,69,78)(H,70,81)(H,71,82)(H,72,83)(H,73,84)(H4,58,59,65)(H4,60,61,66)/t38-,39-,40-,41-,42+,43-,44-/m0/s1
Synonyms:
  • L-Argininamide, N-methyl-L-tyrosylglycylglycyl-L-phenylalanyl-L-leucyl-L-arginyl-N2-methyl-L-arginyl-D-leucyl-N-ethyl-
  • N-methyl-L-tyrosylglycylglycyl-L-phenylalanyl-L-leucyl-N~5~-(diaminomethylidene)-L-ornithyl-N~5~-(diaminomethylidene)-N~2~-methyl-L-ornithyl-D-leucyl-N~5~-carbamimidoyl-N~5~-ethyl-L-ornithinamide
  • 1-Metyr-7-mearg-8-leu-dynorphin (1-9)-nhet
  • Daeatal
  • Dynorphin A ethylamide (1-9), metyr(1)-mearg(7)-leu(8)-
  • Dynorphin A ethylamide (1-9), methyltyrosyl(1)-methylarginyl(7)-leucine(8)-
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Found 1 products.
  • Daeatal
    Targetmol
    + Info

    Daeatal

    CAS:
    <p>Dynorphin A ethylamide (1-9), the opioid activities were examined in the bioassays.</p>
    Formula:C56H93N19O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1192.46

    Ref: TM-T23963