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CAS 106266-09-5

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Desfluororisperidone

Description:
Desfluororisperidone is a chemical compound that serves as an active metabolite of risperidone, an atypical antipsychotic medication. It is characterized by its structural modifications that enhance its pharmacological properties. The compound is known for its affinity for various neurotransmitter receptors, particularly dopamine D2 and serotonin 5-HT2A receptors, which contribute to its antipsychotic effects. Desfluororisperidone exhibits a relatively high lipophilicity, influencing its distribution and bioavailability in biological systems. Its pharmacokinetic profile indicates a significant half-life, allowing for sustained therapeutic effects. Additionally, the compound is subject to metabolic processes in the liver, primarily through cytochrome P450 enzymes. Safety and efficacy profiles are evaluated in clinical settings, with attention to potential side effects, including metabolic syndrome and extrapyramidal symptoms. Overall, desfluororisperidone plays a crucial role in the pharmacological landscape of treating schizophrenia and other mood disorders, reflecting the importance of its chemical characteristics in therapeutic applications.
Formula:C23H28N4O2
InChI:InChI=1S/C23H28N4O2/c1-16-18(23(28)27-12-5-4-8-21(27)24-16)11-15-26-13-9-17(10-14-26)22-19-6-2-3-7-20(19)29-25-22/h2-3,6-7,17H,4-5,8-15H2,1H3
InChI key:InChIKey=PLOGUXWMVNJOPF-UHFFFAOYSA-N
SMILES:C(CC=1C(=O)N2C(=NC1C)CCCC2)N3CCC(C=4C=5C(ON4)=CC=CC5)CC3
Synonyms:
  • 3-[2-[4-(1,2-Benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
  • 1,2-Benzisoxazole, 4H-pyrido[1,2-a]pyrimidin-4-one deriv.
  • 4H-Pyrido[1,2-a]pyrimidin-4-one, 3-[2-[4-(1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-
  • Desfluororisperidone
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