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CAS 108687-08-7

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Teludipine

Description:
Teludipine is a chemical compound classified as a calcium channel blocker, primarily used in the treatment of hypertension and certain cardiovascular conditions. It functions by inhibiting the influx of calcium ions through L-type calcium channels in vascular smooth muscle and cardiac tissues, leading to vasodilation and reduced blood pressure. Teludipine is characterized by its selective action, which minimizes side effects commonly associated with non-selective calcium channel blockers. The compound has a specific molecular structure that contributes to its pharmacological properties, including its solubility and bioavailability. It is typically administered orally and has a moderate half-life, allowing for once-daily dosing in clinical settings. As with many medications, potential side effects may include dizziness, headache, and peripheral edema, although these are generally manageable. Overall, Teludipine represents a valuable option in the therapeutic management of hypertension, contributing to improved cardiovascular health outcomes.
Formula:C28H38N2O6
InChI:InChI=1/C28H38N2O6/c1-9-34-26(32)23-18(3)29-21(17-30(7)8)25(27(33)35-10-2)24(23)20-14-12-11-13-19(20)15-16-22(31)36-28(4,5)6/h11-16,24,29H,9-10,17H2,1-8H3/b16-15+
Synonyms:
  • Teludipine [INN:BAN]
  • Diethyl (E)-2-((dimethylamino)methyl)-4-(2-(3-(1,1-dimethylethoxy)-3-oxo-1-propenyl)phenyl)-1,4-dihydro-6-methyl-3,5-pyridinedicarboxylate
  • Teludipino
  • Teludipino [INN-Spanish]
  • Teludipinum
  • Teludipinum [INN-Latin]
  • Unii-Z9Oj72Bm3O
  • 3,5-Pyridinedicarboxylic acid, 2-((dimethylamino)methyl)-4-(2-(3-(1,1-dimethylethoxy)-3-oxo-1-propenyl)phenyl)-1,4-dihydro-6-methyl-, diethyl ester, (E)-
  • diethyl 4-{2-[(1E)-3-tert-butoxy-3-oxoprop-1-en-1-yl]phenyl}-2-[(dimethylamino)methyl]-6-methyl-1,4-dihydropyridine-3,5-dicarboxylate
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Found 1 products.
  • Teludipine
    TRC
    + Info

    Teludipine

    Controlled Product
    CAS:
    <p>Applications A new lipophilic calcium channel blocker; a new dihydropyridine derivative, on cell lines displaying the multidrug resistant phenotype.<br>References Tolomeo M., et al.: Haematologica, 79, 328 (1994),<br></p>
    Formula:C28H38N2O6
    Color and Shape:Neat
    Molecular weight:498.61

    Ref: TR-T017100

    5mg
    298.00€
    50mg
    1,918.00€