CAS 113-92-8

Chlorpheniramine maleate

Description:

Chlorpheniramine maleate is an antihistamine commonly used to relieve allergy symptoms such as runny nose, sneezing, and itching. It is a salt formed from chlorpheniramine, a first-generation antihistamine, and maleic acid. This compound is characterized by its ability to cross the blood-brain barrier, which can lead to sedative effects, a common trait of first-generation antihistamines. Chlorpheniramine maleate exhibits anticholinergic properties, which can result in side effects such as dry mouth, dizziness, and drowsiness. It is typically administered orally and is available in various formulations, including tablets and syrups. The substance is soluble in water and has a relatively stable shelf life when stored properly. Due to its sedative effects, caution is advised when operating machinery or driving after consumption. As with any medication, it is important to follow dosage recommendations and consult healthcare professionals regarding potential interactions with other drugs or underlying health conditions.

Formula: C₁₆H₁₉ClN₂·C₄H₄O₄

InChI: InChI=1S/C16H19ClN2.C4H4O4/c1-19(2)12-10-15(16-5-3-4-11-18-16)13-6-8-14(17)9-7-13;5-3(6)1-2-4(7)8/h3-9,11,15H,10,12H2,1-2H3;1-2H,(H,5,6)(H,7,8)/b;2-1-

InChI key: InChIKey=DBAKFASWICGISY-BTJKTKAUSA-N

SMILES: C(CCN(C)C)(C1=CC=C(Cl)C=C1)C2=CC=CC=N2.C(=C\C(O)=O)\C(O)=O

Synonyms:

• (.+-.)-Chlorpheniramine maleate
• 1-Parachlorophenyl-1-(2-pyridyl)-3-dimethylaminopropane maleate
• 1-p-Chlorophenyl-1-(2-pyridyl)-3-dimethylaminopropane maleate
• 2-Pyridinepropanamine, γ-(4-chlorophenyl)-N,N-dimethyl-, (Z)-2-butenedioate (1:1)
• 2-[P-Chloro-Α-[2-(Dimethylamino)Ethyl]Benzyl]Pyridine Maleate (1:1)
• Allergin
• Allergisan
• Anallerge 4
• Antagonate
• C-Meton
• Calimal
• Carbinoxamide maleate
• Chlor-Trimeton
• Chlor-Tripolon
• Chlorophenamine
• Chloroprophenpyridamine maleate
• Chlorphenamine
• Chlorphenamine Hydrogen Maleate
• Chlorphenamine maleate
• Chlorphenaminhydrogenmaleat
• Chlorprophenpyridamine maleate
• Cloropiril
• Hidrogenomaleato De Clorfenamina
• Histadur
• Histadur dura-tabs
• Histamil
• Histaspan
• Hydrogenomaleate de chlorphenamine
• Ibioton
• Iramine
• Lorphen
• Neorestamin
• Niramine
• Pirafene
• Piriex
• Piriton
• Puermin
• Pyridamal 100
• Pyridine, 2-[p-chloro-α-[2-(dimethylamino)ethyl]benzyl]-, maleate (1:1)
• Synistamin
• Teldrin
• dl-Chlorpheniramine maleate
• but-2-enedioic acid
• Chloropheniramine maleate
• 3-(4-chlorophenyl)-N,N-dimethyl-3-pyridin-2-ylpropan-1-amine (2E)-but-2-enedioate
• 3-(4-chlorophenyl)-N,N-dimethyl-3-(2-pyridyl)propan-1-amine
• 2-Pyridinepropanamine, γ-(4-chlorophenyl)-N,N-dimethyl-, (2Z)-2-butenedioate (1:1)
• (3R)-3-(4-chlorophenyl)-N,N-dimethyl-3-pyridin-2-ylpropan-1-amine (2Z)-but-2-enedioate
• 3-(4-chlorophenyl)-N,N-dimethyl-3-pyridin-2-ylpropan-1-amine (2Z)-but-2-enedioate

Chlorpheniramine Maleate Salt

Controlled Product

CAS: 113-92-8

Applications Antihistaminic.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Roth, F.E., et al.: J. Pharmacol. Exp. Ther., 124, 347 (1958), Smith, R.B., et al.: Toxicol. Appl. Pharmacol., 28, 240 (1974), Eckhart, C.G., et al.: Anal. Profiles Drug Subs., 7, 43 (1978)

Formula: C₁₆H₁₉ClN₂·C₄H₄O₄

Color and Shape: Neat

Molecular weight: 390.86

Ref: TR-C424300

Chlorpheniramine-d4 Maleate Salt

Controlled Product

CAS: 113-92-8

Applications Chlorpheniramine-d4 Maleate Salt is the labeled analogue of Chlorpheniramine Maleate Salt (C424300), an antihistaminic.
References Roth, F.E., et al.: J. Pharmacol. Exp. Ther., 124, 347 (1958); Smith, R.B., et al.: Toxicol. Appl. Pharmacol., 28, 240 (1974); Eckhart, C.G., et al.: Anal. Profiles Drug Subs., 7, 43 (1978)

Formula: C₂₀H₁₉D₄ClN₂O₄

Color and Shape: Neat

Molecular weight: 394.89

Ref: TR-C424304

Chlorpheniramine maleate

CAS: 113-92-8

Histamine (H1) antagonist; used to treat allergies

Formula: C₁₆H₁₉ClN₂•C₄H₄O₄

Purity: Min. 95%

Color and Shape: White Powder

Molecular weight: 390.86 g/mol

Ref: 3D-FC15474