CAS 114298-18-9

Zalospirone

Description:

Zalospirone is a chemical compound that belongs to the class of azapirones, which are known for their anxiolytic properties. It is primarily characterized by its ability to interact with serotonin receptors, particularly the 5-HT1A receptor, which plays a significant role in mood regulation and anxiety. The compound has been studied for its potential therapeutic effects in treating anxiety disorders and depression, exhibiting a favorable side effect profile compared to traditional anxiolytics. Zalospirone is typically administered in oral form and has a moderate bioavailability. Its pharmacokinetics suggest a relatively short half-life, necessitating multiple doses for sustained effects. The compound's safety and efficacy have been evaluated in clinical trials, although it may not be widely available in all regions. As with any pharmacological agent, the potential for side effects exists, and its use should be monitored by healthcare professionals. Overall, zalospirone represents a promising avenue in the development of anxiolytic medications, contributing to the ongoing research in mental health therapeutics.

Formula: C₂₄H₂₉N₅O₂

InChI: InChI=1/C24H29N5O2/c30-22-20-18-6-7-19(17-5-4-16(17)18)21(20)23(31)29(22)11-2-1-10-27-12-14-28(15-13-27)24-25-8-3-9-26-24/h3-9,16-21H,1-2,10-15H2/t16-,17+,18-,19+,20-,21+

InChI key: InChIKey=AERLHOTUXIJQFV-RCPZPFRWNA-N

SMILES: O=C1[C@]2([C@]([C@@]3([C@@]4([C@]([C@]2(C=C3)[H])(C=C4)[H])[H])[H])(C(=O)N1CCCCN5CCN(CC5)C=6N=CC=CN6)[H])[H]

Synonyms:

• 4,7-Etheno-1H-cyclobut[f]isoindole-1,3(2H)-dione, 3a,4,4a,6a,7,7a-hexahydro-2-[4-[4-(2-pyrimidinyl)-1-piperazinyl]butyl]-, (3aα,4β,4aα,6aα,7β,7aα)-
• Zalospirone
• 4,7-Etheno-1H-cyclobut[f]isoindole-1,3(2H)-dione, 3a,4,4a,6a,7,7a-hexahydro-2-[4-[4-(2-pyrimidinyl)-1-piperazinyl]butyl]-, (3aR,4R,4aR,6aS,7S,7aS)-rel-
• Wy 47846
• rel-(3aR,4R,4aR,6aS,7S,7aS)-3a,4,4a,6a,7,7a-Hexahydro-2-[4-[4-(2-pyrimidinyl)-1-piperazinyl]butyl]-4,7-etheno-1H-cyclobut[f]isoindole-1,3(2H)-dione

Zalospirone

CAS: 114298-18-9

Zalospirone

Purity: ≥98%

Molecular weight: 419.52g/mol

Ref: 54-BUP08253

Zalospirone

CAS: 114298-18-9

Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.

Formula: C₂₄H₂₉N₅O₂

Purity: 98.24% - 99.82%

Color and Shape: Solid

Molecular weight: 419.52

Ref: TM-T68172