CAS 115344-47-3

Siguazodan

Description:

Siguazodan, with the CAS number 115344-47-3, is a chemical compound that belongs to the class of benzodiazepines. It is primarily recognized for its pharmacological properties, particularly as a potential anxiolytic and antidepressant agent. The compound exhibits a unique mechanism of action, influencing neurotransmitter systems in the brain, which may contribute to its therapeutic effects. Siguazodan is characterized by its ability to modulate GABAergic activity, enhancing the inhibitory effects of gamma-aminobutyric acid (GABA), a key neurotransmitter involved in regulating neuronal excitability. Additionally, it may possess neuroprotective properties, making it a subject of interest in research related to neurodegenerative diseases. The compound's solubility, stability, and bioavailability are important factors that influence its efficacy and safety profile. As with many pharmacological agents, understanding its pharmacokinetics and potential side effects is crucial for its application in clinical settings. Further studies are necessary to fully elucidate its therapeutic potential and mechanisms of action.

Formula: C₁₄H₁₆N₆O

InChI: InChI=1S/C14H16N6O/c1-9-7-12(21)19-20-13(9)10-3-5-11(6-4-10)18-14(16-2)17-8-15/h3-6,9H,7H2,1-2H3,(H,19,21)(H2,16,17,18)

InChI key: InChIKey=NUHPODZZKHQQET-UHFFFAOYSA-N

SMILES: CC1C(C2=CC=C(N=C(NC#N)NC)C=C2)=NNC(=O)C1

Synonyms:

• 1-Cyano-2-Methyl-3-[4-(4-Methyl-6-Oxo-1,4,5,6-Tetrahydropyridazin-3-Yl)Phenyl]Guanidine
• Guanidine, N-cyano-N′-methyl-N′′-[4-(1,4,5,6-tetrahydro-4-methyl-6-oxo-3-pyridazinyl)phenyl]-
• N-Cyano-N'-Methyl-N'-[4-(1,4,5,6-Tetrahydro-4-Methyl-6-Oxo-3-Pyridazinyl)Phenyl]Guanidine
• N-Cyano-Nmethyl-N��-[4-(1,4,5,6-tetrahydro-4-methyl-6-oxo-3-pyridazinyl)phenyl]guanidine
• Siguazodan (SKF 94836)
• Siguazodan, N-Cyano-Nμ-methyl-N-[4-(1,4,5,6-tetrahydro-4-methyl-6-oxo-3-pyridazinyl)phenyl]guanidine
• Sk And F-94836
• Skf 94836
• Siguazodan

Guanidine, N-cyano-N'-methyl-N''-[4-(1,4,5,6-tetrahydro-4-methyl-6-oxo-3-pyridazinyl)phenyl]-

CAS: 115344-47-3

Formula: C₁₄H₁₆N₆O

Purity: 95%

Color and Shape: Solid

Molecular weight: 284.3164

Ref: IN-DA000GMB

Siguazodan

CAS: 115344-47-3

Siguazodan

Purity: ≥98%

Molecular weight: 284.32g/mol

Ref: 54-BUP15258

Siguazodan

CAS: 115344-47-3

Siguazodan (SKF 94836) is an effective, selective, orally active phosphodiesterase III ((PDE-III)) inhibitor with an IC50 of 117 nM.

Formula: C₁₄H₁₆N₆O

Purity: 99.62% - 99.87%

Color and Shape: Solid

Molecular weight: 284.32

Ref: TM-T12913