CAS 1166-34-3

Cinanserin

Description:

Cinanserin, with the CAS number 1166-34-3, is a chemical compound primarily recognized for its pharmacological properties. It is classified as a serotonin antagonist and has been studied for its potential applications in treating various psychiatric disorders. The compound exhibits a complex structure that includes a piperazine moiety, which is common in many psychoactive substances. Cinanserin is known to interact with serotonin receptors, particularly the 5-HT2 subtype, influencing neurotransmitter activity in the brain. This interaction can lead to effects such as anxiolytic and antipsychotic properties. Additionally, cinanserin has been investigated for its potential use in managing conditions like anxiety and depression. Its pharmacokinetics, including absorption, distribution, metabolism, and excretion, are essential for understanding its therapeutic efficacy and safety profile. While cinanserin has shown promise in clinical studies, its use may be limited by side effects and the availability of alternative treatments. Overall, cinanserin represents an interesting compound in the field of psychopharmacology, warranting further research to fully elucidate its mechanisms and therapeutic potential.

Formula: C₂₀H₂₄N₂OS

InChI: InChI=1S/C20H24N2OS/c1-22(2)15-8-16-24-19-12-7-6-11-18(19)21-20(23)14-13-17-9-4-3-5-10-17/h3-7,9-14H,8,15-16H2,1-2H3,(H,21,23)

InChI key: InChIKey=RSUVYMGADVXGOU-UHFFFAOYSA-N

SMILES: S(CCCN(C)C)C1=C(NC(C=CC2=CC=CC=C2)=O)C=CC=C1

Synonyms:

• (2E)-N-(2-{[3-(dimethylamino)propyl]sulfanyl}phenyl)-3-phenylprop-2-enamide
• (2E)-N-(2-{[3-(dimethylamino)propyl]sulfanyl}phenyl)-3-phenylprop-2-enamide hydrochloride
• 2'-((3-Dimethylaminopropyl)thio)cinnamanilide
• 2-Propenamide, N-(2-((3-(dimethylamino)propyl)thio)phenyl)-3-phenyl-
• 2′-[[3-(Dimethylamino)propyl]thio]cinnamanilide
• Cinanserin [INN]
• Cinanserina
• Cinanserina [INN-Spanish]
• Cinanserine
• Cinanserine [INN-French]
• Cinanserinum
• Cinanserinum [INN-Latin]
• Cinnamanilide, 2′-[[3-(dimethylamino)propyl]thio]-
• N-[2-[[3-(Dimethylamino)propyl]thio]phenyl]-3-phenyl-2-propenamide
• Unii-Ki6J9Oy7A3
• Cinanserin

N-(2-((3-(Dimethylamino)propyl)thio)phenyl)-3-phenylacrylamide

CAS: 1166-34-3

Formula: C₂₀H₂₄N₂OS

Color and Shape: Solid

Molecular weight: 340.4824

Ref: IN-DA000CV6

Cinanserin

CAS: 1166-34-3

Cinanserin is a serotonin 5-HT2 antagonist.

Formula: C₂₀H₂₄N₂OS

Color and Shape: Solid

Molecular weight: 340.48

Ref: TM-T71350

Cinanserin

Controlled Product

CAS: 1166-34-3

Applications Cinanserin is a serotonin 5-HT2 antagonist.

Formula: C₂₀H₂₄N₂OS

Color and Shape: Neat

Molecular weight: 340.48

Ref: TR-C441903

Cinanserin

CAS: 1166-34-3

Cinanserin is a 5-HT receptor agonist that blocks the effects of serotonin in the central nervous system. It has been shown to have an effect on locomotor activity in vivo and to increase lymphocyte transformation in vitro. Cinanserin also inhibits fatty acid synthesis, which may account for its anti-carcinoid properties, and it has been found to act as a coumarin derivative. This drug binds with high affinity to 5-HT2 receptors, inhibiting viral life by blocking activation of the transcription factor NF-kappaB. Cinanserin also inhibits signal pathways such as MAPK and PI3K/AKT, which are involved in cell proliferation, differentiation, and apoptosis.

Formula: C₂₀H₂₄N₂OS

Purity: Min. 95%

Molecular weight: 340.48 g/mol

Ref: 3D-FC175263