CAS 117374-84-2

carazolol glucuronide

Description:

Carazolol glucuronide is a chemical compound that serves as a metabolite of carazolol, a non-selective beta-adrenergic antagonist. This substance is characterized by the presence of a glucuronic acid moiety, which is typically involved in the detoxification and excretion of various drugs and xenobiotics in the body. The glucuronidation process enhances the solubility of lipophilic compounds, facilitating their elimination. Carazolol glucuronide is generally studied in the context of pharmacokinetics and drug metabolism, particularly in understanding how the body processes beta-blockers. Its structure includes a beta-blocking agent linked to a glucuronic acid, which may influence its biological activity and pharmacological effects. The compound is of interest in clinical research, especially regarding its role in the therapeutic effects and side effects of carazolol. As with many metabolites, the specific characteristics such as solubility, stability, and biological activity can vary based on the conditions under which they are studied.

Formula: C₂₄H₃₀N₂O₈

InChI: InChI=1/C24H30N2O8/c1-4-32-23(12-25-13(2)3)24(31,21(28)19(27)20(34-23)22(29)30)33-17-11-7-10-16-18(17)14-8-5-6-9-15(14)26-16/h5-11,13,19-21,25-28,31H,4,12H2,1-3H3,(H,29,30)/t19-,20+,21+,23-,24+/m1/s1

Synonyms:

• (2S,3S,4S,5S,6R)-5-(9H-carbazol-4-yloxy)-6-ethoxy-3,4,5-trihydroxy-6-[(propan-2-ylamino)methyl]tetrahydro-2H-pyran-2-carboxylic acid (non-preferred name)
• Carazolol glucuronide

(R)-Carazolol Glucuronide

Controlled Product

CAS: 117374-84-2

Formula: C₂₄H₃₀N₂O₈

Color and Shape: Neat

Molecular weight: 474.504

Ref: TR-C176140