Tyrphostin 47, identified by its CAS number 118409-60-2, is a synthetic compound that functions primarily as a selective inhibitor of receptor tyrosine kinases, particularly the epidermal growth factor receptor (EGFR). This compound is part of a broader class of tyrphostins, which are known for their ability to interfere with signal transduction pathways involved in cell proliferation and differentiation. Tyrphostin 47 exhibits characteristics such as moderate solubility in organic solvents and a relatively low molecular weight, which facilitates its use in biological assays. Its mechanism of action involves competitive inhibition, which can lead to the modulation of various cellular processes, making it a valuable tool in cancer research and therapeutic development. Additionally, studies have indicated that tyrphostin 47 may have implications in understanding the role of tyrosine phosphorylation in cellular signaling and its potential effects on tumor growth and metastasis. As with many chemical compounds, proper handling and safety measures should be observed due to its biological activity.

tyrphostin 47

118409-60-2: Tyrphostin 47, identified by its CAS number 118409-60-2, is a synthetic compound that functions primarily as a selective inhibitor of receptor tyrosine kinases, particularly the epidermal growth factor receptor (EGFR). This compound is part of a broader class of tyrphostins, which are known for their ability to interfere with signal transduction pathways involved in cell proliferation and differentiation. Tyrphostin 47 exhibits characteristics such as moderate solubility in organic solvents and a relatively low molecular weight, which facilitates its use in biological assays. Its mechanism of action involves competitive inhibition, which can lead to the modulation of various cellular processes, making it a valuable tool in cancer research and therapeutic development. Additionally, studies have indicated that tyrphostin 47 may have implications in understanding the role of tyrosine phosphorylation in cellular signaling and its potential effects on tumor growth and metastasis. As with many chemical compounds, proper handling and safety measures should be observed due to its biological activity.

<p>Tyrphostin 47 inhibits the protein-tyrosine kinase activity of EGF-R.</p>

CAS 118409-60-2

tyrphostin 47

Tyrphostin 47

Ref: TM-T24908