CAS 1191900-51-2

Brexpiprazole Sulfoxide

CAS: 1191900-51-2

Formula: C₂₅H₂₇N₃O₃S

Molecular weight: 449.57

Ref: ST-EA-CP-B15023

Brexpiprazole S-oxide

CAS: 1191900-51-2

Brexpiprazole S-oxide is the main metabolite of Brexpiprazole, a human 5-HT1A and dopamine receptor partial agonist (Ki: 0.12, 0.3 nM).

Formula: C₂₅H₂₇N₃O₃S

Purity: 98%

Color and Shape: Solid

Molecular weight: 449.57

Ref: TM-T10612

Brexpiprazole Sulfoxide

CAS: 1191900-51-2

Formula: C₂₅H₂₇N₃O₃S

Molecular weight: 449.57

Ref: 4Z-B-115022

Brexpiprazole S-Oxide

CAS: 1191900-51-2

Applications Brexpiprazole S-Oxide is an impurity and potential metabolite of Brexpiprazole (B677385), a drug candidate useful in treatment and prevention of mental disorders including CNS disorders.
References Yamashita, H., et al.: PCT Int. Appl., WO 2006112464 A1 20061026 (2006);

Formula: C₂₅H₂₇N₃O₃S

Color and Shape: Neat

Molecular weight: 449.565

Ref: TR-B677420

Brexpiprazole S-oxide

CAS: 1191900-51-2

Brexpiprazole S-oxide is a high purity peptide that inhibits the activity of the dopamine D2 receptor. Brexpiprazole S-oxide is an inhibitor of protein interactions and can be used as a research tool to study the function of various proteins in cells. Brexpiprazole S-oxide is also an activator of ligands and receptors, which means it can be used to identify new drugs or drug targets. Brexpiprazole S-oxide has been shown to be a high affinity ligand for the dopamine D2 receptor, with no binding to other receptors, such as serotonin 5HT2A and muscarinic M3 receptors.

Formula: C₂₅H₂₇N₃O₃S

Purity: Min. 95%

Molecular weight: 449.6 g/mol

Ref: 3D-RXB90051