CAS 1202916-90-2
:CX-6258
Description:
CX-6258, identified by its CAS number 1202916-90-2, is a chemical compound that has garnered attention in pharmaceutical research, particularly in the context of cancer treatment. It is classified as a small molecule inhibitor, specifically targeting certain pathways involved in tumor growth and proliferation. The compound exhibits a unique mechanism of action, which may involve the modulation of specific protein interactions or enzymatic activities critical to cancer cell survival. CX-6258 has been evaluated in preclinical studies for its efficacy and safety profile, showing potential in inhibiting the growth of various cancer cell lines. Its solubility, stability, and bioavailability are important characteristics that influence its therapeutic application. As with many investigational drugs, ongoing research is essential to fully understand its pharmacokinetics, pharmacodynamics, and potential side effects. Overall, CX-6258 represents a promising candidate in the ongoing search for effective cancer therapies, although further clinical trials are necessary to establish its clinical utility.
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Found 5 products.
CX6258
CAS:<p>CX6258 is a kinase inhibitor that selectively inhibits the serine/threonine kinase pim-1, which is involved in the induction of apoptosis. CX6258 has potent antitumor activity and minimal toxicity. It has been shown to inhibit prostate cancer cells in vitro and in vivo. This agent also inhibits epidermal growth factor receptor, thereby preventing cell proliferation. CX6258 binds to the ATP-binding site on the ribosome and prevents protein synthesis by inhibiting the binding of aminoacyl-tRNA to the ribosome. This drug also has potent structural similarity to one of its targets, Pim-1.</p>Formula:C26H24ClN3O3Purity:Min. 95%Molecular weight:461.94 g/molCX-6258
CAS:CX-6258 is an orally valid Pim 1/2/3 kinase(IC50=5 nM/25 nM/16 nM) inhibitor. It has good biological activity and kinase specificity.Formula:C26H24ClN3O3Purity:97.46%Color and Shape:SolidMolecular weight:461.94
