CAS 120656-74-8
:Trefentanil
Description:
Trefentanil is a synthetic opioid analgesic that is structurally related to fentanyl, designed for use in veterinary medicine, particularly for sedation and analgesia in animals. It is characterized by its high potency, being significantly more potent than morphine, which makes it effective in managing pain but also raises concerns regarding potential for misuse and overdose. Trefentanil acts primarily on the mu-opioid receptors in the central nervous system, leading to its analgesic effects. Its pharmacokinetics include rapid onset and a relatively short duration of action, necessitating careful dosing and monitoring. Due to its potency, it is typically administered in microgram quantities, often via injection. Safety precautions are essential when handling trefentanil, as accidental exposure can lead to severe respiratory depression and other opioid-related effects. As with other opioids, the potential for dependence and abuse exists, making it crucial for veterinary professionals to adhere to strict guidelines when using this substance.
Formula:C25H31FN6O2
InChI:InChI=1S/C25H31FN6O2/c1-3-23(33)32(22-13-9-8-12-21(22)26)25(20-10-6-5-7-11-20)14-16-29(17-15-25)18-19-31-24(34)30(4-2)27-28-31/h5-13H,3-4,14-19H2,1-2H3
InChI key:InChIKey=RJSCINHYBGMIFT-UHFFFAOYSA-N
SMILES:N(C(CC)=O)(C1(CCN(CCN2C(=O)N(CC)N=N2)CC1)C3=CC=CC=C3)C4=C(F)C=CC=C4
Synonyms:- A 2665
- Propanamide, N-[1-[2-(4-ethyl-4,5-dihydro-5-oxo-1H-tetrazol-1-yl)ethyl]-4-phenyl-4-piperidinyl]-N-(2-fluorophenyl)-
- Trefentanil
- N-[1-[2-(4-Ethyl-4,5-dihydro-5-oxo-1H-tetrazol-1-yl)ethyl]-4-phenyl-4-piperidinyl]-N-(2-fluorophenyl)propanamide
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Found 2 products.
N-[1-[2-(4-Ethyl-5-Oxotetrazol-1-Yl)Ethyl]-4-Phenylpiperidin-4-Yl]-N-(2-Fluorophenyl)Propanamide
CAS:Controlled Product<p>N-[1-[2-(4-Ethyl-5-Oxotetrazol-1-Yl)Ethyl]-4-Phenylpiperidin-4-Yl]-N-(2-Fluorophenyl)Propanamide is a drug that is used clinically for the treatment of depression. It is an analog of amitriptyline, an antidepressant and a tricyclic compound. N-[1-[2-(4-Ethyl-5-Oxotetrazol-1-Yl)Ethyl]-4-Phenylpiperidin-4-Yl]-N-(2-Fluorophenyl)Propanamide has been shown to increase the concentration of plasma drug levels by increasing transporter gene expression in muscle tissue. This drug also has clinical pharmacology and thermal expansion properties.</p>Formula:C25H31FN6O2Purity:Min. 95%Molecular weight:466.55 g/mol

