CAS 1213781-59-9

Varenicline Acetamide (1-(6,7,9,10-tetrahydro-8H-6,10-methanoazepino[4,5-g]quinoxalin-8-yl)ethan-1-one)

CAS: 1213781-59-9

Heterocyclic compounds with nitrogen hetero-atom(s) only, aromatic or modified aromatic, nesoi

Formula: C₁₅H₁₅N₃O

Color and Shape: Yellow Solid

Molecular weight: 253.12151

Ref: 45-1A03370

N-Acetyl Varenicline

CAS: 1213781-59-9

Formula: C₁₅H₁₅N₃O

Color and Shape: Yellow Solid

Molecular weight: 253.31

Ref: 4Z-V-2521

1-(6,7,9,10-Tetrahydro-6,10-methano-8H-pyrazino[2,3-h][3]benzazepin-8-yl)ethanone

Controlled Product

CAS: 1213781-59-9

Applications 1-(6,7,9,10-Tetrahydro-6,10-methano-8H-pyrazino[2,3-h][3]benzazepin-8-yl)ethanone is related to its parent compound N-Formyl Varenicline (F701650), which is a metabolite of Varenicline and metabolite M5. Also, it is derived from Varenicline Tartrate (V098490), which is a nicotinic α4β2 acetylcholine receptor partial agonist and used to aid in smoking cessation (1,2,3,4).
References Dow, J., et al.: Drug Metab. Dispos., 22, 738 (1994), Toide, K., et al.: Biochem. Pharmacol., 67, 1269 (2004), Coe, J., et al.: J. Med. Chem., 48, 3474 (2005), Doll, R., et al.: Br. J. Cancer, 92, 426 (2005)

Formula: C₁₅H₁₅N₃O

Color and Shape: Neat

Molecular weight: 253.299

Ref: TR-T310085

N-Acetyl Varenicline

CAS: 1213781-59-9

Formula: C₁₅H₁₅N₃O

Molecular weight: 253.31

Ref: ST-EA-CP-V8025