CAS 1216984-85-8

Rizatriptan-d6 Benzoate

Description:

Rizatriptan-d6 benzoate is a deuterated derivative of rizatriptan, a medication primarily used to treat migraines. The "d6" designation indicates that the compound contains six deuterium atoms, which are isotopes of hydrogen, replacing the regular hydrogen atoms in the molecular structure. This modification is often employed in research to enhance the stability and detectability of the compound in analytical studies, such as mass spectrometry. Rizatriptan itself is a selective agonist for serotonin receptors, particularly the 5-HT_1B and 5-HT_1D subtypes, which play a crucial role in the vasoconstriction of cranial blood vessels and the inhibition of pro-inflammatory neuropeptide release. The benzoate moiety suggests that the compound is in a salt form, which can influence its solubility and pharmacokinetic properties. Overall, rizatriptan-d6 benzoate serves as a valuable tool in pharmacological research, particularly in studies involving drug metabolism and receptor binding assays.

Formula: C₂₂H₂₄N₅O₂

Synonyms:

• N,N-Dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-indole-3-ethanamine-d6 Benzoate
• Rizatriptan-d6 Benzoate
• MK-462-d6
• Maxalt-d6
• MK-0462-d6
• N,N-(DiMethyl-d6)-5-(1H-1,2,4-triazol-1-ylMethyl)-1H-indole-3-ethanaMine Benzoate

Rizatriptan-d6 Benzoate

CAS: 1216984-85-8

Formula: C₁₅H₁₃D₆N₅·C₇H₆O₂

Color and Shape: White To Off-White Solid

Molecular weight: 275.39 122.12

Ref: 4Z-R-121

Rizatriptan EP Impurity B Chloride

CAS: 1216984-85-8, 606927-07-5

Formula: C₂₈H₃₂N₉·Cl

Color and Shape: White To Off-White Solid

Molecular weight: 494.63 35.45

Ref: 4Z-R-1212

Rizatriptan-d6 Benzoate

Controlled Product

CAS: 1216984-85-8

Formula: C₂₂H₁₉D₆N₅O₂

Color and Shape: Neat

Molecular weight: 397.5

Ref: TR-R545002