CAS 123040-96-0

2H-1,4-Benzoxazine-8-carboxamide,N-1-azabicyclo[2.2.2]oct-3-yl-6-chloro-3,4-dihydro-4-methyl-3-oxo-,monohydrochloride, (-)- (9CI)

Description:

2H-1,4-Benzoxazine-8-carboxamide, N-1-azabicyclo[2.2.2]oct-3-yl-6-chloro-3,4-dihydro-4-methyl-3-oxo-, monohydrochloride, (-)- (9CI) is a complex organic compound characterized by its unique bicyclic structure and functional groups. This substance features a benzoxazine ring, which contributes to its potential biological activity, and an azabicyclo structure that may influence its pharmacological properties. The presence of a carboxamide group suggests potential for hydrogen bonding, which can enhance solubility and interaction with biological targets. The chloro and methyl substituents on the bicyclic framework may affect its reactivity and stability. As a hydrochloride salt, it is likely to exhibit improved solubility in aqueous environments, making it suitable for various applications, including medicinal chemistry. The (-) designation indicates that it is the enantiomer with specific stereochemical properties, which can be crucial for its biological activity. Overall, this compound's intricate structure and functional groups suggest potential utility in pharmaceutical research and development.

Formula: C₁₇H₂₀ClN₃O₃ClH

Synonyms:

• 2H-1,4-Benzoxazine-8-carboxamide, N-1-azabicyclo[2.2.2]oct-3-yl-6-chloro-3,4-dihydro-4-methyl-3-oxo-, monohydrochloride, (-)-

(-)-Azasetron hydrochloride

CAS: 123040-96-0

(-)-Azasetron hydrochloride is a potent antiemetic pharmaceutical agent, which is chemically synthesized through organic synthesis processes. It functions as a selective serotonin 5-HT3 receptor antagonist. The mode of action of (-)-Azasetron hydrochloride involves the competitive inhibition of serotonin binding to the 5-HT3 receptors located in the central and peripheral nervous systems. By blocking these pathways, it effectively mitigates the emetic signaling induced by chemotherapeutic agents or surgical procedures.

Formula: C₉H₇NO₂

Purity: Min. 95%

Molecular weight: 161.16 g/mol

Ref: 3D-YEA04096