CAS 1236199-60-2

1H-Benzimidazole-2-heptanamide, 5-[bis(2-chloroethyl)amino]-N-hydroxy-1-methyl-

CAS: 1236199-60-2

Formula: C₁₉H₂₈Cl₂N₄O₂

Purity: 99%

Color and Shape: Solid

Molecular weight: 415.3572

Ref: IN-DA000KV6

EDO-S101

CAS: 1236199-60-2

EDO-S101

Purity: ≥98%

Molecular weight: 415.36g/mol

Ref: 54-BUP02383

EDO-S101

CAS: 1236199-60-2

EDO-S101 (Tinostamustine) is a pan HDAC inhibitor with IC50 values of 9, 9 and 25 nM for HDAC1, HDAC2 and HDAC3 , respectively.

Formula: C₁₉H₂₈Cl₂N₄O₂

Purity: 98.02% - 99.44%

Color and Shape: Solid

Molecular weight: 415.36

Ref: TM-T3516

EDO-S101

CAS: 1236199-60-2

EDO-S101 is a molecule that binds to the ubiquitin-proteasome pathway and inhibits the function of effector proteins, such as caspases. It has been shown to have anticancer properties in animal models. This drug also inhibits the mitochondrial membrane potential, protein synthesis, and protein transport in cell cultures. EDO-S101 has also been shown to induce pro-apoptotic activity and inhibit histone deacetylase activity in vitro. Clinical trials are currently underway to study the effects of this drug on solid tumours.

Formula: C₁₉H₂₈Cl₂O₂

Purity: Min. 95%

Molecular weight: 359.33 g/mol

Ref: 3D-BE170657