CAS 124423-84-3

Panadiplon

Description:

Panadiplon is a chemical compound that belongs to the class of non-benzodiazepine anxiolytics, primarily developed for the treatment of anxiety and sleep disorders. It acts as a selective modulator of the GABA-A receptor, which is a key player in the central nervous system's inhibitory neurotransmission. This compound is characterized by its rapid onset of action and relatively short half-life, making it suitable for acute anxiety relief without the prolonged sedation associated with some traditional anxiolytics. Panadiplon exhibits a favorable side effect profile, with a lower risk of dependence compared to benzodiazepines. Its pharmacological properties include anxiolytic, sedative, and muscle relaxant effects, which are beneficial in managing anxiety-related conditions. Additionally, research has indicated that Panadiplon may have a unique mechanism of action that differentiates it from other anxiolytics, potentially leading to fewer cognitive impairments. However, as with any pharmacological agent, its use should be carefully monitored to mitigate any adverse effects or interactions with other medications.

Formula: C₁₈H₁₇N₅O₂

InChI: InChI=1S/C18H17N5O2/c1-10(2)23-13-6-4-3-5-12(13)22-9-19-14(15(22)18(23)24)16-20-17(25-21-16)11-7-8-11/h3-6,9-11H,7-8H2,1-2H3

InChI key: InChIKey=ZGEGOFCLSWVVKG-UHFFFAOYSA-N

SMILES: O=C1C=2N(C=3C(N1C(C)C)=CC=CC3)C=NC2C=4N=C(ON4)C5CC5

Synonyms:

• Panadiplonum
• U 78875
• FG 10571
• Panadiplon [USAN:INN]
• FG 10571
• Panadiplone
• Panadiplonum [INN-Latin]
• 3-(5-Cyclopropyl-1,2,4-oxadiazol-3-yl)-5-isopropylimidazo(1,5-a)quinoxalin-4(5H)-one
• Panadiplon
• Panadiplone [INN-French]
• U 78875
• 3-(5-Cyclopropyl-1,2,4-oxadiazol-3-yl)-5-(1-methylethyl)imidazo[1,5-a]quinoxalin-4(5H)-one
• UNII-V4PW0S7ZP7
• Imidazo[1,5-a]quinoxalin-4(5H)-one, 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5-(1-methylethyl)-
• 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5-(1-methylethyl)imidazo[1,5-a]quinoxalin-4(5H)-one

Imidazo[1,5-a]quinoxalin-4(5H)-one, 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5-(1-methylethyl)-

CAS: 124423-84-3

Formula: C₁₈H₁₇N₅O₂

Purity: 95%

Molecular weight: 335.3599

Ref: IN-DA000LZ1

Panadiplon

CAS: 124423-84-3

Panadiplon

Purity: ≥98%

Molecular weight: 335.36g/mol

Ref: 54-BUP00949

Panadiplon

CAS: 124423-84-3

Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of

Formula: C₁₈H₁₇N₅O₂

Purity: 98.30% - 98.94%

Color and Shape: Solid

Molecular weight: 335.36

Ref: TM-T28294