CAS 124937-51-5: Tolterodine

Description: Tolterodine is a pharmaceutical compound primarily used as an antimuscarinic agent for the treatment of overactive bladder. It functions by selectively blocking muscarinic receptors, which helps reduce involuntary bladder contractions and urinary urgency. The chemical formula of tolterodine is C19H25N, and it has a molecular weight of approximately 281.42 g/mol. This substance is typically administered in the form of its tartrate salt, which enhances its solubility and bioavailability. Tolterodine is characterized by its moderate lipophilicity, allowing it to cross biological membranes effectively. It exhibits a relatively long half-life, which supports once-daily dosing in clinical settings. Common side effects may include dry mouth, constipation, and dizziness, reflecting its anticholinergic properties. Due to its mechanism of action, tolterodine is contraindicated in patients with certain conditions, such as narrow-angle glaucoma or urinary retention. Overall, tolterodine represents a significant advancement in the management of urinary disorders, providing symptomatic relief for patients with overactive bladder syndrome.

Formula: C₂₂H₃₂ClNO

InChI: InChI=1/C22H31NO.ClH/c1-16(2)23(17(3)4)14-13-20(19-9-7-6-8-10-19)21-15-18(5)11-12-22(21)24;/h6-12,15-17,20,24H,13-14H2,1-5H3;1H

InChI key: InChIKey=OOGJQPCLVADCPB-HXUWFJFHSA-N

SMILES: OC1=CC=C(C=C1C(C=2C=CC=CC2)CCN(C(C)C)C(C)C)C

Synonyms:

• 124937-51-5
• 2-[3-(dipropan-2-ylamino)-1-phenylpropyl]-4-methylphenol
• 2-[(1R)-3-(dipropan-2-ylamino)-1-phenylpropyl]-4-methylphenol 2,3-dihydroxybutanedioate (1:1)
• phenol, 2-[3-[bis(1-methylethyl)amino]-1-phenylpropyl]-4-methyl-
• 2-{3-[bis(1-methylethyl)amino]-1-phenylpropyl}-4-methylphenol
• 2-[(1S)-3-(dipropan-2-ylamino)-1-phenylpropyl]-4-methylphenol
• 2-[3-(diisopropylamino)-1-phenyl-propyl]-4-methyl-phenol hydrochloride

Phenol, 2-[(1R)-3-[bis(1-methylethyl)amino]-1-phenylpropyl]-4-methyl-

CAS: 124937-51-5

• Formula: C₂₂H₃₁NO
• Purity: 99%
• Color and Shape: Solid
• Molecular weight: 325.4876

Tolterodine

CAS: 124937-51-5

• Purity: 99.7%
• Molecular weight: 325.49g/mol

Tolterodine Tartrate

CAS: 124937-51-5124937-52-6

• Formula: C₂₂H₃₁NO·C₄H₆O₆
• Color and Shape: White To Off-White Solid
• Molecular weight: 325.50 150.09

Tolterodine

CAS: 124937-51-5

Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive …

• Formula: C₂₂H₃₁NO
• Purity: 99.71%
• Color and Shape: White Like Or Light Brown Crystalline Powder
• Molecular weight: 325.49

R-(+)-Tolterodine

CAS: 124937-51-5

Tolterodine is a drug that acts as a selective antagonist at the muscarinic receptor M3. …

• Formula: C₂₂H₃₁NO
• Purity: Min. 95%
• Molecular weight: 325.49 g/mol