CAS 1254730-81-8

4-[8-[(2,6-Diethoxy-4′-fluoro[1,1′-biphenyl]-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]dec-2-yl]benzoic acid

CAS: 1254730-81-8

4-[8-[(2,6-Diethoxy-4′-fluoro[1,1′-biphenyl]-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]dec-2-yl]benzoic acid is a potent and selective inhibitor of the ion channel TRPV1. It blocks the activation of TRPV1 channels by capsaicin, thereby preventing the transmission of pain signals to the brain. 4-[8-[(2,6-Diethoxy-4′-fluoro[1,1′-biphenyl]-4-yl)methyl]-3-oxo-2,8-- diazaspiro[4.5]decan]-2 yl]benzoic acid has been shown to inhibit peptide binding to the receptor GPCR in a ligand displacement assay. This compound also inhibits protein interactions with their partners and is

Formula: C₃₂H₃₅FN₂O₅

Purity: Min. 95%

Color and Shape: Powder

Molecular weight: 546.6 g/mol

Ref: 3D-EAC73081

SSTR5 antagonist 2

CAS: 1254730-81-8

SSTR5 antagonist 2: potent, orally active, selective SSTR5 inhibitor, may treat Type 2 diabetes.

Formula: C₃₂H₃₅FN₂O₅

Purity: 98%

Color and Shape: Solid

Molecular weight: 546.63

Ref: TM-T13022