CAS 125697-92-9

Lavendustin A

Description:

Lavendustin A is a natural compound that belongs to the class of indole alkaloids, primarily derived from the plant Lavandula. It is recognized for its potential biological activities, particularly its role as a selective inhibitor of certain protein kinases, which are crucial in various cellular processes, including cell growth and division. The compound exhibits a complex molecular structure characterized by multiple rings and functional groups, contributing to its unique chemical properties. Lavendustin A has garnered interest in medicinal chemistry due to its potential therapeutic applications, particularly in cancer treatment, as it may interfere with the signaling pathways that promote tumor growth. Additionally, it has been studied for its effects on other biological systems, showcasing a range of pharmacological activities. Its solubility and stability in various solvents make it a subject of interest for further research in drug development and pharmacology. Overall, Lavendustin A represents a significant area of study in the quest for novel therapeutic agents.

Formula: C₂₁H₁₉NO₆

InChI: InChI=1S/C21H19NO6/c23-16-6-8-19(25)14(9-16)12-22(11-13-3-1-2-4-18(13)24)15-5-7-20(26)17(10-15)21(27)28/h1-10,23-26H,11-12H2,(H,27,28)

InChI key: InChIKey=ULTTYPMRMMDONC-UHFFFAOYSA-N

SMILES: N(CC1=C(O)C=CC(O)=C1)(CC2=C(O)C=CC=C2)C3=CC(C(O)=O)=C(O)C=C3

Synonyms:

• 5-Amino-[(N-2,5-Dihydroxybenzyl)-N'-2-Hydroxybenzyl]Salicylic Acid
• 5-[(2,5-Dihydroxybenzyl)(2-Hydroxybenzyl)Amino]-2-Hydroxybenzoate
• 5-[(2,5-Dihydroxybenzyl)(2-Hydroxybenzyl)Amino]-2-Hydroxybenzoic Acid
• 5-[[(2,5-Dihydroxyphenyl)Methyl][(2-Hydroxyphenyl)Methyl]Amino]-2-Hydroxybenzoic Acid
• Benzoic acid, 5-[[(2,5-dihydroxyphenyl)methyl][(2-hydroxyphenyl)methyl]amino]-2-hydroxy-
• NSC 678027
• Rg14355
• Lavendustin A

Benzoic acid, 5-[[(2,5-dihydroxyphenyl)methyl][(2-hydroxyphenyl)methyl]amino]-2-hydroxy-

CAS: 125697-92-9

Formula: C₂₁H₁₉NO₆

Purity: 95%

Color and Shape: Solid

Molecular weight: 381.3787

Ref: IN-DA000OIB

Lavendustin A

Controlled Product

CAS: 125697-92-9

Applications A potent tyrosine kinase inhibitor. Inhibition is competitive with ATP and is noncompetitive with the peptide.
References Onoda, T., et al.: Journal of Natural Products, 52, 6, 1252 (1989)

Formula: C₂₁H₁₉NO₆

Color and Shape: Neat

Molecular weight: 381.38

Ref: TR-L215000

lavendustin A

CAS: 125697-92-9

lavendustin A (RG-14355) is a potent, cell-permeable inhibitor of epidermal growth factor receptor (EGFR) tyrosine kinase.

Formula: C₂₁H₁₉NO₆

Purity: 98%

Color and Shape: Off-White Solid

Molecular weight: 381.38

Ref: TM-T4183

Lavendustin A

CAS: 125697-92-9

Lavendustin A is a potent tyrosine kinase inhibitor, which is derived from marine sponge sources. It functions by specifically targeting and inhibiting the activity of tyrosine kinases, enzymes crucial for the phosphorylation of tyrosine residues on protein substrates, thereby interfering with signaling pathways essential for various cellular processes.

Formula: C₂₁H₁₉NO₆

Purity: Min. 95%

Molecular weight: 381.38 g/mol

Ref: 3D-FL24861